Asawa Y - Search Results

1

Discovery of Disubstituted Carboranes as Inhibitors of Heat Shock Protein 90-Heat Shock Factor 1 Interaction.

Shao Y, Miura K, Asawa Y, Morita T, Li G, Nakamura H. Shao Y, et al. Among authors: asawa y. ACS Med Chem Lett. 2024 Apr 8;15(5):619-625. doi: 10.1021/acsmedchemlett.4c00022. eCollection 2024 May 9. ACS Med Chem Lett. 2024. PMID: 38746882

2

Development of 1-aryl-3-furanyl/thienyl-imidazopyridine templates for inhibitors against hypoxia inducible factor (HIF)-1 transcriptional activity.

Fuse S, Ohuchi T, Asawa Y, Sato S, Nakamura H. Fuse S, et al. Among authors: asawa y. Bioorg Med Chem Lett. 2016 Dec 15;26(24):5887-5890. doi: 10.1016/j.bmcl.2016.11.009. Epub 2016 Nov 5. Bioorg Med Chem Lett. 2016. PMID: 27847273

3

Structure-based drug design of novel carborane-containing nicotinamide phosphoribosyltransferase inhibitors.

Asawa Y, Katsuragi K, Sato A, Yoshimori A, Tanuma SI, Nakamura H. Asawa Y, et al. Bioorg Med Chem. 2019 Jul 1;27(13):2832-2844. doi: 10.1016/j.bmc.2019.05.013. Epub 2019 May 10. Bioorg Med Chem. 2019. PMID: 31103405

4

Regulation of CD28 binding to SH2 domains of Grb2 and PI3K by trisubstituted carboranes for T-cell activation.

Ogawa S, Asawa Y, Iiyama M, Yoshimori A, Nakamura H, Oda M. Ogawa S, et al. Among authors: asawa y. Bioorg Med Chem Lett. 2022 Dec 15;78:129049. doi: 10.1016/j.bmcl.2022.129049. Epub 2022 Nov 7. Bioorg Med Chem Lett. 2022. PMID: 36356833

5

Design and synthesis of 14 and 15-membered macrocyclic scaffolds exhibiting inhibitory activities of hypoxia-inducible factor 1α.

Shimizu T, Takahashi N, Huber VJ, Asawa Y, Ueda H, Yoshimori A, Muramatsu Y, Seimiya H, Kouji H, Nakamura H, Oguri H. Shimizu T, et al. Among authors: asawa y. Bioorg Med Chem. 2021 Jan 15;30:115949. doi: 10.1016/j.bmc.2020.115949. Epub 2020 Dec 13. Bioorg Med Chem. 2021. PMID: 33360196

6

Enantioselective Synthesis of Oxazaborolidines by Palladium-Catalyzed N-H/B-H Double Activation of 1,2-Azaborines.

Morita T, Murakami H, Asawa Y, Nakamura H. Morita T, et al. Among authors: asawa y. Angew Chem Int Ed Engl. 2022 Feb 7;61(7):e202113558. doi: 10.1002/anie.202113558. Epub 2021 Dec 29. Angew Chem Int Ed Engl. 2022. PMID: 34913232

7

Comprehensive exploration of chemical space using trisubstituted carboranes.

Asawa Y, Hatsuzawa S, Yoshimori A, Yamada K, Katoh A, Kouji H, Nakamura H. Asawa Y, et al. Sci Rep. 2021 Dec 16;11(1):24101. doi: 10.1038/s41598-021-03459-6. Sci Rep. 2021. PMID: 34916538 Free PMC article.

8

Prediction of an MMP-1 inhibitor activity cliff using the SAR matrix approach and its experimental validation.

Asawa Y, Yoshimori A, Bajorath J, Nakamura H. Asawa Y, et al. Sci Rep. 2020 Sep 7;10(1):14710. doi: 10.1038/s41598-020-71696-2. Sci Rep. 2020. PMID: 32895466 Free PMC article.

9

Development of curcumin-based amyloid β aggregation inhibitors for Alzheimer's disease using the SAR matrix approach.

Yudi Utomo R, Asawa Y, Okada S, Ban HS, Yoshimori A, Bajorath J, Nakamura H. Yudi Utomo R, et al. Among authors: asawa y. Bioorg Med Chem. 2021 Sep 15;46:116357. doi: 10.1016/j.bmc.2021.116357. Epub 2021 Aug 8. Bioorg Med Chem. 2021. PMID: 34391121

10

Carborane as an Alternative Efficient Hydrophobic Tag for Protein Degradation.

Asawa Y, Nishida K, Kawai K, Domae K, Ban HS, Kitazaki A, Asami H, Kohno JY, Okada S, Tokuma H, Sakano D, Kume S, Tanaka M, Nakamura H. Asawa Y, et al. Bioconjug Chem. 2021 Nov 17;32(11):2377-2385. doi: 10.1021/acs.bioconjchem.1c00431. Epub 2021 Oct 26. Bioconjug Chem. 2021. PMID: 34699716

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