R01 AI028731/AI/NIAID NIH HHS/United States[Grants and Funding] - Search Results

Year	Number of Results
1999	1
2007	1
2013	2
2014	2
2015	2
2016	5
2017	2
2018	2
2025	0

1

CCR5 receptor antagonists in preclinical to phase II clinical development for treatment of HIV.

Kim MB, Giesler KE, Tahirovic YA, Truax VM, Liotta DC, Wilson LJ. Kim MB, et al. Expert Opin Investig Drugs. 2016 Dec;25(12):1377-1392. doi: 10.1080/13543784.2016.1254615. Expert Opin Investig Drugs. 2016. PMID: 27791451 Free PMC article. Review.

2

Discovery of novel N-aryl piperazine CXCR4 antagonists.

Zhao H, Prosser AR, Liotta DC, Wilson LJ. Zhao H, et al. Bioorg Med Chem Lett. 2015 Nov 1;25(21):4950-4955. doi: 10.1016/j.bmcl.2015.04.036. Epub 2015 Apr 17. Bioorg Med Chem Lett. 2015. PMID: 25935642 Free PMC article.

3

Discovery of Tetrahydroisoquinoline-Containing CXCR4 Antagonists with Improved in Vitro ADMET Properties.

Miller EJ, Jecs E, Truax VM, Katzman BM, Tahirovic YA, Wilson RJ, Kuo KM, Kim MB, Nguyen HH, Saindane MT, Zhao H, Wang T, Sum CS, Cvijic ME, Schroeder GM, Wilson LJ, Liotta DC. Miller EJ, et al. J Med Chem. 2018 Feb 8;61(3):946-979. doi: 10.1021/acs.jmedchem.7b01420. Epub 2018 Jan 30. J Med Chem. 2018. PMID: 29350534

4

Discovery of tetrahydroisoquinoline-based CXCR4 antagonists.

Truax VM, Zhao H, Katzman BM, Prosser AR, Alcaraz AA, Saindane MT, Howard RB, Culver D, Arrendale RF, Gruddanti PR, Evers TJ, Natchus MG, Snyder JP, Liotta DC, Wilson LJ. Truax VM, et al. ACS Med Chem Lett. 2013 Sep 5;4(11):1025-30. doi: 10.1021/ml400183q. eCollection 2013 Nov 14. ACS Med Chem Lett. 2013. PMID: 24936240 Free PMC article.

5

Discovery and Development of the Anti-Human Immunodeficiency Virus Drug, Emtricitabine (Emtriva, FTC).

Liotta DC, Painter GR. Liotta DC, et al. Acc Chem Res. 2016;49(10):2091-2098. doi: 10.1021/acs.accounts.6b00274. Epub 2016 Oct 5. Acc Chem Res. 2016. PMID: 27704821 Free PMC article.

6

Synthesis and SAR of 1,2,3,4-Tetrahydroisoquinoline-Based CXCR4 Antagonists.

Wilson RJ, Jecs E, Miller EJ, Nguyen HH, Tahirovic YA, Truax VM, Kim MB, Kuo KM, Wang T, Sum CS, Cvijic ME, Paiva AA, Schroeder GM, Wilson LJ, Liotta DC. Wilson RJ, et al. ACS Med Chem Lett. 2017 Dec 8;9(1):17-22. doi: 10.1021/acsmedchemlett.7b00381. eCollection 2018 Jan 11. ACS Med Chem Lett. 2017. PMID: 29348805 Free PMC article.

7

Reduction Sensitive Lipid Conjugates of Tenofovir: Synthesis, Stability, and Antiviral Activity.

Giesler KE, Marengo J, Liotta DC. Giesler KE, et al. J Med Chem. 2016 Aug 11;59(15):7097-110. doi: 10.1021/acs.jmedchem.6b00428. Epub 2016 Jul 22. J Med Chem. 2016. PMID: 27405794 Free PMC article.

8

Structure-activity relationships and pharmacophore model of a noncompetitive pyrazoline containing class of GluN2C/GluN2D selective antagonists.

Acker TM, Khatri A, Vance KM, Slabber C, Bacsa J, Snyder JP, Traynelis SF, Liotta DC. Acker TM, et al. J Med Chem. 2013 Aug 22;56(16):6434-56. doi: 10.1021/jm400652r. Epub 2013 Aug 2. J Med Chem. 2013. PMID: 23909910 Free PMC article.

9

Next-Generation Reduction Sensitive Lipid Conjugates of Tenofovir: Antiviral Activity and Mechanism of Release.

Giesler KE, Liotta DC. Giesler KE, et al. J Med Chem. 2016 Nov 23;59(22):10244-10252. doi: 10.1021/acs.jmedchem.6b01292. Epub 2016 Nov 2. J Med Chem. 2016. PMID: 27933889 Free PMC article.

10

Pyrazolo-Piperidines Exhibit Dual Inhibition of CCR5/CXCR4 HIV Entry and Reverse Transcriptase.

Cox BD, Prosser AR, Sun Y, Li Z, Lee S, Huang MB, Bond VC, Snyder JP, Krystal M, Wilson LJ, Liotta DC. Cox BD, et al. ACS Med Chem Lett. 2015 May 6;6(7):753-7. doi: 10.1021/acsmedchemlett.5b00036. eCollection 2015 Jul 9. ACS Med Chem Lett. 2015. PMID: 26191361 Free PMC article.

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