Ramaa CS - Search Results

1

Discovery of novel N-substituted thiazolidinediones (TZDs) as HDAC8 inhibitors: in-silico studies, synthesis, and biological evaluation.

Upadhyay N, Tilekar K, Jänsch N, Schweipert M, Hess JD, Henze Macias L, Mrowka P, Aguilera RJ, Choe JY, Meyer-Almes FJ, Ramaa CS. Upadhyay N, et al. Among authors: ramaa cs. Bioorg Chem. 2020 Jul;100:103934. doi: 10.1016/j.bioorg.2020.103934. Epub 2020 May 15. Bioorg Chem. 2020. PMID: 32446120 Free PMC article.

2

Novel Anthraquinone Derivatives as Dual Inhibitors of Topoisomerase 2 and Casein Kinase 2: In Silico Studies, Synthesis and Biological Evaluation on Leukemic Cell Lines.

Kabir A, Tilekar K, Upadhyay N, Ramaa CS. Kabir A, et al. Among authors: ramaa cs. Anticancer Agents Med Chem. 2018;18(11):1551-1562. doi: 10.2174/1871520618666180423111309. Anticancer Agents Med Chem. 2018. PMID: 29683096

3

Discovery of 5-naphthylidene-2,4-thiazolidinedione derivatives as selective HDAC8 inhibitors and evaluation of their cytotoxic effects in leukemic cell lines.

Tilekar K, Upadhyay N, Jänsch N, Schweipert M, Mrowka P, Meyer-Almes FJ, Ramaa CS. Tilekar K, et al. Among authors: ramaa cs. Bioorg Chem. 2020 Jan;95:103522. doi: 10.1016/j.bioorg.2019.103522. Epub 2019 Dec 18. Bioorg Chem. 2020. PMID: 31901516

4

Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential.

Tilekar K, Upadhyay N, Hess JD, Macias LH, Mrowka P, Aguilera RJ, Meyer-Almes FJ, Iancu CV, Choe JY, Ramaa CS. Tilekar K, et al. Among authors: ramaa cs. Eur J Med Chem. 2020 Sep 15;202:112603. doi: 10.1016/j.ejmech.2020.112603. Epub 2020 Jul 2. Eur J Med Chem. 2020. PMID: 32634629 Free PMC article.

5

Permuted 2,4-thiazolidinedione (TZD) analogs as GLUT inhibitors and their in-vitro evaluation in leukemic cells.

Tilekar K, Upadhyay N, Schweipert M, Hess JD, Macias LH, Mrowka P, Meyer-Almes FJ, Aguilera RJ, Iancu CV, Choe JY, Ramaa CS. Tilekar K, et al. Among authors: ramaa cs. Eur J Pharm Sci. 2020 Nov 1;154:105512. doi: 10.1016/j.ejps.2020.105512. Epub 2020 Aug 12. Eur J Pharm Sci. 2020. PMID: 32801003 Free PMC article.

6

Benzylidene thiazolidinediones: Synthesis, in vitro investigations of antiproliferative mechanisms and in vivo efficacy determination in combination with Imatinib.

Joshi H, Patil V, Tilekar K, Upadhyay N, Gota V, Ramaa CS. Joshi H, et al. Among authors: ramaa cs. Bioorg Med Chem Lett. 2020 Dec 1;30(23):127561. doi: 10.1016/j.bmcl.2020.127561. Epub 2020 Sep 19. Bioorg Med Chem Lett. 2020. PMID: 32961322

7

Pharmacophore hybridization approach to discover novel pyrazoline-based hydantoin analogs with anti-tumor efficacy.

Upadhyay N, Tilekar K, Loiodice F, Anisimova NY, Spirina TS, Sokolova DV, Smirnova GB, Choe JY, Meyer-Almes FJ, Pokrovsky VS, Lavecchia A, Ramaa CS. Upadhyay N, et al. Among authors: ramaa cs. Bioorg Chem. 2021 Feb;107:104527. doi: 10.1016/j.bioorg.2020.104527. Epub 2020 Dec 3. Bioorg Chem. 2021. PMID: 33317839

8

Double-edged Swords: Diaryl pyrazoline thiazolidinediones synchronously targeting cancer epigenetics and angiogenesis.

Upadhyay N, Tilekar K, Safuan S, Kumar AP, Schweipert M, Meyer-Almes FJ, Ramaa CS. Upadhyay N, et al. Among authors: ramaa cs. Bioorg Chem. 2021 Nov;116:105350. doi: 10.1016/j.bioorg.2021.105350. Epub 2021 Sep 11. Bioorg Chem. 2021. PMID: 34547645

9

Synthesis and primary cytotoxicity evaluation of new 5-benzylidene-2,4-thiazolidinedione derivatives.

Patil V, Tilekar K, Mehendale-Munj S, Mohan R, Ramaa CS. Patil V, et al. Among authors: ramaa cs. Eur J Med Chem. 2010 Oct;45(10):4539-44. doi: 10.1016/j.ejmech.2010.07.014. Epub 2010 Jul 11. Eur J Med Chem. 2010. PMID: 20667627

10

Development of 1,2,4-Triazole-5-Thione Derivatives as Potential Inhibitors of Enoyl Acyl Carrier Protein Reductase (InhA) in Tuberculosis.

Vora D, Upadhyay N, Tilekar K, Jain V, Ramaa CS. Vora D, et al. Among authors: ramaa cs. Iran J Pharm Res. 2019 Fall;18(4):1742-1758. doi: 10.22037/ijpr.2019.112039.13495. Iran J Pharm Res. 2019. PMID: 32184843 Free PMC article.

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