Escarpe PA - Search Results

1

Oral administration of a prodrug of the influenza virus neuraminidase inhibitor GS 4071 protects mice and ferrets against influenza infection.

Mendel DB, Tai CY, Escarpe PA, Li W, Sidwell RW, Huffman JH, Sweet C, Jakeman KJ, Merson J, Lacy SA, Lew W, Williams MA, Zhang L, Chen MS, Bischofberger N, Kim CU. Mendel DB, et al. Among authors: escarpe pa. Antimicrob Agents Chemother. 1998 Mar;42(3):640-6. doi: 10.1128/AAC.42.3.640. Antimicrob Agents Chemother. 1998. PMID: 9517945 Free PMC article.

2

Identification of GS 4104 as an orally bioavailable prodrug of the influenza virus neuraminidase inhibitor GS 4071.

Li W, Escarpe PA, Eisenberg EJ, Cundy KC, Sweet C, Jakeman KJ, Merson J, Lew W, Williams M, Zhang L, Kim CU, Bischofberger N, Chen MS, Mendel DB. Li W, et al. Among authors: escarpe pa. Antimicrob Agents Chemother. 1998 Mar;42(3):647-53. doi: 10.1128/AAC.42.3.647. Antimicrob Agents Chemother. 1998. PMID: 9517946 Free PMC article.

3

Structure-activity relationship studies of novel carbocyclic influenza neuraminidase inhibitors.

Kim CU, Lew W, Williams MA, Wu H, Zhang L, Chen X, Escarpe PA, Mendel DB, Laver WG, Stevens RC. Kim CU, et al. Among authors: escarpe pa. J Med Chem. 1998 Jul 2;41(14):2451-60. doi: 10.1021/jm980162u. J Med Chem. 1998. PMID: 9651151

4

Characterization of human influenza virus variants selected in vitro in the presence of the neuraminidase inhibitor GS 4071.

Tai CY, Escarpe PA, Sidwell RW, Williams MA, Lew W, Wu H, Kim CU, Mendel DB. Tai CY, et al. Among authors: escarpe pa. Antimicrob Agents Chemother. 1998 Dec;42(12):3234-41. doi: 10.1128/AAC.42.12.3234. Antimicrob Agents Chemother. 1998. PMID: 9835519 Free PMC article.

5

A new series of C3-aza carbocyclic influenza neuraminidase inhibitors: synthesis and inhibitory activity.

Lew W, Wu H, Mendel DB, Escarpe PA, Chen X, Laver WG, Graves BJ, Kim CU. Lew W, et al. Among authors: escarpe pa. Bioorg Med Chem Lett. 1998 Dec 1;8(23):3321-4. doi: 10.1016/s0960-894x(98)00587-3. Bioorg Med Chem Lett. 1998. PMID: 9873727

6

Synthesis and evaluation of 1,4,5,6-tetrahydropyridazine derivatives as influenza neuraminidase inhibitors.

Zhang L, Williams MA, Mendel DB, Escarpe PA, Chen X, Wang KY, Graves BJ, Lawton G, Kim CU. Zhang L, et al. Among authors: escarpe pa. Bioorg Med Chem Lett. 1999 Jul 5;9(13):1751-6. doi: 10.1016/s0960-894x(99)00280-2. Bioorg Med Chem Lett. 1999. PMID: 10406636

7

Stereospecific synthesis of a GS 4104 metabolite: determination of absolute stereochemistry and influenza neuraminidase inhibitory activity.

Lew W, Escarpe PA, Mendel DB, Sweeny DJ, Kim CU. Lew W, et al. Among authors: escarpe pa. Bioorg Med Chem Lett. 1999 Oct 4;9(19):2811-4. doi: 10.1016/s0960-894x(99)00479-5. Bioorg Med Chem Lett. 1999. PMID: 10522696

8

Carbocyclic influenza neuraminidase inhibitors possessing a C3-cyclic amine side chain: synthesis and inhibitory activity.

Lew W, Wu H, Chen X, Graves BJ, Escarpe PA, MacArthur HL, Mendel DB, Kim CU. Lew W, et al. Among authors: escarpe pa. Bioorg Med Chem Lett. 2000 Jun 5;10(11):1257-60. doi: 10.1016/s0960-894x(00)00214-6. Bioorg Med Chem Lett. 2000. PMID: 10866394

9

A DLL3-targeted antibody-drug conjugate eradicates high-grade pulmonary neuroendocrine tumor-initiating cells in vivo.

Saunders LR, Bankovich AJ, Anderson WC, Aujay MA, Bheddah S, Black K, Desai R, Escarpe PA, Hampl J, Laysang A, Liu D, Lopez-Molina J, Milton M, Park A, Pysz MA, Shao H, Slingerland B, Torgov M, Williams SA, Foord O, Howard P, Jassem J, Badzio A, Czapiewski P, Harpole DH, Dowlati A, Massion PP, Travis WD, Pietanza MC, Poirier JT, Rudin CM, Stull RA, Dylla SJ. Saunders LR, et al. Among authors: escarpe pa. Sci Transl Med. 2015 Aug 26;7(302):302ra136. doi: 10.1126/scitranslmed.aac9459. Sci Transl Med. 2015. PMID: 26311731 Free PMC article.

10

Lentiviral vectors pseudotyped with baculovirus gp64 efficiently transduce mouse cells in vivo and show tropism restriction against hematopoietic cell types in vitro.

Schauber CA, Tuerk MJ, Pacheco CD, Escarpe PA, Veres G. Schauber CA, et al. Among authors: escarpe pa. Gene Ther. 2004 Feb;11(3):266-75. doi: 10.1038/sj.gt.3302170. Gene Ther. 2004. PMID: 14737086

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