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Page 1
Pharmacological characterization of GLPG1972/S201086, a potent and selective small-molecule inhibitor of ADAMTS5.
Clement-Lacroix P, Little CB, Smith MM, Cottereaux C, Merciris D, Meurisse S, Mollat P, Touitou R, Brebion F, Gosmini R, De Ceuninck F, Botez I, Lepescheux L, van der Aar E, Christophe T, Vandervoort N, Blanqué R, Comas D, Deprez P, Amantini D. Clement-Lacroix P, et al. Among authors: brebion f. Osteoarthritis Cartilage. 2022 Feb;30(2):291-301. doi: 10.1016/j.joca.2021.08.012. Epub 2021 Oct 6. Osteoarthritis Cartilage. 2022. PMID: 34626798 Free article.
Discovery of GLPG1972/S201086, a Potent, Selective, and Orally Bioavailable ADAMTS-5 Inhibitor for the Treatment of Osteoarthritis.
Brebion F, Gosmini R, Deprez P, Varin M, Peixoto C, Alvey L, Jary H, Bienvenu N, Triballeau N, Blanque R, Cottereaux C, Christophe T, Vandervoort N, Mollat P, Touitou R, Leonard P, De Ceuninck F, Botez I, Monjardet A, van der Aar E, Amantini D. Brebion F, et al. J Med Chem. 2021 Mar 25;64(6):2937-2952. doi: 10.1021/acs.jmedchem.0c02008. Epub 2021 Mar 15. J Med Chem. 2021. PMID: 33719441 Free article.
Conjugate additions to alkylidene bis(sulfoxides).
Brebion F, Vincent G, Chelli S, Kwasnieski O, Najera F, Delouvrié B, Marek I, Derat E, Goddard JP, Malacria M, Fensterbank L. Brebion F, et al. Chem Asian J. 2011 Jul 4;6(7):1825-33. doi: 10.1002/asia.201000904. Epub 2011 Mar 11. Chem Asian J. 2011. PMID: 21400664
Dechalcogenative allylic selenosulfide and disulfide rearrangements: complementary methods for the formation of allylic sulfides in the absence of electrophiles. Scope, limitations, and application to the functionalization of unprotected peptides in aqueous media.
Crich D, Krishnamurthy V, Brebion F, Karatholuvhu M, Subramanian V, Hutton TK. Crich D, et al. Among authors: brebion f. J Am Chem Soc. 2007 Aug 22;129(33):10282-94. doi: 10.1021/ja072969u. Epub 2007 Jul 27. J Am Chem Soc. 2007. PMID: 17655306 Free PMC article.