Schweipert M - Search Results

1

Permuted 2,4-thiazolidinedione (TZD) analogs as GLUT inhibitors and their in-vitro evaluation in leukemic cells.

Tilekar K, Upadhyay N, Schweipert M, Hess JD, Macias LH, Mrowka P, Meyer-Almes FJ, Aguilera RJ, Iancu CV, Choe JY, Ramaa CS. Tilekar K, et al. Among authors: schweipert m. Eur J Pharm Sci. 2020 Nov 1;154:105512. doi: 10.1016/j.ejps.2020.105512. Epub 2020 Aug 12. Eur J Pharm Sci. 2020. PMID: 32801003 Free PMC article.

2

Discovery of 5-naphthylidene-2,4-thiazolidinedione derivatives as selective HDAC8 inhibitors and evaluation of their cytotoxic effects in leukemic cell lines.

Tilekar K, Upadhyay N, Jänsch N, Schweipert M, Mrowka P, Meyer-Almes FJ, Ramaa CS. Tilekar K, et al. Among authors: schweipert m. Bioorg Chem. 2020 Jan;95:103522. doi: 10.1016/j.bioorg.2019.103522. Epub 2019 Dec 18. Bioorg Chem. 2020. PMID: 31901516

3

Discovery of novel N-substituted thiazolidinediones (TZDs) as HDAC8 inhibitors: in-silico studies, synthesis, and biological evaluation.

Upadhyay N, Tilekar K, Jänsch N, Schweipert M, Hess JD, Henze Macias L, Mrowka P, Aguilera RJ, Choe JY, Meyer-Almes FJ, Ramaa CS. Upadhyay N, et al. Among authors: schweipert m. Bioorg Chem. 2020 Jul;100:103934. doi: 10.1016/j.bioorg.2020.103934. Epub 2020 May 15. Bioorg Chem. 2020. PMID: 32446120 Free PMC article.

4

Thiazolidinedione "Magic Bullets" Simultaneously Targeting PPARγ and HDACs: Design, Synthesis, and Investigations of their In Vitro and In Vivo Antitumor Effects.

Tilekar K, Hess JD, Upadhyay N, Bianco AL, Schweipert M, Laghezza A, Loiodice F, Meyer-Almes FJ, Aguilera RJ, Lavecchia A, C S R. Tilekar K, et al. Among authors: schweipert m. J Med Chem. 2021 May 27;64(10):6949-6971. doi: 10.1021/acs.jmedchem.1c00491. Epub 2021 May 18. J Med Chem. 2021. PMID: 34006099 Free PMC article.

5

Double-edged Swords: Diaryl pyrazoline thiazolidinediones synchronously targeting cancer epigenetics and angiogenesis.

Upadhyay N, Tilekar K, Safuan S, Kumar AP, Schweipert M, Meyer-Almes FJ, Ramaa CS. Upadhyay N, et al. Among authors: schweipert m. Bioorg Chem. 2021 Nov;116:105350. doi: 10.1016/j.bioorg.2021.105350. Epub 2021 Sep 11. Bioorg Chem. 2021. PMID: 34547645

6

Development and investigation of thiazolidinedione and pyrazoline compounds as antiangiogenic weapons targeting VEGFR-2.

Upadhyay N, Tilekar K, Safuan S, Kumar AP, Schweipert M, Meyer-Almes FJ, Ramaa CS. Upadhyay N, et al. Among authors: schweipert m. Future Med Chem. 2021 Nov;13(22):1963-1986. doi: 10.4155/fmc-2021-0139. Epub 2021 Sep 28. Future Med Chem. 2021. PMID: 34581188

7

Multi-target weapons: diaryl-pyrazoline thiazolidinediones simultaneously targeting VEGFR-2 and HDAC cancer hallmarks.

Upadhyay N, Tilekar K, Safuan S, Kumar AP, Schweipert M, Meyer-Almes FJ, C S R. Upadhyay N, et al. Among authors: schweipert m. RSC Med Chem. 2021 Jul 27;12(9):1540-1554. doi: 10.1039/d1md00125f. eCollection 2021 Sep 23. RSC Med Chem. 2021. PMID: 34671737 Free PMC article.

8

Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4.

Schweipert M, Jänsch N, Upadhyay N, Tilekar K, Wozny E, Basheer S, Wurster E, Müller M, C S R, Meyer-Almes FJ. Schweipert M, et al. Pharmaceuticals (Basel). 2021 Oct 11;14(10):1032. doi: 10.3390/ph14101032. Pharmaceuticals (Basel). 2021. PMID: 34681256 Free PMC article.

9

Kinetically selective and potent inhibitors of HDAC8.

Schweipert M, Jänsch N, Sugiarto WO, Meyer-Almes FJ. Schweipert M, et al. Biol Chem. 2019 May 27;400(6):733-743. doi: 10.1515/hsz-2018-0363. Biol Chem. 2019. PMID: 30521473

10

Synthesis and Characterization of Reversible Covalent HDAC4 Inhibitors.

Frühauf A, Wolff B, Schweipert M, Meyer-Almes FJ. Frühauf A, et al. Among authors: schweipert m. Methods Mol Biol. 2023;2589:207-221. doi: 10.1007/978-1-0716-2788-4_14. Methods Mol Biol. 2023. PMID: 36255627

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