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Page 1
Mechanistic understanding of human SLFN11.
Metzner FJ, Wenzl SJ, Kugler M, Krebs S, Hopfner KP, Lammens K. Metzner FJ, et al. Among authors: kugler m. Nat Commun. 2022 Sep 17;13(1):5464. doi: 10.1038/s41467-022-33123-0. Nat Commun. 2022. PMID: 36115853 Free PMC article.
Direct Introduction of an Alkylsulfonamido Group on C-sites of Isomeric Dicarba-closo-dodecaboranes: The Influence of Stereochemistry on Inhibitory Activity against the Cancer-Associated Carbonic Anhydrase IX Isoenzyme.
Nekvinda J, Kugler M, Holub J, El Anwar S, Brynda J, Pospíšilová K, Růžičková Z, Řezáčová P, Grüner B. Nekvinda J, et al. Among authors: kugler m. Chemistry. 2020 Dec 9;26(69):16541-16553. doi: 10.1002/chem.202002809. Epub 2020 Nov 3. Chemistry. 2020. PMID: 32757220
X-ray structure of human aldo-keto reductase 1C3 in complex with a bile acid fused tetrazole inhibitor: experimental validation, molecular docking and structural analysis.
Marinović MA, Bekić SS, Kugler M, Brynda J, Škerlová J, Škorić DĐ, Řezáčová P, Petri ET, Ćelić AS. Marinović MA, et al. Among authors: kugler m. RSC Med Chem. 2022 Dec 1;14(2):341-355. doi: 10.1039/d2md00387b. eCollection 2023 Feb 22. RSC Med Chem. 2022. PMID: 36846371 Free PMC article.
Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX.
Grüner B, Brynda J, Das V, Šícha V, Štěpánková J, Nekvinda J, Holub J, Pospíšilová K, Fábry M, Pachl P, Král V, Kugler M, Mašek V, Medvedíková M, Matějková S, Nová A, Lišková B, Gurská S, Džubák P, Hajdúch M, Řezáčová P. Grüner B, et al. Among authors: kugler m. J Med Chem. 2019 Nov 14;62(21):9560-9575. doi: 10.1021/acs.jmedchem.9b00945. Epub 2019 Oct 16. J Med Chem. 2019. PMID: 31568723
Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX.
Dvořanová J, Kugler M, Holub J, Šícha V, Das V, Nekvinda J, El Anwar S, Havránek M, Pospíšilová K, Fábry M, Král V, Medvedíková M, Matějková S, Lišková B, Gurská S, Džubák P, Brynda J, Hajdúch M, Grüner B, Řezáčová P. Dvořanová J, et al. Among authors: kugler m. Eur J Med Chem. 2020 Aug 15;200:112460. doi: 10.1016/j.ejmech.2020.112460. Epub 2020 May 18. Eur J Med Chem. 2020. PMID: 32505851
Identification of Novel Carbonic Anhydrase IX Inhibitors Using High-Throughput Screening of Pooled Compound Libraries by DNA-Linked Inhibitor Antibody Assay (DIANA).
Tykvart J, Navrátil V, Kugler M, Šácha P, Schimer J, Hlaváčková A, Tenora L, Zemanová J, Dejmek M, Král V, Potáček M, Majer P, Jahn U, Brynda J, Řezáčová P, Konvalinka J. Tykvart J, et al. Among authors: kugler m. SLAS Discov. 2020 Oct;25(9):1026-1037. doi: 10.1177/2472555220918836. Epub 2020 May 26. SLAS Discov. 2020. PMID: 32452709 Free article.
113 results