Sleebs BE - Search Results

1

Design and characterization of a heterobifunctional degrader of KEAP1.

Chen H, Nguyen NH, Magtoto CM, Cobbold SA, Bidgood GM, Meza Guzman LG, Richardson LW, Corbin J, Au AE, Lechtenberg BC, Feltham R, Sutherland KD, Grohmann C, Nicholson SE, Sleebs BE. Chen H, et al. Among authors: sleebs be. Redox Biol. 2023 Feb;59:102552. doi: 10.1016/j.redox.2022.102552. Epub 2022 Nov 26. Redox Biol. 2023. PMID: 36473314 Free PMC article.

2

Diastereoselective synthesis of alpha-methyl and alpha-hydroxy-beta-amino acids via 4-substituted-1,3-oxazinan-6-ones.

Sleebs BE, Hughes AB. Sleebs BE, et al. J Org Chem. 2007 Apr 27;72(9):3340-52. doi: 10.1021/jo0700326. Epub 2007 Apr 3. J Org Chem. 2007. PMID: 17402786

3

M2, a novel anthracenedione, elicits a potent DNA damage response that can be subverted through checkpoint kinase inhibition to generate mitotic catastrophe.

Evison BJ, Pastuovic M, Bilardi RA, Forrest RA, Pumuye PP, Sleebs BE, Watson KG, Phillips DR, Cutts SM. Evison BJ, et al. Among authors: sleebs be. Biochem Pharmacol. 2011 Dec 1;82(11):1604-18. doi: 10.1016/j.bcp.2011.08.013. Epub 2011 Aug 30. Biochem Pharmacol. 2011. PMID: 21889927

4

Synthetic Kavalactone Analogues with Increased Potency and Selective Anthelmintic Activity against Larvae of Haemonchus contortus In Vitro.

Herath HMPD, Taki AC, Nguyen N, Garcia-Bustos J, Hofmann A, Wang T, Ma G, Chang BCH, Jabbar A, Sleebs BE, Gasser RB. Herath HMPD, et al. Among authors: sleebs be. Molecules. 2020 Apr 24;25(8):2004. doi: 10.3390/molecules25082004. Molecules. 2020. PMID: 32344703 Free PMC article.

5

Advances in the discovery and development of anthelmintics by harnessing natural product scaffolds.

Herath HMPD, Taki AC, Sleebs BE, Hofmann A, Nguyen N, Preston S, Davis RA, Jabbar A, Gasser RB. Herath HMPD, et al. Among authors: sleebs be. Adv Parasitol. 2021;111:203-251. doi: 10.1016/bs.apar.2020.10.002. Epub 2021 Jan 8. Adv Parasitol. 2021. PMID: 33482975 Review.

6

Late Stage Phosphotyrosine Mimetic Functionalization of Peptides Employing Metallaphotoredox Catalysis.

Chen H, Mao R, Brzozowski M, Nguyen NH, Sleebs BE. Chen H, et al. Among authors: sleebs be. Org Lett. 2021 Jun 4;23(11):4244-4249. doi: 10.1021/acs.orglett.1c01200. Epub 2021 May 24. Org Lett. 2021. PMID: 34029466

7

High-Throughput Phenotypic Assay to Screen for Anthelmintic Activity on Haemonchus contortus.

Taki AC, Byrne JJ, Wang T, Sleebs BE, Nguyen N, Hall RS, Korhonen PK, Chang BCH, Jackson P, Jabbar A, Gasser RB. Taki AC, et al. Among authors: sleebs be. Pharmaceuticals (Basel). 2021 Jun 26;14(7):616. doi: 10.3390/ph14070616. Pharmaceuticals (Basel). 2021. PMID: 34206910 Free PMC article.

8

Optimization of Phosphotyrosine Peptides that Target the SH2 Domain of SOCS1 and Block Substrate Ubiquitination.

Chen H, Wu Y, Li K, Currie I, Keating N, Dehkhoda F, Grohmann C, Babon JJ, Nicholson SE, Sleebs BE. Chen H, et al. Among authors: sleebs be. ACS Chem Biol. 2022 Feb 18;17(2):449-462. doi: 10.1021/acschembio.1c00884. Epub 2022 Jan 6. ACS Chem Biol. 2022. PMID: 34989544

9

A High-Throughput Phenotypic Screen of the 'Pandemic Response Box' Identifies a Quinoline Derivative with Significant Anthelmintic Activity.

Shanley HT, Taki AC, Byrne JJ, Jabbar A, Wells TNC, Samby K, Boag PR, Nguyen N, Sleebs BE, Gasser RB. Shanley HT, et al. Among authors: sleebs be. Pharmaceuticals (Basel). 2022 Feb 21;15(2):257. doi: 10.3390/ph15020257. Pharmaceuticals (Basel). 2022. PMID: 35215369 Free PMC article.

10

Substrate Peptidomimetic Inhibitors of P. falciparum Plasmepsin X with Potent Antimalarial Activity.

Richardson LW, Ashton TD, Dans MG, Nguyen N, Favuzza P, Triglia T, Hodder AN, Ngo A, Jarman KE, Cowman AF, Sleebs BE. Richardson LW, et al. Among authors: sleebs be. ChemMedChem. 2022 Sep 16;17(18):e202200306. doi: 10.1002/cmdc.202200306. Epub 2022 Aug 18. ChemMedChem. 2022. PMID: 35906744 Free PMC article.

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