Trapani AJ - Search Results

1

Design and synthesis of an orally active macrocyclic neutral endopeptidase 24.11 inhibitor.

MacPherson LJ, Bayburt EK, Capparelli MP, Bohacek RS, Clarke FH, Ghai RD, Sakane Y, Berry CJ, Peppard JV, Trapani AJ. MacPherson LJ, et al. Among authors: trapani aj. J Med Chem. 1993 Nov 26;36(24):3821-8. doi: 10.1021/jm00076a009. J Med Chem. 1993. PMID: 8254611

2

Dicarboxylic acid dipeptide neutral endopeptidase inhibitors.

Ksander GM, Ghai RD, deJesus R, Diefenbacher CG, Yuan A, Berry C, Sakane Y, Trapani A. Ksander GM, et al. J Med Chem. 1995 May 12;38(10):1689-700. doi: 10.1021/jm00010a014. J Med Chem. 1995. PMID: 7752193

3

Ortho-substituted benzofused macrocyclic lactams as zinc metalloprotease inhibitors.

Ksander GM, de Jesus R, Yuan A, Ghai RD, Trapani A, McMartin C, Bohacek R. Ksander GM, et al. J Med Chem. 1997 Feb 14;40(4):495-505. doi: 10.1021/jm960582o. J Med Chem. 1997. PMID: 9046340

4

Pharmacologic profile of CGS 24128, a potent, long-acting inhibitor of neutral endopeptidase 24.11.

Trapani AJ, Beil ME, Coté DT, de Lombaert S, Erion MD, Gerlock TE, Ghai RD, Hopkins MF, Peppard JV, Webb RL, et al. Trapani AJ, et al. J Cardiovasc Pharmacol. 1994 Mar;23(3):358-64. J Cardiovasc Pharmacol. 1994. PMID: 7515977

5

A rapid indirect method to determine the plasma concentrations of neutral endopeptidase inhibitors.

Ghai RD, De Lombaert S, Ksander GM, Berry C, Sakane Y, Trapani AJ. Ghai RD, et al. Among authors: trapani aj. Res Commun Mol Pathol Pharmacol. 1995 Feb;87(2):211-20. Res Commun Mol Pathol Pharmacol. 1995. PMID: 7749658

6

Pharmacological profile of a non-peptidic dual inhibitor of neutral endopeptidase 24.11 and endothelin-converting enzyme.

De Lombaert S, Ghai RD, Jeng AY, Trapani AJ, Webb RL. De Lombaert S, et al. Among authors: trapani aj. Biochem Biophys Res Commun. 1994 Oct 14;204(1):407-12. doi: 10.1006/bbrc.1994.2473. Biochem Biophys Res Commun. 1994. PMID: 7945387

7

N-Phosphonomethyl dipeptides and their phosphonate prodrugs, a new generation of neutral endopeptidase (NEP, EC 3.4.24.11) inhibitors.

De Lombaert S, Erion MD, Tan J, Blanchard L, el-Chehabi L, Ghai RD, Sakane Y, Berry C, Trapani AJ. De Lombaert S, et al. Among authors: trapani aj. J Med Chem. 1994 Feb 18;37(4):498-511. doi: 10.1021/jm00030a009. J Med Chem. 1994. PMID: 8120868

8

The pharmacology of CGS 25462: a potent, orally bioavailable, long-acting inhibitor of neutral endopeptidase 24.11.

Trapani AJ, De Lombaert S, Erion MD, Ghai RD, Peppard JV, Lappe RW, Worcel M. Trapani AJ, et al. J Hypertens Suppl. 1993 Dec;11(5):S220-1. J Hypertens Suppl. 1993. PMID: 8158354 No abstract available.

9

Heterocyclic lactam derivatives as dual angiotensin converting enzyme and neutral endopeptidase 24.11 inhibitors.

Stanton JL, Sperbeck DM, Trapani AJ, Cote D, Sakane Y, Berry CJ, Ghai RD. Stanton JL, et al. Among authors: trapani aj. J Med Chem. 1993 Nov 26;36(24):3829-33. doi: 10.1021/jm00076a010. J Med Chem. 1993. PMID: 8254612

10

New alpha-thiol dipeptide dual inhibitors of angiotensin-I converting enzyme and neutral endopeptidase EC 3.4.24.11.

Fink CA, Qiao Y, Berry CJ, Sakane Y, Ghai RD, Trapani AJ. Fink CA, et al. Among authors: trapani aj. J Med Chem. 1995 Dec 22;38(26):5023-30. doi: 10.1021/jm00026a009. J Med Chem. 1995. PMID: 8544178

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