Gust R - Search Results

1

Heterodimeric GW7604 Derivatives: Modification of the Pharmacological Profile by Additional Interactions at the Coactivator Binding Site.

Knox AK, Kalchschmid C, Schuster D, Gaggia F, Gust R. Knox AK, et al. Among authors: gust r. J Med Chem. 2021 May 13;64(9):5766-5786. doi: 10.1021/acs.jmedchem.0c02230. Epub 2021 Apr 27. J Med Chem. 2021. PMID: 33904307 Free PMC article.

2

Synthesis, structural evaluation, and estrogen receptor interaction of 2,3-diarylpiperazines.

Gust R, Keilitz R, Schmidt K. Gust R, et al. J Med Chem. 2002 May 23;45(11):2325-37. doi: 10.1021/jm0208368. J Med Chem. 2002. PMID: 12014971

3

(4R,5S)/(4S,5R)-4,5-Bis(4-hydroxyphenyl)-2-imidazolines: ligands for the estrogen receptor with a novel binding mode.

Gust R, Keilitz R, Schmidt K, von Rauch M. Gust R, et al. J Med Chem. 2002 Aug 1;45(16):3356-65. doi: 10.1021/jm020809h. J Med Chem. 2002. PMID: 12139447

4

Investigations on estrogen receptor binding. The estrogenic, antiestrogenic, and cytotoxic properties of C2-alkyl-substituted 1,1-bis(4-hydroxyphenyl)-2-phenylethenes.

Lubczyk V, Bachmann H, Gust R. Lubczyk V, et al. Among authors: gust r. J Med Chem. 2002 Nov 21;45(24):5358-64. doi: 10.1021/jm0209230. J Med Chem. 2002. PMID: 12431063

5

Antiestrogenically active 1,1,2-tris(4-hydroxyphenyl)alkenes without basic side chain: synthesis and biological activity.

Lubczyk V, Bachmann H, Gust R. Lubczyk V, et al. Among authors: gust r. J Med Chem. 2003 Apr 10;46(8):1484-91. doi: 10.1021/jm0210562. J Med Chem. 2003. PMID: 12672249

6

Effects of C2-alkylation, N-alkylation, and N,N'-dialkylation on the stability and estrogen receptor interaction of (4R,5S)/(4S,5R)-4,5-bis(4-hydroxyphenyl)-2-imidazolines.

von Rauch M, Schlenk M, Gust R. von Rauch M, et al. Among authors: gust r. J Med Chem. 2004 Feb 12;47(4):915-27. doi: 10.1021/jm0309809. J Med Chem. 2004. PMID: 14761193

7

Investigations on the effects of basic side chains on the hormonal profile of (4R,5S)/(4S,5R)-4,5-bis(4-hydroxyphenyl)-2-imidazolines.

von Rauch M, Busch S, Gust R. von Rauch M, et al. Among authors: gust r. J Med Chem. 2005 Jan 27;48(2):466-74. doi: 10.1021/jm040855c. J Med Chem. 2005. PMID: 15658860

8

Synthesis and pharmacological evaluation of 1H-imidazoles as ligands for the estrogen receptor and cytotoxic inhibitors of the cyclooxygenase.

Wiglenda T, Ott I, Kircher B, Schumacher P, Schuster D, Langer T, Gust R. Wiglenda T, et al. Among authors: gust r. J Med Chem. 2005 Oct 6;48(20):6516-21. doi: 10.1021/jm050190u. J Med Chem. 2005. PMID: 16190777

9

Structure-activity relationship study to understand the estrogen receptor-dependent gene activation of aryl- and alkyl-substituted 1H-imidazoles.

Wiglenda T, Gust R. Wiglenda T, et al. Among authors: gust r. J Med Chem. 2007 Apr 5;50(7):1475-84. doi: 10.1021/jm061106t. Epub 2007 Mar 13. J Med Chem. 2007. PMID: 17352461

10

Cobalt-alkyne complexes with imidazoline ligands as estrogenic carriers: synthesis and pharmacological investigations.

Schlenk M, Ott I, Gust R. Schlenk M, et al. Among authors: gust r. J Med Chem. 2008 Nov 27;51(22):7318-22. doi: 10.1021/jm8008376. J Med Chem. 2008. PMID: 18942824

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