Maklad RM - Search Results

1

Development of novel isatin thiazolyl-pyrazoline hybrids as promising antimicrobials in MDR pathogens.

Al-Warhi T, Elimam DM, Elsayed ZM, Abdel-Aziz MM, Maklad RM, Al-Karmalawy AA, Afarinkia K, Abourehab MAS, Abdel-Aziz HA, Eldehna WM. Al-Warhi T, et al. Among authors: maklad rm. RSC Adv. 2022 Nov 2;12(48):31466-31477. doi: 10.1039/d2ra04385h. eCollection 2022 Oct 27. RSC Adv. 2022. PMID: 36382148 Free PMC article.

2

Development of 3-methyl/3-(morpholinomethyl)benzofuran derivatives as novel antitumor agents towards non-small cell lung cancer cells.

Al-Sanea MM, Al-Ansary GH, Elsayed ZM, Maklad RM, Elkaeed EB, Abdelgawad MA, Bukhari SNA, Abdel-Aziz MM, Suliman H, Eldehna WM. Al-Sanea MM, et al. Among authors: maklad rm. J Enzyme Inhib Med Chem. 2021 Dec;36(1):987-999. doi: 10.1080/14756366.2021.1915302. J Enzyme Inhib Med Chem. 2021. PMID: 33985397 Free PMC article.

3

Identification of 3-(piperazinylmethyl)benzofuran derivatives as novel type II CDK2 inhibitors: design, synthesis, biological evaluation, and in silico insights.

Eldehna WM, Maklad RM, Almahli H, Al-Warhi T, Elkaeed EB, Abourehab MAS, Abdel-Aziz HA, El Kerdawy AM. Eldehna WM, et al. Among authors: maklad rm. J Enzyme Inhib Med Chem. 2022 Dec;37(1):1227-1240. doi: 10.1080/14756366.2022.2062337. J Enzyme Inhib Med Chem. 2022. PMID: 35470754 Free PMC article.

4

1-Benzyl-5-bromo-3-hydrazonoindolin-2-ones as Novel Anticancer Agents: Synthesis, Biological Evaluation and Molecular Modeling Insights.

Al-Warhi T, Almahli H, Maklad RM, Elsayed ZM, El Hassab MA, Alotaibi OJ, Aljaeed N, Ayyad RR, Ghabour HA, Eldehna WM, El-Ashrey MK. Al-Warhi T, et al. Among authors: maklad rm. Molecules. 2023 Apr 4;28(7):3203. doi: 10.3390/molecules28073203. Molecules. 2023. PMID: 37049966 Free PMC article.

5

Tetrahydrobenzo[h]quinoline derivatives as a novel chemotype for dual antileishmanial-antimalarial activity graced with antitubercular activity: Design, synthesis and biological evaluation.

Ibrahim TM, Abada G, Dammann M, Maklad RM, Eldehna WM, Salem R, Abdelaziz MM, El-Domany RA, Bekhit AA, Beockler FM. Ibrahim TM, et al. Among authors: maklad rm. Eur J Med Chem. 2023 Sep 5;257:115534. doi: 10.1016/j.ejmech.2023.115534. Epub 2023 May 29. Eur J Med Chem. 2023. PMID: 37269671

6

Thieno[2,3-c]isoquinolines: A novel chemotype of antiproliferative agents inducing cellular apoptosis while targeting the G2/M phase and Tubulin.

Marae IS, Maklad RM, Samir S, Bakhite EA, Sharmoukh W. Marae IS, et al. Among authors: maklad rm. Drug Dev Res. 2023 Jun;84(4):747-766. doi: 10.1002/ddr.22054. Epub 2023 Mar 31. Drug Dev Res. 2023. PMID: 36999479

7

Synthesis, cytotoxicity, docking study, and tubulin polymerization inhibitory activity of novel 1-(3,4-dimethoxyphenyl)-5-(3,4,5-trimethoxyphenyl)-1H-1,2,4-triazole-3-carboxanilides.

Aly OM, Beshr EA, Maklad RM, Mustafa M, Gamal-Eldeen AM. Aly OM, et al. Among authors: maklad rm. Arch Pharm (Weinheim). 2014 Sep;347(9):658-67. doi: 10.1002/ardp.201400096. Epub 2014 Jul 3. Arch Pharm (Weinheim). 2014. PMID: 24996189

8

Tubulin inhibitors: Discovery of a new scaffold targeting extra-binding residues within the colchicine site through anchoring substituents properly adapted to their pocket by a semi-flexible linker.

Maklad RM, AbdelHafez EMN, Abdelhamid D, Aly OM. Maklad RM, et al. Bioorg Chem. 2020 Jun;99:103767. doi: 10.1016/j.bioorg.2020.103767. Epub 2020 Apr 6. Bioorg Chem. 2020. PMID: 32325332

9

Trapping Anions within Stacks of Tetra-Urea Macrocycles.

Li J, Catal O, Marques I, McNaughton DA, Maklad RM, Ryder WG, Hill MJS, Seddon A, Lewis W, Adams DJ, Félix V, Wu X, Gale PA. Li J, et al. Among authors: maklad rm. J Am Chem Soc. 2025 Jan 29;147(4):3392-3401. doi: 10.1021/jacs.4c14194. Epub 2025 Jan 13. J Am Chem Soc. 2025. PMID: 39805740

10

Design, synthesis, and in silico insights of novel N'-(2-oxoindolin-3-ylidene)piperidine-4-carbohydrazide derivatives as VEGFR-2 inhibitors.

Eldehna WM, Habib YA, Mahmoud AE, Barghash MF, Elsayed ZM, Elsawi AE, Maklad RM, Rashed M, Khalil A, Hammad SF, Ali MM, El Kerdawy AM. Eldehna WM, et al. Among authors: maklad rm. Bioorg Chem. 2024 Dec;153:107829. doi: 10.1016/j.bioorg.2024.107829. Epub 2024 Sep 18. Bioorg Chem. 2024. PMID: 39317037

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