Kumar R - Search Results

1

2-(4-Bromobenzyl) tethered 4-amino aryl/alkyl-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidines: design, synthesis, anticancer assessment via dual topoisomerase-I/II inhibition, and in silico studies.

Arora S, Patra B, Dhamija I, Guru SK, Kumar R. Arora S, et al. Among authors: kumar r. RSC Med Chem. 2024 Dec 17. doi: 10.1039/d4md00817k. Online ahead of print. RSC Med Chem. 2024. PMID: 39697244 Free PMC article.

2

Anticancer potential of some imidazole and fused imidazole derivatives: exploring the mechanism via epidermal growth factor receptor (EGFR) inhibition.

Kalra S, Joshi G, Kumar M, Arora S, Kaur H, Singh S, Munshi A, Kumar R. Kalra S, et al. Among authors: kumar r, kumar m. RSC Med Chem. 2020 Jul 8;11(8):923-939. doi: 10.1039/d0md00146e. eCollection 2020 Aug 1. RSC Med Chem. 2020. PMID: 33479688 Free PMC article.

3

A Perspective on Medicinal Chemistry Approaches for Targeting Pyruvate Kinase M2.

Arora S, Joshi G, Chaturvedi A, Heuser M, Patil S, Kumar R. Arora S, et al. Among authors: kumar r. J Med Chem. 2022 Jan 27;65(2):1171-1205. doi: 10.1021/acs.jmedchem.1c00981. Epub 2021 Nov 2. J Med Chem. 2022. PMID: 34726055

4

Design, synthesis and anticancer activity of 2-arylimidazo[1,2-a]pyridinyl-3-amines.

Yadav UP, Ansari AJ, Arora S, Joshi G, Singh T, Kaur H, Dogra N, Kumar R, Kumar S, Sawant DM, Singh S. Yadav UP, et al. Among authors: kumar s, kumar r. Bioorg Chem. 2022 Jan;118:105464. doi: 10.1016/j.bioorg.2021.105464. Epub 2021 Nov 1. Bioorg Chem. 2022. PMID: 34785441

5

Design and Synthesis of Non-Covalent Imidazo[1,2-a]quinoxaline-Based Inhibitors of EGFR and Their Anti-Cancer Assessment.

Kumar M, Joshi G, Arora S, Singh T, Biswas S, Sharma N, Bhat ZR, Tikoo K, Singh S, Kumar R. Kumar M, et al. Among authors: kumar r. Molecules. 2021 Mar 9;26(5):1490. doi: 10.3390/molecules26051490. Molecules. 2021. PMID: 33803355 Free PMC article.

6

Synthesis of 1,4-dihydropyrazolo[4,3-b]indoles via intramolecular C(sp²)-N bond formation involving nitrene insertion, DFT study and their anticancer assessment.

Kaur M, Mehta V, Abdullah Wani A, Arora S, Bharatam PV, Sharon A, Singh S, Kumar R. Kaur M, et al. Among authors: kumar r. Bioorg Chem. 2021 Sep;114:105114. doi: 10.1016/j.bioorg.2021.105114. Epub 2021 Jun 29. Bioorg Chem. 2021. PMID: 34243073

7

Rationalization of the activity Profile of Pyruvate Kinase Isozyme M2 (PKM2) Inhibitors using 3D QSAR.

Kusuma M, Arora S, Kalra S, Chaturvedi A, Heuser M, Kumar R. Kusuma M, et al. Among authors: kumar r. Curr Top Med Chem. 2021;21(25):2258-2271. doi: 10.2174/1568026621666210804124555. Curr Top Med Chem. 2021. PMID: 34348626

8

Targeting the Epidermal Growth Factor Receptor with Molecular Degraders: State-of-the-Art and Future Opportunities.

Maity P, Chatterjee J, Patil KT, Arora S, Katiyar MK, Kumar M, Samarbakhsh A, Joshi G, Bhutani P, Chugh M, Gavande NS, Kumar R. Maity P, et al. Among authors: kumar r, kumar m. J Med Chem. 2023 Mar 9;66(5):3135-3172. doi: 10.1021/acs.jmedchem.2c01242. Epub 2023 Feb 22. J Med Chem. 2023. PMID: 36812395 Review.

9

Pore-forming proteins and their role in cancer and inflammation: Mechanistic insights and plausible druggable targets.

Sankar J, Arora S, Joshi G, Kumar R. Sankar J, et al. Among authors: kumar r. Chem Biol Interact. 2022 Oct 1;366:110127. doi: 10.1016/j.cbi.2022.110127. Epub 2022 Aug 30. Chem Biol Interact. 2022. PMID: 36055376 Review.

10

Design, synthesis, and anticancer assessment of structural analogues of (E)-1-((3,4,5-trimethoxybenzylidene)amino)-4-(3,4,5-trimethoxyphenyl)imidazo[1,2-a]quinoxaline-2-carbonitrile (6b), an imidazo[1,2-a]quinoxaline-based non-covalent EGFR inhibitor.

Kumar M, Patil KT, Maity P, Chatterjee J, Singh T, Joshi G, Singh S, Kumar R. Kumar M, et al. Among authors: kumar r. RSC Med Chem. 2024 Jun 20;15(7):2322-2339. doi: 10.1039/d4md00237g. eCollection 2024 Jul 17. RSC Med Chem. 2024. PMID: 39026650

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