Jetter JW - Search Results

1

Structure-activity relationships (SAR) of some tetracyclic heterocycles related to the immunosuppressive agent Brequinar Sodium.

Pitts WJ, Jetter JW, Pinto DJ, Orwat MJ, Batt DG, Sherk SR, Petraitis JJ, Jacobson IC, Copeland RA, Dowling RL, Jaffee BD, Gardner TL, Jones EA, Magolda RL. Pitts WJ, et al. Among authors: jetter jw. Bioorg Med Chem Lett. 1998 Feb 3;8(3):307-12. doi: 10.1016/s0960-894x(98)00010-9. Bioorg Med Chem Lett. 1998. PMID: 9871675

2

Terphenyl cyclooxygenase-2 (COX-2) inhibitors: optimization of the central ring and o-biphenyl analogs.

Pinto DJ, Batt DG, Pitts WJ, Petraitis JJ, Orwat MJ, Wang S, Jetter JW, Sherk SR, Houghton GC, Copeland RA, Covington MB, Trzaskos JM, Magolda RL. Pinto DJ, et al. Among authors: jetter jw. Bioorg Med Chem Lett. 1999 Apr 5;9(7):919-24. doi: 10.1016/s0960-894x(99)00105-5. Bioorg Med Chem Lett. 1999. PMID: 10230611

3

Isoxazolines as potent antagonists of the integrin alpha(v)beta(3).

Pitts WJ, Wityak J, Smallheer JM, Tobin AE, Jetter JW, Buynitsky JS, Harlow PP, Solomon KA, Corjay MH, Mousa SA, Wexler RR, Jadhav PK. Pitts WJ, et al. Among authors: jetter jw. J Med Chem. 2000 Jan 13;43(1):27-40. doi: 10.1021/jm9900321. J Med Chem. 2000. PMID: 10633036

4

Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): an orally active antagonist of the gonadotropin releasing hormone receptor (GnRH-R).

Pelletier JC, Chengalvala MV, Cottom JE, Feingold IB, Green DM, Hauze DB, Huselton CA, Jetter JW, Kopf GS, Lundquist JT, Magolda RL, Mann CW, Mehlmann JF, Rogers JF, Shanno LK, Adams WR, Tio CO, Wrobel JE. Pelletier JC, et al. Among authors: jetter jw. J Med Chem. 2009 Apr 9;52(7):2148-52. doi: 10.1021/jm801572m. J Med Chem. 2009. PMID: 19271735

5

Synthesis and SAR of 2-carboxylic acid indoles as inhibitors of plasminogen activator inhibitor-1.

Hu B, Jetter JW, Wrobel JE, Antrilli TM, Bauer JS, Di L, Polakowski S, Jain U, Crandall DL. Hu B, et al. Among authors: jetter jw. Bioorg Med Chem Lett. 2005 Aug 1;15(15):3514-8. doi: 10.1016/j.bmcl.2005.05.095. Bioorg Med Chem Lett. 2005. PMID: 15982877

6

Synthesis of (bis)sulfonic acid, (bis)benzamides as follicle-stimulating hormone (FSH) antagonists.

Wrobel J, Green D, Jetter J, Kao W, Rogers J, Pérez MC, Hardenburg J, Deecher DC, López FJ, Arey BJ, Shen ES. Wrobel J, et al. Bioorg Med Chem. 2002 Mar;10(3):639-56. doi: 10.1016/s0968-0896(01)00324-8. Bioorg Med Chem. 2002. PMID: 11814852

7

2-phenyl-4-piperazinylbenzimidazoles: orally active inhibitors of the gonadotropin releasing hormone (GnRH) receptor.

Pelletier JC, Chengalvala M, Cottom J, Feingold I, Garrick L, Green D, Hauze D, Huselton C, Jetter J, Kao W, Kopf GS, Lundquist JT 4th, Mann C, Mehlmann J, Rogers J, Shanno L, Wrobel J. Pelletier JC, et al. Bioorg Med Chem. 2008 Jul 1;16(13):6617-40. doi: 10.1016/j.bmc.2008.05.024. Epub 2008 May 11. Bioorg Med Chem. 2008. PMID: 18511284

8

5-Alkylated thiazolidinones as follicle-stimulating hormone (FSH) receptor agonists.

Wrobel J, Jetter J, Kao W, Rogers J, Di L, Chi J, Peréz MC, Chen GC, Shen ES. Wrobel J, et al. Bioorg Med Chem. 2006 Aug 15;14(16):5729-41. doi: 10.1016/j.bmc.2006.04.012. Epub 2006 May 3. Bioorg Med Chem. 2006. PMID: 16675221

9

Synthesis of 4-(3-biaryl)quinoline sulfones as potent liver X receptor agonists.

Ullrich JW, Morris R, Bernotas RC, Travins JM, Jetter J, Unwalla R, Quinet E, Nambi P, Feingold I, Huselton C, Enroth C, Wilhelmsson A, Goos-Nilsson A, Wrobel J. Ullrich JW, et al. Among authors: jetter j. Bioorg Med Chem Lett. 2010 May 1;20(9):2903-7. doi: 10.1016/j.bmcl.2010.03.031. Epub 2010 Mar 9. Bioorg Med Chem Lett. 2010. PMID: 20382019

10

Identification of phenylsulfone-substituted quinoxaline (WYE-672) as a tissue selective liver X-receptor (LXR) agonist.

Hu B, Unwalla RJ, Goljer I, Jetter JW, Quinet EM, Berrodin TJ, Basso MD, Feingold IB, Nilsson AG, Wilhelmsson A, Evans MJ, Wrobel JE. Hu B, et al. Among authors: jetter jw. J Med Chem. 2010 Apr 22;53(8):3296-304. doi: 10.1021/jm100034x. J Med Chem. 2010. PMID: 20350005

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