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Page 1
Design of Development Candidate eFT226, a First in Class Inhibitor of Eukaryotic Initiation Factor 4A RNA Helicase.
Ernst JT, Thompson PA, Nilewski C, Sprengeler PA, Sperry S, Packard G, Michels T, Xiang A, Tran C, Wegerski CJ, Eam B, Young NP, Fish S, Chen J, Howard H, Staunton J, Molter J, Clarine J, Nevarez A, Chiang GG, Appleman JR, Webster KR, Reich SH. Ernst JT, et al. Among authors: fish s. J Med Chem. 2020 Jun 11;63(11):5879-5955. doi: 10.1021/acs.jmedchem.0c00182. Epub 2020 May 29. J Med Chem. 2020. PMID: 32470302
Targeting Oncogene mRNA Translation in B-Cell Malignancies with eFT226, a Potent and Selective Inhibitor of eIF4A.
Thompson PA, Eam B, Young NP, Fish S, Chen J, Barrera M, Howard H, Sung E, Parra A, Staunton J, Chiang GG, Gerson-Gurwitz A, Wegerski CJ, Nevarez A, Clarine J, Sperry S, Xiang A, Nilewski C, Packard GK, Michels T, Tran C, Sprengeler PA, Ernst JT, Reich SH, Webster KR. Thompson PA, et al. Among authors: fish s. Mol Cancer Ther. 2021 Jan;20(1):26-36. doi: 10.1158/1535-7163.MCT-19-0973. Epub 2020 Oct 9. Mol Cancer Ther. 2021. PMID: 33037136
1-Aminomethyl SAR in a novel series of flavagline-inspired eIF4A inhibitors: Effects of amine substitution on cell potency and in vitro PK properties.
Nilewski C, Michels TD, Packard GK, Xiang AX, Sprengeler PA, Eam B, Fish S, Thompson PA, Wegerski CJ, Nevarez A, Clarine J, Sperry S, Ernst JT, Reich SH. Nilewski C, et al. Among authors: fish s. Bioorg Med Chem Lett. 2021 Sep 1;47:128111. doi: 10.1016/j.bmcl.2021.128111. Epub 2021 Aug 2. Bioorg Med Chem Lett. 2021. PMID: 34353608
Discovery of Monovalent Direct Degraders of BRD4 That Act Via the Recruitment of DCAF11.
Parker GS, Toth JI, Fish S, Blanco GA, Kampert T, Li X, Yang L, Stumpf CR, Steadman K, Jamborcic A, Chien S, Daniele E, Dearie A, Leriche G, Bailey S, Thompson PA. Parker GS, et al. Among authors: fish s. Mol Cancer Ther. 2024 Jun 22. doi: 10.1158/1535-7163.MCT-24-0219. Online ahead of print. Mol Cancer Ther. 2024. PMID: 38907538
Discovery of Monovalent Direct Degraders of BRD4 that Act via the Recruitment of DCAF11.
Parker GS, Toth JI, Fish S, Blanco G, Kampert T, Li X, Yang L, Stumpf CR, Steadman K, Jamborcic A, Chien S, Daniele E, Dearie A, Leriche G, Bailey S, Thompson PA. Parker GS, et al. Among authors: fish s. Mol Cancer Ther. 2024 Jul 5:OF1-OF13. doi: 10.1158/1535-7163.MCT-24-0219. Online ahead of print. Mol Cancer Ther. 2024. PMID: 38967115
Anti-miRs competitively inhibit microRNAs in Argonaute complexes.
Hogan DJ, Vincent TM, Fish S, Marcusson EG, Bhat B, Chau BN, Zisoulis DG. Hogan DJ, et al. Among authors: fish s. PLoS One. 2014 Jul 3;9(7):e100951. doi: 10.1371/journal.pone.0100951. eCollection 2014. PLoS One. 2014. PMID: 24992387 Free PMC article.
316 results