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Structural design, synthesis and anti-Trypanosoma cruzi profile of the second generation of 4-thiazolidinones chlorine derivatives.
Bezerra de Oliveira Filho G, Veríssimo de Oliveira Cardoso M, Caroline da Silva Santos A, Ramos Dos Santos TA, Cristovão-Silva AC, Rubio LG, da Silva Maia Neto L, Leite PG, Machado FS, Alves LC, Brayner FA, Alves Pereira VR, Lima Leite AC. Bezerra de Oliveira Filho G, et al. Among authors: leite pg, lima leite ac. Chem Biol Interact. 2021 Aug 25;345:109514. doi: 10.1016/j.cbi.2021.109514. Epub 2021 May 21. Chem Biol Interact. 2021. PMID: 34023282
Dual Parasiticidal Activities of Phthalimides: Synthesis and Biological Profile against Trypanosoma cruzi and Plasmodium falciparum.
Teixeira de Moraes Gomes PA, Veríssimo de Oliveira Cardoso M, Dos Santos IR, Amaro de Sousa F, da Conceição JM, Gouveia de Melo Silva V, Duarte D, Pereira R, Oliveira R, Nogueira F, Alves LC, Brayner FA, da Silva Santos AC, Rêgo Alves Pereira V, Lima Leite AC. Teixeira de Moraes Gomes PA, et al. Among authors: lima leite ac. ChemMedChem. 2020 Nov 18;15(22):2164-2175. doi: 10.1002/cmdc.202000331. Epub 2020 Oct 19. ChemMedChem. 2020. PMID: 32813331
Structural improvement of new thiazolyl-isatin derivatives produces potent and selective trypanocidal and leishmanicidal compounds.
Barros Freitas LA, Caroline da Silva Santos A, de Cássia Silva G, Nayara do Nascimento Albuquerque F, Silva ED, Alberto de Simone C, Alves Pereira VR, Alves LC, Brayner FA, Lima Leite AC, de Moraes Gomes PAT. Barros Freitas LA, et al. Among authors: lima leite ac. Chem Biol Interact. 2021 Aug 25;345:109561. doi: 10.1016/j.cbi.2021.109561. Epub 2021 Jun 24. Chem Biol Interact. 2021. PMID: 34174251
Structural design, synthesis and pharmacological evaluation of 4-thiazolidinones against Trypanosoma cruzi.
de Oliveira Filho GB, de Oliveira Cardoso MV, Espíndola JW, Ferreira LF, de Simone CA, Ferreira RS, Coelho PL, Meira CS, Magalhaes Moreira DR, Soares MB, Lima Leite AC. de Oliveira Filho GB, et al. Among authors: lima leite ac. Bioorg Med Chem. 2015 Dec 1;23(23):7478-86. doi: 10.1016/j.bmc.2015.10.048. Epub 2015 Nov 2. Bioorg Med Chem. 2015. PMID: 26549870 Free article.
Synthesis of 4'-(2-ferrocenyl)-2,2':6'2''-terpyridine: characterization and antiprotozoal activity of Mn(II), Co(II), Ni(II), Cu(II) and Zn(II) complexes.
Juneja A, Macedo TS, Magalhaes Moreira DR, Pereira Soares MB, Lima Leite AC, Kelle de Andrade Lemoine Neves J, Alves Pereira VR, Avecilla F, Azam A. Juneja A, et al. Among authors: lima leite ac. Eur J Med Chem. 2014 Mar 21;75:203-10. doi: 10.1016/j.ejmech.2014.01.051. Epub 2014 Jan 31. Eur J Med Chem. 2014. PMID: 24534536
Study of acute oral toxicity of the thiazole derivative N-(1-methyl-2-methyl-pyridine)-N-(p-bromophenylthiazol-2-yl)-hydrazine in a Syrian hamster.
Vasconcelos Gomes de Oliveira V, Angela Aranda de Souza M, Ramos Mororó Cavalcanti R, Veríssimo de Oliveira Cardoso M, Lima Leite AC, de Figueiredo RCBQ, Rogério de Freitas Silva S, Câmara Alves L, Amaro da Silva Junior V. Vasconcelos Gomes de Oliveira V, et al. Among authors: lima leite ac. Toxicol Mech Methods. 2021 Mar;31(3):197-204. doi: 10.1080/15376516.2020.1867681. Epub 2021 Jan 11. Toxicol Mech Methods. 2021. PMID: 33349088
The prophylactic and anti-fibrotic activity of phthalimido-thiazole derivatives in schistosomiasis mansoni.
Laranjeira Miranda Filho CA, de Oliveira Barbosa M, Rodrigues Oliveira A, Ferreira Pinto A, Araújo DL, Lucena JP, de Araújo RE, de Oliveira SA, Lima Leite AC. Laranjeira Miranda Filho CA, et al. Among authors: lima leite ac. Parasitol Res. 2022 Jul;121(7):2111-2120. doi: 10.1007/s00436-022-07533-4. Epub 2022 May 23. Parasitol Res. 2022. PMID: 35599272
28 results