U01 MH087965/MH/NIMH NIH HHS/United States[Grants and Funding] - Search Results

Year	Number of Results
2011	3
2012	13
2013	10
2014	6
2015	6
2016	7
2017	11
2018	6
2019	5
2020	3
2021	1
2024	2
2025	0

1

Practical Strategies and Concepts in GPCR Allosteric Modulator Discovery: Recent Advances with Metabotropic Glutamate Receptors.

Lindsley CW, Emmitte KA, Hopkins CR, Bridges TM, Gregory KJ, Niswender CM, Conn PJ. Lindsley CW, et al. Chem Rev. 2016 Jun 8;116(11):6707-41. doi: 10.1021/acs.chemrev.5b00656. Epub 2016 Feb 16. Chem Rev. 2016. PMID: 26882314 Free PMC article. Review.

2

Allosteric modulators for the treatment of schizophrenia: targeting glutamatergic networks.

Menniti FS, Lindsley CW, Conn PJ, Pandit J, Zagouras P, Volkmann RA. Menniti FS, et al. Curr Top Med Chem. 2013;13(1):26-54. doi: 10.2174/1568026611313010005. Curr Top Med Chem. 2013. PMID: 23409764 Free PMC article. Review.

3

Discovery of VU6016235: A Highly Selective, Orally Bioavailable, and Structurally Distinct Tricyclic M₄ Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM).

Engers JL, Baker LA, Chang S, Luscombe VB, Rodriguez AL, Niswender CM, Cho HP, Bubser M, Gray AT, Jones CK, Peng W, Rook JM, Bridges TM, Boutaud O, Conn PJ, Engers DW, Lindsley CW, Temple KJ. Engers JL, et al. ACS Chem Neurosci. 2024 Sep 24;15(20):3744-54. doi: 10.1021/acschemneuro.4c00465. Online ahead of print. ACS Chem Neurosci. 2024. PMID: 39316465 Free PMC article.

4

Modulation of arousal and sleep/wake architecture by M₁ PAM VU0453595 across young and aged rodents and nonhuman primates.

Gould RW, Russell JK, Nedelcovych MT, Bubser M, Blobaum AL, Bridges TM, Newhouse PA, Lindsley CW, Conn PJ, Nader MA, Jones CK. Gould RW, et al. Neuropsychopharmacology. 2020 Dec;45(13):2219-2228. doi: 10.1038/s41386-020-00812-7. Epub 2020 Aug 31. Neuropsychopharmacology. 2020. PMID: 32868847 Free PMC article.

5

Emerging approaches for treatment of schizophrenia: modulation of cholinergic signaling.

Foster DJ, Jones CK, Conn PJ. Foster DJ, et al. Discov Med. 2012 Dec;14(79):413-20. Discov Med. 2012. PMID: 23272693 Free PMC article. Review.

6

Development of allosteric modulators of GPCRs for treatment of CNS disorders.

Nickols HH, Conn PJ. Nickols HH, et al. Neurobiol Dis. 2014 Jan;61:55-71. doi: 10.1016/j.nbd.2013.09.013. Epub 2013 Sep 27. Neurobiol Dis. 2014. PMID: 24076101 Free PMC article. Review.

7

Allosteric modulation of Class C GPCRs: a novel approach for the treatment of CNS disorders.

Engers DW, Lindsley CW. Engers DW, et al. Drug Discov Today Technol. 2013 Summer;10(2):e269-76. doi: 10.1016/j.ddtec.2012.10.007. Drug Discov Today Technol. 2013. PMID: 24050278 Free PMC article. Review.

8

Emerging approaches for treatment of schizophrenia: modulation of glutamatergic signaling.

Noetzel MJ, Jones CK, Conn PJ. Noetzel MJ, et al. Discov Med. 2012 Nov;14(78):335-43. Discov Med. 2012. PMID: 23200065 Free PMC article. Review.

9

Discovery of a novel 2,3-dimethylimidazo[1,2-a]pyrazine-6-carboxamide M₄ positive allosteric modulator (PAM) chemotype.

Temple KJ, Engers JL, Long MF, Watson KJ, Chang S, Luscombe VB, Jenkins MT, Rodriguez AL, Niswender CM, Bridges TM, Conn PJ, Engers DW, Lindsley CW. Temple KJ, et al. Bioorg Med Chem Lett. 2020 Feb 1;30(3):126812. doi: 10.1016/j.bmcl.2019.126812. Epub 2019 Nov 13. Bioorg Med Chem Lett. 2020. PMID: 31784320

10

Anticholinergic drugs rescue synaptic plasticity in DYT1 dystonia: role of M1 muscarinic receptors.

Maltese M, Martella G, Madeo G, Fagiolo I, Tassone A, Ponterio G, Sciamanna G, Burbaud P, Conn PJ, Bonsi P, Pisani A. Maltese M, et al. Mov Disord. 2014 Nov;29(13):1655-65. doi: 10.1002/mds.26009. Epub 2014 Sep 4. Mov Disord. 2014. PMID: 25195914 Free PMC article.

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