Kessler H - Search Results

1

A backbone-cyclic, receptor 5-selective somatostatin analogue: synthesis, bioactivity, and nuclear magnetic resonance conformational analysis.

Gilon C, Huenges M, Mathä B, Gellerman G, Hornik V, Afargan M, Amitay O, Ziv O, Feller E, Gamliel A, Shohat D, Wanger M, Arad O, Kessler H. Gilon C, et al. Among authors: kessler h. J Med Chem. 1998 Mar 12;41(6):919-29. doi: 10.1021/jm970633x. J Med Chem. 1998. PMID: 9526566

2

Structure-activity relationship of the ring portion in backbone-cyclic C-terminal hexapeptide analogs of substance P. NMR and molecular dynamics.

Behrens S, Mathä B, Bitan G, Gilon C, Kessler H. Behrens S, et al. Among authors: kessler h. Int J Pept Protein Res. 1996 Dec;48(6):569-79. doi: 10.1111/j.1399-3011.1996.tb00876.x. Int J Pept Protein Res. 1996. PMID: 8985790

3

N-Methylated cyclic RGD peptides as highly active and selective alpha(V)beta(3) integrin antagonists.

Dechantsreiter MA, Planker E, Mathä B, Lohof E, Hölzemann G, Jonczyk A, Goodman SL, Kessler H. Dechantsreiter MA, et al. Among authors: kessler h. J Med Chem. 1999 Aug 12;42(16):3033-40. doi: 10.1021/jm970832g. J Med Chem. 1999. PMID: 10447947

4

Structure investigation of amphiphilic cyclopeptides in isotropic and anisotropic environments-A model study simulating peptide-membrane interactions.

Koppitz M, Mathä B, Kessler H. Koppitz M, et al. Among authors: kessler h. J Pept Sci. 1999 Nov;5(11):507-18. doi: 10.1002/(SICI)1099-1387(199911)5:11<507::AID-PSC219>3.0.CO;2-U. J Pept Sci. 1999. PMID: 10587314

5

Comparison of the conformation of active and nonactive backbone cyclic analogs of substance P as a tool to elucidate features of the bioactive conformation: NMR and molecular dynamics in DMSO and water.

Grdadolnik SG, Mierke DF, Byk G, Zeltser I, Gilon C, Kessler H. Grdadolnik SG, et al. Among authors: kessler h. J Med Chem. 1994 Jul 8;37(14):2145-52. doi: 10.1021/jm00040a005. J Med Chem. 1994. PMID: 7518522

6

Multiple N-methylation by a designed approach enhances receptor selectivity.

Chatterjee J, Ovadia O, Zahn G, Marinelli L, Hoffman A, Gilon C, Kessler H. Chatterjee J, et al. Among authors: kessler h. J Med Chem. 2007 Nov 29;50(24):5878-81. doi: 10.1021/jm701044r. Epub 2007 Nov 1. J Med Chem. 2007. PMID: 17973471

7

Improvement of drug-like properties of peptides: the somatostatin paradigm.

Ovadia O, Greenberg S, Laufer B, Gilon C, Hoffman A, Kessler H. Ovadia O, et al. Among authors: kessler h. Expert Opin Drug Discov. 2010 Jul;5(7):655-71. doi: 10.1517/17460441.2010.493935. Epub 2010 Jun 3. Expert Opin Drug Discov. 2010. PMID: 22823205

8

Cyclopropane-derived peptidomimetics. Design, synthesis, evaluation, and structure of novel HIV-1 protease inhibitors.

Martin SF, Dorsey GO, Gane T, Hillier MC, Kessler H, Baur M, Mathä B, Erickson JW, Bhat TN, Munshi S, Gulnik SV, Topol IA. Martin SF, et al. Among authors: kessler h. J Med Chem. 1998 May 7;41(10):1581-97. doi: 10.1021/jm980033d. J Med Chem. 1998. PMID: 9572884

9

cis-Peptide Bonds: A Key for Intestinal Permeability of Peptides? .

Marelli UK, Ovadia O, Frank AO, Chatterjee J, Gilon C, Hoffman A, Kessler H. Marelli UK, et al. Among authors: kessler h. Chemistry. 2015 Oct 19;21(43):15148-52. doi: 10.1002/chem.201501600. Epub 2015 Sep 4. Chemistry. 2015. PMID: 26337831

10

The effect of multiple N-methylation on intestinal permeability of cyclic hexapeptides.

Ovadia O, Greenberg S, Chatterjee J, Laufer B, Opperer F, Kessler H, Gilon C, Hoffman A. Ovadia O, et al. Among authors: kessler h. Mol Pharm. 2011 Apr 4;8(2):479-87. doi: 10.1021/mp1003306. Epub 2011 Mar 21. Mol Pharm. 2011. PMID: 21375270

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