Thaisrivongs S - Search Results

1

Structure-based design of HIV protease inhibitors: 5,6-dihydro-4-hydroxy-2-pyrones as effective, nonpeptidic inhibitors.

Thaisrivongs S, Romero DL, Tommasi RA, Janakiraman MN, Strohbach JW, Turner SR, Biles C, Morge RR, Johnson PD, Aristoff PA, Tomich PK, Lynn JC, Horng MM, Chong KT, Hinshaw RR, Howe WJ, Finzel BC, Watenpaugh KD. Thaisrivongs S, et al. J Med Chem. 1996 Nov 8;39(23):4630-42. doi: 10.1021/jm960228q. J Med Chem. 1996. PMID: 8917652

2

Inhibitors of the protease from human immunodeficiency virus: design and modeling of a compound containing a dihydroxyethylene isostere insert with high binding affinity and effective antiviral activity.

Thaisrivongs S, Tomasselli AG, Moon JB, Hui J, McQuade TJ, Turner SR, Strohbach JW, Howe WJ, Tarpley WG, Heinrikson RL. Thaisrivongs S, et al. J Med Chem. 1991 Aug;34(8):2344-56. doi: 10.1021/jm00112a005. J Med Chem. 1991. PMID: 1875334

3

Conformationally constrained renin inhibitory peptides: cyclic (3-1)-1-(carboxymethyl)-L-prolyl-L-phenylalanyl-L-histidinamide as a conformational restriction at the P2-P4 tripeptide portion of the angiotensinogen template.

Thaisrivongs S, Blinn JR, Pals DT, Turner SR. Thaisrivongs S, et al. J Med Chem. 1991 Apr;34(4):1276-82. doi: 10.1021/jm00108a006. J Med Chem. 1991. PMID: 2016704

4

Renin inhibitory peptides. A beta-aspartyl residue as a replacement for the histidyl residue at the P-2 site.

Thaisrivongs S, Mao B, Pals DT, Turner SR, Kroll LT. Thaisrivongs S, et al. J Med Chem. 1990 May;33(5):1337-43. doi: 10.1021/jm00167a009. J Med Chem. 1990. PMID: 2184238

5

Conformationally constrained renin inhibitory peptides: gamma-lactam-bridged dipeptide isostere as conformational restriction.

Thaisrivongs S, Pals DT, Turner SR, Kroll LT. Thaisrivongs S, et al. J Med Chem. 1988 Jul;31(7):1369-76. doi: 10.1021/jm00402a021. J Med Chem. 1988. PMID: 3290485

6

Structure-based design of novel HIV protease inhibitors: carboxamide-containing 4-hydroxycoumarins and 4-hydroxy-2-pyrones as potent nonpeptidic inhibitors.

Thaisrivongs S, Watenpaugh KD, Howe WJ, Tomich PK, Dolak LA, Chong KT, Tomich CC, Tomasselli AG, Turner SR, Strohbach JW, et al. Thaisrivongs S, et al. J Med Chem. 1995 Sep 1;38(18):3624-37. doi: 10.1021/jm00018a023. J Med Chem. 1995. PMID: 7658450

7

Structure-based design of HIV protease inhibitors: 4-hydroxycoumarins and 4-hydroxy-2-pyrones as non-peptidic inhibitors.

Thaisrivongs S, Tomich PK, Watenpaugh KD, Chong KT, Howe WJ, Yang CP, Strohbach JW, Turner SR, McGrath JP, Bohanon MJ, et al. Thaisrivongs S, et al. J Med Chem. 1994 Sep 30;37(20):3200-4. doi: 10.1021/jm00046a002. J Med Chem. 1994. PMID: 7932546 No abstract available.

8

Peptidomimetic HIV protease inhibitors: phosphate prodrugs with improved biological activities.

Chong KT, Ruwart MJ, Hinshaw RR, Wilkinson KF, Rush BD, Yancey MF, Strohbach JW, Thaisrivongs S. Chong KT, et al. Among authors: thaisrivongs s. J Med Chem. 1993 Aug 20;36(17):2575-7. doi: 10.1021/jm00069a018. J Med Chem. 1993. PMID: 8355256 No abstract available.

9

Inhibitors of the protease from human immunodeficiency virus: synthesis, enzyme inhibition, and antiviral activity of a series of compounds containing the dihydroxyethylene transition-state isostere.

Thaisrivongs S, Turner SR, Strohbach JW, TenBrink RE, Tarpley WG, McQuade TJ, Heinrikson RL, Tomasselli AG, Hui JO, Howe WJ. Thaisrivongs S, et al. J Med Chem. 1993 Apr 16;36(8):941-52. doi: 10.1021/jm00060a001. J Med Chem. 1993. PMID: 8478908

10

Structure-based design of novel HIV protease inhibitors: sulfonamide-containing 4-hydroxycoumarins and 4-hydroxy-2-pyrones as potent non-peptidic inhibitors.

Thaisrivongs S, Janakiraman MN, Chong KT, Tomich PK, Dolak LA, Turner SR, Strohbach JW, Lynn JC, Horng MM, Hinshaw RR, Watenpaugh KD. Thaisrivongs S, et al. J Med Chem. 1996 Jun 7;39(12):2400-10. doi: 10.1021/jm950888f. J Med Chem. 1996. PMID: 8691434

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