Goudet C - Search Results

1

Novel Inhibitory Site Revealed by XAP044 Mode of Action on the Metabotropic Glutamate 7 Receptor Venus Flytrap Domain.

Cristiano N, Cabayé A, Brabet I, Glatthar R, Tora A, Goudet C, Bertrand HO, Goupil-Lamy A, Flor PJ, Pin JP, McCort-Tranchepain I, Acher FC. Cristiano N, et al. Among authors: goudet c. J Med Chem. 2024 Jul 25;67(14):11662-11687. doi: 10.1021/acs.jmedchem.3c01924. Epub 2024 May 1. J Med Chem. 2024. PMID: 38691510 Free article.

2

Heptahelical domain of metabotropic glutamate receptor 5 behaves like rhodopsin-like receptors.

Goudet C, Gaven F, Kniazeff J, Vol C, Liu J, Cohen-Gonsaud M, Acher F, Prézeau L, Pin JP. Goudet C, et al. Proc Natl Acad Sci U S A. 2004 Jan 6;101(1):378-83. doi: 10.1073/pnas.0304699101. Epub 2003 Dec 22. Proc Natl Acad Sci U S A. 2004. PMID: 14691258 Free PMC article.

3

Locking the dimeric GABA(B) G-protein-coupled receptor in its active state.

Kniazeff J, Saintot PP, Goudet C, Liu J, Charnet A, Guillon G, Pin JP. Kniazeff J, et al. Among authors: goudet c. J Neurosci. 2004 Jan 14;24(2):370-7. doi: 10.1523/JNEUROSCI.3141-03.2004. J Neurosci. 2004. PMID: 14724235 Free PMC article.

4

Molecular mechanisms of GABA(B) receptor activation: new insights from the mechanism of action of CGP7930, a positive allosteric modulator.

Binet V, Goudet C, Brajon C, Le Corre L, Acher F, Pin JP, Prézeau L. Binet V, et al. Among authors: goudet c. Biochem Soc Trans. 2004 Nov;32(Pt 5):871-2. doi: 10.1042/BST0320871. Biochem Soc Trans. 2004. PMID: 15494037 Review.

5

Asymmetric functioning of dimeric metabotropic glutamate receptors disclosed by positive allosteric modulators.

Goudet C, Kniazeff J, Hlavackova V, Malhaire F, Maurel D, Acher F, Blahos J, Prézeau L, Pin JP. Goudet C, et al. J Biol Chem. 2005 Jul 1;280(26):24380-5. doi: 10.1074/jbc.M502642200. Epub 2005 Apr 29. J Biol Chem. 2005. PMID: 15863499 Free PMC article.

6

Interaction of novel positive allosteric modulators of metabotropic glutamate receptor 5 with the negative allosteric antagonist site is required for potentiation of receptor responses.

Chen Y, Nong Y, Goudet C, Hemstapat K, de Paulis T, Pin JP, Conn PJ. Chen Y, et al. Among authors: goudet c. Mol Pharmacol. 2007 May;71(5):1389-98. doi: 10.1124/mol.106.032425. Epub 2007 Feb 15. Mol Pharmacol. 2007. PMID: 17303702

7

Synthesis and biological evaluation of 1-amino-2-phosphonomethylcyclopropanecarboxylic acids, new group III metabotropic glutamate receptor agonists.

Sibille P, Lopez S, Brabet I, Valenti O, Oueslati N, Gaven F, Goudet C, Bertrand HO, Neyton J, Marino MJ, Amalric M, Pin JP, Acher FC. Sibille P, et al. Among authors: goudet c. J Med Chem. 2007 Jul 26;50(15):3585-95. doi: 10.1021/jm070262c. Epub 2007 Jun 28. J Med Chem. 2007. PMID: 17602546

8

L-(+)-2-Amino-4-thiophosphonobutyric acid (L-thioAP4), a new potent agonist of group III metabotropic glutamate receptors: increased distal acidity affords enhanced potency.

Selvam C, Goudet C, Oueslati N, Pin JP, Acher FC. Selvam C, et al. Among authors: goudet c. J Med Chem. 2007 Sep 20;50(19):4656-64. doi: 10.1021/jm070400y. Epub 2007 Aug 28. J Med Chem. 2007. PMID: 17722902

9

Group III metabotropic glutamate receptors inhibit hyperalgesia in animal models of inflammation and neuropathic pain.

Goudet C, Chapuy E, Alloui A, Acher F, Pin JP, Eschalier A. Goudet C, et al. Pain. 2008 Jul;137(1):112-124. doi: 10.1016/j.pain.2007.08.020. Epub 2007 Sep 27. Pain. 2008. PMID: 17900808 Free article.

10

N-{4-Chloro-2-[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)methyl]phenyl}-2-hydroxybenzamide (CPPHA) acts through a novel site as a positive allosteric modulator of group 1 metabotropic glutamate receptors.

Chen Y, Goudet C, Pin JP, Conn PJ. Chen Y, et al. Among authors: goudet c. Mol Pharmacol. 2008 Mar;73(3):909-18. doi: 10.1124/mol.107.040097. Epub 2007 Dec 4. Mol Pharmacol. 2008. PMID: 18056795

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