Brackett CM - Search Results

1

Enniatin A Analogues as Novel Hsp90 Inhibitors that Modulate Triple-Negative Breast Cancer.

Serwetnyk MA, Crowley VM, Brackett CM, Carter TR, Elahi A, Kommalapati VK, Chadli A, Blagg BSJ. Serwetnyk MA, et al. Among authors: brackett cm. ACS Med Chem Lett. 2023 Nov 17;14(12):1785-1790. doi: 10.1021/acsmedchemlett.3c00423. eCollection 2023 Dec 14. ACS Med Chem Lett. 2023. PMID: 38116437 Free PMC article.

2

The discovery of N-1 substituted 2-aminobenzimidazoles as zinc-dependent S. aureus biofilm inhibitors.

Lindsey EA, Brackett CM, Mullikin T, Alcaraz C, Melander C. Lindsey EA, et al. Among authors: brackett cm. Medchemcomm. 2012 Jan 1;3(11):1462-1465. doi: 10.1039/C2MD20244A. Epub 2012 Sep 18. Medchemcomm. 2012. PMID: 23162679 Free PMC article.

3

Catalysis-Enabled Access to Cryptic Geldanamycin Oxides.

Hilton MJ, Brackett CM, Mercado BQ, Blagg BSJ, Miller SJ. Hilton MJ, et al. Among authors: brackett cm. ACS Cent Sci. 2020 Mar 25;6(3):426-435. doi: 10.1021/acscentsci.0c00024. Epub 2020 Feb 24. ACS Cent Sci. 2020. PMID: 32232143 Free PMC article.

4

Current Status of SUMOylation Inhibitors.

Brackett CM, Blagg BSJ. Brackett CM, et al. Curr Med Chem. 2021;28(20):3892-3912. doi: 10.2174/0929867327666200810135039. Curr Med Chem. 2021. PMID: 32778019 Free PMC article. Review.

5

Synthesis and Evaluation of Ginkgolic Acid Derivatives as SUMOylation Inhibitors.

Brackett CM, García-Casas A, Castillo-Lluva S, Blagg BSJ. Brackett CM, et al. ACS Med Chem Lett. 2020 Sep 24;11(11):2221-2226. doi: 10.1021/acsmedchemlett.0c00353. eCollection 2020 Nov 12. ACS Med Chem Lett. 2020. PMID: 33214832 Free PMC article.

6

Biological Evaluation of 5'-(N-Ethylcarboxamido)adenosine Analogues as Grp94-Selective Inhibitors.

Tosh DK, Brackett CM, Jung YH, Gao ZG, Banerjee M, Blagg BSJ, Jacobson KA. Tosh DK, et al. Among authors: brackett cm. ACS Med Chem Lett. 2021 Mar 1;12(3):373-379. doi: 10.1021/acsmedchemlett.0c00509. eCollection 2021 Mar 11. ACS Med Chem Lett. 2021. PMID: 33738064 Free PMC article.

7

The biology and inhibition of glucose-regulated protein 94/gp96.

Pugh KW, Alnaed M, Brackett CM, Blagg BSJ. Pugh KW, et al. Among authors: brackett cm. Med Res Rev. 2022 Nov;42(6):2007-2024. doi: 10.1002/med.21915. Epub 2022 Jul 21. Med Res Rev. 2022. PMID: 35861260 Free PMC article. Review.

8

Elucidation of novel TRAP1-Selective inhibitors that regulate mitochondrial processes.

Merfeld T, Peng S, Keegan BM, Crowley VM, Brackett CM, Gutierrez A, McCann NR, Reynolds TS, Rhodes MC, Byrd KM, Deng J, Matts RL, Blagg BSJ. Merfeld T, et al. Among authors: brackett cm. Eur J Med Chem. 2023 Oct 5;258:115531. doi: 10.1016/j.ejmech.2023.115531. Epub 2023 Jun 5. Eur J Med Chem. 2023. PMID: 37307624 Free PMC article.

9

Inhibiting spinal cord-specific hsp90 isoforms reveals a novel strategy to improve the therapeutic index of opioid treatment.

Duron DI, Tanguturi P, Campbell CS, Chou K, Bejarano P, Gabriel KA, Bowden JL, Mishra S, Brackett C, Barlow D, Houseknecht KL, Blagg BSJ, Streicher JM. Duron DI, et al. Sci Rep. 2024 Jun 26;14(1):14715. doi: 10.1038/s41598-024-65637-6. Sci Rep. 2024. PMID: 38926482 Free PMC article.

10

Small-molecule suppression of β-lactam resistance in multidrug-resistant gram-negative pathogens.

Brackett CM, Melander RJ, An IH, Krishnamurthy A, Thompson RJ, Cavanagh J, Melander C. Brackett CM, et al. J Med Chem. 2014 Sep 11;57(17):7450-8. doi: 10.1021/jm501050e. Epub 2014 Aug 28. J Med Chem. 2014. PMID: 25137478

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