Leurs R - Search Results

1

Pharmacological Characterization and Radiolabeling of VUF15485, a High-Affinity Small-Molecule Agonist for the Atypical Chemokine Receptor ACKR3.

Zarca AM, Adlere I, Viciano CP, Arimont-Segura M, Meyrath M, Simon IA, Bebelman JP, Laan D, Custers HGJ, Janssen E, Versteegh KL, Buzink MCML, Nesheva DN, Bosma R, de Esch IJP, Vischer HF, Wijtmans M, Szpakowska M, Chevigné A, Hoffmann C, de Graaf C, Zarzycka BA, Windhorst AD, Smit MJ, Leurs R. Zarca AM, et al. Among authors: leurs r. Mol Pharmacol. 2024 Mar 14;105(4):301-312. doi: 10.1124/molpharm.123.000835. Mol Pharmacol. 2024. PMID: 38346795

2

Short-term desensitization of the histamine H1 receptor in human HeLa cells: involvement of protein kinase C dependent and independent pathways.

Smit MJ, Bloemers SM, Leurs R, Tertoolen LG, Bast A, de Laat SW, Timmerman H. Smit MJ, et al. Among authors: leurs r. Br J Pharmacol. 1992 Oct;107(2):448-55. doi: 10.1111/j.1476-5381.1992.tb12766.x. Br J Pharmacol. 1992. PMID: 1422591 Free PMC article.

3

Effects of histamine H1-, H2- and H3-receptor selective drugs on the mechanical activity of guinea-pig small and large intestine.

Leurs R, Brozius MM, Smit MJ, Bast A, Timmerman H. Leurs R, et al. Br J Pharmacol. 1991 Jan;102(1):179-85. doi: 10.1111/j.1476-5381.1991.tb12150.x. Br J Pharmacol. 1991. PMID: 1646056 Free PMC article.

4

Is protein kinase C involved in histamine H1-receptor desensitization?

Leurs R, Smit MJ, Brozius MM, Jansen W, Bast A, Timmerman H. Leurs R, et al. Agents Actions Suppl. 1991;33:393-402. doi: 10.1007/978-3-0348-7309-3_29. Agents Actions Suppl. 1991. PMID: 1647131

5

Homologous histamine H1 receptor desensitization results in reduction of H1 receptor agonist efficacy.

Leurs R, Smit MJ, Bast A, Timmerman H. Leurs R, et al. Eur J Pharmacol. 1991 Apr 24;196(3):319-22. doi: 10.1016/0014-2999(91)90446-w. Eur J Pharmacol. 1991. PMID: 1654256

6

Different profiles of desensitization dynamics in guinea-pig jejunal longitudinal smooth muscle after stimulation with histamine and methacholine.

Leurs R, Smit MJ, Bast A, Timmerman H. Leurs R, et al. Br J Pharmacol. 1990 Dec;101(4):881-8. doi: 10.1111/j.1476-5381.1990.tb14175.x. Br J Pharmacol. 1990. PMID: 2085711 Free PMC article.

7

Molecular pharmacological aspects of histamine receptors.

Leurs R, Smit MJ, Timmerman H. Leurs R, et al. Pharmacol Ther. 1995 Jun;66(3):413-63. doi: 10.1016/0163-7258(95)00006-3. Pharmacol Ther. 1995. PMID: 7494855 Review.

8

Visualization of agonist-induced internalization of histamine H2 receptors.

Smit MJ, Timmerman H, Alewijnse AE, Punin M, van den Nieuwenhof I, Blauw J, van Minnen J, Leurs R. Smit MJ, et al. Among authors: leurs r. Biochem Biophys Res Commun. 1995 Sep 25;214(3):1138-45. doi: 10.1006/bbrc.1995.2404. Biochem Biophys Res Commun. 1995. PMID: 7575521

9

Lysine200 located in the fifth transmembrane domain of the histamine H1 receptor interacts with histamine but not with all H1 agonists.

Leurs R, Smit MJ, Meeder R, Ter Laak AM, Timmerman H. Leurs R, et al. Biochem Biophys Res Commun. 1995 Sep 5;214(1):110-7. doi: 10.1006/bbrc.1995.2263. Biochem Biophys Res Commun. 1995. PMID: 7669031

10

Rapid desensitization of the histamine H2 receptor on the human monocytic cell line U937.

Smit MJ, Leurs R, Shukrula SR, Bast A, Timmerman H. Smit MJ, et al. Among authors: leurs r. Eur J Pharmacol. 1994 Dec 15;288(1):17-25. doi: 10.1016/0922-4106(94)90005-1. Eur J Pharmacol. 1994. PMID: 7705464

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