An amide to thioamide substitution improves the permeability and bioavailability of macrocyclic peptides.
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Ghosh P, et al. Among authors: anandakumar sr.
Nat Commun. 2023 Sep 28;14(1):6050. doi: 10.1038/s41467-023-41748-y.
Nat Commun. 2023.
PMID: 37770425
Free PMC article.