Perdih A - Search Results

1

Substituted 4,5'-Bithiazoles as Catalytic Inhibitors of Human DNA Topoisomerase IIα.

Bergant Loboda K, Janežič M, Štampar M, Žegura B, Filipič M, Perdih A. Bergant Loboda K, et al. Among authors: perdih a. J Chem Inf Model. 2020 Jul 27;60(7):3662-3678. doi: 10.1021/acs.jcim.0c00202. Epub 2020 Jun 22. J Chem Inf Model. 2020. PMID: 32484690 Free PMC article.

2

In silico discovery of 2-amino-4-(2,4-dihydroxyphenyl)thiazoles as novel inhibitors of DNA gyrase B.

Brvar M, Perdih A, Oblak M, Masic LP, Solmajer T. Brvar M, et al. Among authors: perdih a. Bioorg Med Chem Lett. 2010 Feb 1;20(3):958-62. doi: 10.1016/j.bmcl.2009.12.060. Epub 2009 Dec 22. Bioorg Med Chem Lett. 2010. PMID: 20045642

3

In silico discovery and biophysical evaluation of novel 5-(2-hydroxybenzylidene) rhodanine inhibitors of DNA gyrase B.

Brvar M, Perdih A, Hodnik V, Renko M, Anderluh G, Jerala R, Solmajer T. Brvar M, et al. Among authors: perdih a. Bioorg Med Chem. 2012 Apr 15;20(8):2572-80. doi: 10.1016/j.bmc.2012.02.052. Epub 2012 Mar 3. Bioorg Med Chem. 2012. PMID: 22444877

4

Structure-based discovery of substituted 4,5'-bithiazoles as novel DNA gyrase inhibitors.

Brvar M, Perdih A, Renko M, Anderluh G, Turk D, Solmajer T. Brvar M, et al. Among authors: perdih a. J Med Chem. 2012 Jul 26;55(14):6413-26. doi: 10.1021/jm300395d. Epub 2012 Jul 5. J Med Chem. 2012. PMID: 22731783

5

Recent advances in the development of catalytic inhibitors of human DNA topoisomerase IIα as novel anticancer agents.

Pogorelčnik B, Perdih A, Solmajer T. Pogorelčnik B, et al. Among authors: perdih a. Curr Med Chem. 2013;20(5):694-709. doi: 10.2174/092986713804999402. Curr Med Chem. 2013. PMID: 23210851 Review.

6

Recent developments of DNA poisons--human DNA topoisomerase IIα inhibitors--as anticancer agents.

Pogorelčnik B, Perdih A, Solmajer T. Pogorelčnik B, et al. Among authors: perdih a. Curr Pharm Des. 2013;19(13):2474-88. doi: 10.2174/1381612811319130016. Curr Pharm Des. 2013. PMID: 23363399 Review.

7

Inhibitor design strategy based on an enzyme structural flexibility: a case of bacterial MurD ligase.

Perdih A, Hrast M, Barreteau H, Gobec S, Wolber G, Solmajer T. Perdih A, et al. J Chem Inf Model. 2014 May 27;54(5):1451-66. doi: 10.1021/ci500104m. Epub 2014 Apr 28. J Chem Inf Model. 2014. PMID: 24724969

8

Monocyclic 4-amino-6-(phenylamino)-1,3,5-triazines as inhibitors of human DNA topoisomerase IIα.

Pogorelčnik B, Brvar M, Zajc I, Filipič M, Solmajer T, Perdih A. Pogorelčnik B, et al. Among authors: perdih a. Bioorg Med Chem Lett. 2014 Dec 15;24(24):5762-5768. doi: 10.1016/j.bmcl.2014.10.042. Epub 2014 Oct 22. Bioorg Med Chem Lett. 2014. PMID: 25453816

9

Discovery of mono- and disubstituted 1H-pyrazolo[3,4]pyrimidines and 9H-purines as catalytic inhibitors of human DNA topoisomerase IIα.

Pogorelčnik B, Brvar M, Žegura B, Filipič M, Solmajer T, Perdih A. Pogorelčnik B, et al. Among authors: perdih a. ChemMedChem. 2015 Feb;10(2):345-59. doi: 10.1002/cmdc.201402459. Epub 2014 Dec 17. ChemMedChem. 2015. PMID: 25522133

10

4,6-Substituted-1,3,5-triazin-2(1H)-ones as monocyclic catalytic inhibitors of human DNA topoisomerase IIα targeting the ATP binding site.

Pogorelčnik B, Janežič M, Sosič I, Gobec S, Solmajer T, Perdih A. Pogorelčnik B, et al. Among authors: perdih a. Bioorg Med Chem. 2015 Aug 1;23(15):4218-4229. doi: 10.1016/j.bmc.2015.06.049. Epub 2015 Jul 2. Bioorg Med Chem. 2015. PMID: 26183545

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