Gluchowski C - Search Results

1

Design, synthesis and evaluation of substituted triarylnipecotic acid derivatives as GABA uptake inhibitors: identification of a ligand with moderate affinity and selectivity for the cloned human GABA transporter GAT-3.

Dhar TG, Borden LA, Tyagarajan S, Smith KE, Branchek TA, Weinshank RL, Gluchowski C. Dhar TG, et al. Among authors: gluchowski c. J Med Chem. 1994 Jul 22;37(15):2334-42. doi: 10.1021/jm00041a012. J Med Chem. 1994. PMID: 8057281

2

Discovery of alpha 1a-adrenergic receptor antagonists based on the L-type Ca2+ channel antagonist niguldipine.

Wetzel JM, Miao SW, Forray C, Borden LA, Branchek TA, Gluchowski C. Wetzel JM, et al. Among authors: gluchowski c. J Med Chem. 1995 May 12;38(10):1579-81. doi: 10.1021/jm00010a001. J Med Chem. 1995. PMID: 7752182 No abstract available.

3

Tiagabine, SK&F 89976-A, CI-966, and NNC-711 are selective for the cloned GABA transporter GAT-1.

Borden LA, Murali Dhar TG, Smith KE, Weinshank RL, Branchek TA, Gluchowski C. Borden LA, et al. Among authors: gluchowski c. Eur J Pharmacol. 1994 Oct 14;269(2):219-24. doi: 10.1016/0922-4106(94)90089-2. Eur J Pharmacol. 1994. PMID: 7851497

4

Cloning of the human homologue of the GABA transporter GAT-3 and identification of a novel inhibitor with selectivity for this site.

Borden LA, Dhar TG, Smith KE, Branchek TA, Gluchowski C, Weinshank RL. Borden LA, et al. Among authors: gluchowski c. Recept Channels. 1994;2(3):207-13. Recept Channels. 1994. PMID: 7874447

5

Design and synthesis of novel alpha1a adrenoceptor-selective dihydropyridine antagonists for the treatment of benign prostatic hyperplasia.

Nagarathnam D, Wetzel JM, Miao SW, Marzabadi MR, Chiu G, Wong WC, Hong X, Fang J, Forray C, Branchek TA, Heydorn WE, Chang RS, Broten T, Schorn TW, Gluchowski C. Nagarathnam D, et al. Among authors: gluchowski c. J Med Chem. 1998 Dec 17;41(26):5320-33. doi: 10.1021/jm980506g. J Med Chem. 1998. PMID: 9857099

6

Modeling the G-protein-coupled neuropeptide Y Y1 receptor agonist and antagonist binding sites.

Du P, Salon JA, Tamm JA, Hou C, Cui W, Walker MW, Adham N, Dhanoa DS, Islam I, Vaysse PJ, Dowling B, Shifman Y, Boyle N, Rueger H, Schmidlin T, Yamaguchi Y, Branchek TA, Weinshank RL, Gluchowski C. Du P, et al. Among authors: gluchowski c. Protein Eng. 1997 Feb;10(2):109-17. doi: 10.1093/protein/10.2.109. Protein Eng. 1997. PMID: 9089810

7

2-amino-2-oxazolines as subtype selective alpha(2) adrenoceptor agonists.

Wong WC, Sun W, Cui W, Chen Y, Forray C, Vaysse PJ, Branchek TA, Gluchowski C. Wong WC, et al. Among authors: gluchowski c. J Med Chem. 2000 May 4;43(9):1699-704. doi: 10.1021/jm9905256. J Med Chem. 2000. PMID: 10794687

8

Modeling and mutagenesis of the human alpha 1a-adrenoceptor: orientation and function of transmembrane helix V sidechains.

Wetzel JM, Salon JA, Tamm JA, Forray C, Craig D, Nakanishi H, Cui W, Vaysse PJ, Chiu G, Weinshank RL, Hartig PR, Branchek TA, Gluchowski C. Wetzel JM, et al. Among authors: gluchowski c. Recept Channels. 1996;4(3):165-77. Recept Channels. 1996. PMID: 9014240

9

Identification of a dihydropyridine as a potent alpha1a adrenoceptor-selective antagonist that inhibits phenylephrine-induced contraction of the human prostate.

Wong WC, Chiu G, Wetzel JM, Marzabadi MR, Nagarathnam D, Wang D, Fang J, Miao SW, Hong X, Forray C, Vaysse PJ, Branchek TA, Gluchowski C, Tang R, Lepor H. Wong WC, et al. Among authors: gluchowski c. J Med Chem. 1998 Jul 2;41(14):2643-50. doi: 10.1021/jm980077m. J Med Chem. 1998. PMID: 9651170

10

Design and synthesis of novel alpha(1)(a) adrenoceptor-selective antagonists. 3. Approaches to eliminate opioid agonist metabolites by using substituted phenylpiperazine side chains.

Lagu B, Tian D, Nagarathnam D, Marzabadi MR, Wong WC, Miao SW, Zhang F, Sun W, Chiu G, Fang J, Forray C, Chang RS, Ransom RW, Chen TB, O'Malley S, Zhang K, Vyas KP, Gluchowski C. Lagu B, et al. Among authors: gluchowski c. J Med Chem. 1999 Nov 18;42(23):4794-803. doi: 10.1021/jm990202+. J Med Chem. 1999. PMID: 10579842

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