Spetea M - Search Results

1

In Vitro, In Vivo and In Silico Characterization of a Novel Kappa-Opioid Receptor Antagonist.

Puls K, Olivé-Marti AL, Pach S, Pinter B, Erli F, Wolber G, Spetea M. Puls K, et al. Among authors: spetea m. Pharmaceuticals (Basel). 2022 May 28;15(6):680. doi: 10.3390/ph15060680. Pharmaceuticals (Basel). 2022. PMID: 35745598 Free PMC article.

2

Morphinans and isoquinolines: acetylcholinesterase inhibition, pharmacophore modeling, and interaction with opioid receptors.

Schuster D, Spetea M, Music M, Rief S, Fink M, Kirchmair J, Schütz J, Wolber G, Langer T, Stuppner H, Schmidhammer H, Rollinger JM. Schuster D, et al. Among authors: spetea m. Bioorg Med Chem. 2010 Jul 15;18(14):5071-80. doi: 10.1016/j.bmc.2010.05.071. Epub 2010 Jun 2. Bioorg Med Chem. 2010. PMID: 20580236

3

Current κ opioid receptor ligands and discovery of a new molecular scaffold as a κ opioid receptor antagonist using pharmacophore-based virtual screening.

Spetea M, Asim MF, Noha S, Wolber G, Schmidhammer H. Spetea M, et al. Curr Pharm Des. 2013;19(42):7362-72. doi: 10.2174/138161281942140105162601. Curr Pharm Des. 2013. PMID: 23448472

4

The µ opioid receptor and ligands acting at the µ opioid receptor, as therapeutics and potential therapeutics.

Spetea M, Asim MF, Wolber G, Schmidhammer H. Spetea M, et al. Curr Pharm Des. 2013;19(42):7415-34. doi: 10.2174/13816128113199990362. Curr Pharm Des. 2013. PMID: 23448479 Review.

5

μ Opioid receptor: novel antagonists and structural modeling.

Kaserer T, Lantero A, Schmidhammer H, Spetea M, Schuster D. Kaserer T, et al. Among authors: spetea m. Sci Rep. 2016 Feb 18;6:21548. doi: 10.1038/srep21548. Sci Rep. 2016. PMID: 26888328 Free PMC article.

6

Structural determinants of diphenethylamines for interaction with the κ opioid receptor: Synthesis, pharmacology and molecular modeling studies.

Guerrieri E, Bermudez M, Wolber G, Berzetei-Gurske IP, Schmidhammer H, Spetea M. Guerrieri E, et al. Among authors: spetea m. Bioorg Med Chem Lett. 2016 Oct 1;26(19):4769-4774. doi: 10.1016/j.bmcl.2016.08.031. Epub 2016 Aug 12. Bioorg Med Chem Lett. 2016. PMID: 27567368

7

Highly Potent and Selective New Diphenethylamines Interacting with the κ-Opioid Receptor: Synthesis, Pharmacology, and Structure-Activity Relationships.

Erli F, Guerrieri E, Ben Haddou T, Lantero A, Mairegger M, Schmidhammer H, Spetea M. Erli F, et al. Among authors: spetea m. J Med Chem. 2017 Sep 14;60(17):7579-7590. doi: 10.1021/acs.jmedchem.7b00981. Epub 2017 Aug 30. J Med Chem. 2017. PMID: 28825813 Free PMC article.

8

In vitro and in vivo Pharmacological Activities of 14-O-Phenylpropyloxymorphone, a Potent Mixed Mu/Delta/Kappa-Opioid Receptor Agonist With Reduced Constipation in Mice.

Lattanzi R, Rief S, Schmidhammer H, Negri L, Spetea M. Lattanzi R, et al. Among authors: spetea m. Front Pharmacol. 2018 Aug 31;9:1002. doi: 10.3389/fphar.2018.01002. eCollection 2018. Front Pharmacol. 2018. PMID: 30233377 Free PMC article.

9

N-Phenethyl Substitution in 14-Methoxy-N-methylmorphinan-6-ones Turns Selective µ Opioid Receptor Ligands into Dual µ/δ Opioid Receptor Agonists.

Dumitrascuta M, Bermudez M, Ben Haddou T, Guerrieri E, Schläfer L, Ritsch A, Hosztafi S, Lantero A, Kreutz C, Massotte D, Schmidhammer H, Wolber G, Spetea M. Dumitrascuta M, et al. Among authors: spetea m. Sci Rep. 2020 Mar 27;10(1):5653. doi: 10.1038/s41598-020-62530-w. Sci Rep. 2020. PMID: 32221355 Free PMC article.

10

Mechanistic Understanding of Peptide Analogues, DALDA, [Dmt¹]DALDA, and KGOP01, Binding to the mu Opioid Receptor.

Dumitrascuta M, Bermudez M, Ballet S, Wolber G, Spetea M. Dumitrascuta M, et al. Among authors: spetea m. Molecules. 2020 Apr 29;25(9):2087. doi: 10.3390/molecules25092087. Molecules. 2020. PMID: 32365707 Free PMC article.

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