Talele TT - Search Results

1

Chemical Space Exploration around Thieno[3,2-d]pyrimidin-4(3H)-one Scaffold Led to a Novel Class of Highly Active Clostridium difficile Inhibitors.

Shao X, AbdelKhalek A, Abutaleb NS, Velagapudi UK, Yoganathan S, Seleem MN, Talele TT. Shao X, et al. Among authors: talele tt. J Med Chem. 2019 Nov 14;62(21):9772-9791. doi: 10.1021/acs.jmedchem.9b01198. Epub 2019 Oct 21. J Med Chem. 2019. PMID: 31584822

2

CoMFA and HQSAR studies on 6,7-dimethoxy-4-pyrrolidylquinazoline derivatives as phosphodiesterase10A inhibitors.

Kulkarni SS, Patel MR, Talele TT. Kulkarni SS, et al. Among authors: talele tt. Bioorg Med Chem. 2008 Apr 1;16(7):3675-86. doi: 10.1016/j.bmc.2008.02.013. Epub 2008 Feb 8. Bioorg Med Chem. 2008. PMID: 18299198

3

Design, synthesis and determination of antifungal activity of 5(6)-substituted benzotriazoles.

Patel PD, Patel MR, Kocsis B, Kocsis E, Graham SM, Warren AR, Nicholson SM, Billack B, Fronczek FR, Talele TT. Patel PD, et al. Among authors: talele tt. Eur J Med Chem. 2010 Jun;45(6):2214-22. doi: 10.1016/j.ejmech.2010.01.062. Epub 2010 Feb 6. Eur J Med Chem. 2010. PMID: 20181413

4

Structure-based virtual screening, synthesis and SAR of novel inhibitors of hepatitis C virus NS5B polymerase.

Talele TT, Arora P, Kulkarni SS, Patel MR, Singh S, Chudayeu M, Kaushik-Basu N. Talele TT, et al. Bioorg Med Chem. 2010 Jul 1;18(13):4630-8. doi: 10.1016/j.bmc.2010.05.030. Epub 2010 May 15. Bioorg Med Chem. 2010. PMID: 20627595 Free PMC article.

5

The synthesis of phenylalanine-derived C5-substituted rhodanines and their activity against selected methicillin-resistant Staphylococcus aureus (MRSA) strains.

Hardej D, Ashby CR Jr, Khadtare NS, Kulkarni SS, Singh S, Talele TT. Hardej D, et al. Among authors: talele tt. Eur J Med Chem. 2010 Dec;45(12):5827-32. doi: 10.1016/j.ejmech.2010.09.045. Epub 2010 Sep 25. Eur J Med Chem. 2010. PMID: 20947220

6

Synthesis and SAR optimization of diketo acid pharmacophore for HCV NS5B polymerase inhibition.

Bhatt A, Gurukumar KR, Basu A, Patel MR, Kaushik-Basu N, Talele TT. Bhatt A, et al. Among authors: talele tt. Eur J Med Chem. 2011 Oct;46(10):5138-45. doi: 10.1016/j.ejmech.2011.08.028. Epub 2011 Aug 26. Eur J Med Chem. 2011. PMID: 21893371 Free PMC article.

7

Synthesis and SAR optimization of quinazolin-4(3H)-ones as poly(ADP-ribose)polymerase-1 inhibitors.

Kulkarni SS, Singh S, Shah JR, Low WK, Talele TT. Kulkarni SS, et al. Among authors: talele tt. Eur J Med Chem. 2012 Apr;50:264-73. doi: 10.1016/j.ejmech.2012.02.001. Epub 2012 Feb 9. Eur J Med Chem. 2012. PMID: 22365563

8

Design and synthesis of L- and D-phenylalanine derived rhodanines with novel C5-arylidenes as inhibitors of HCV NS5B polymerase.

Patel BA, Krishnan R, Khadtare N, Gurukumar KR, Basu A, Arora P, Bhatt A, Patel MR, Dana D, Kumar S, Kaushik-Basu N, Talele TT. Patel BA, et al. Among authors: talele tt. Bioorg Med Chem. 2013 Jun 1;21(11):3262-71. doi: 10.1016/j.bmc.2013.03.041. Epub 2013 Mar 31. Bioorg Med Chem. 2013. PMID: 23598249 Free PMC article.

9

The synthesis and SAR study of phenylalanine-derived (Z)-5-arylmethylidene rhodanines as anti-methicillin-resistant Staphylococcus aureus (MRSA) compounds.

Patel BA, Ashby CR Jr, Hardej D, Talele TT. Patel BA, et al. Among authors: talele tt. Bioorg Med Chem Lett. 2013 Oct 15;23(20):5523-7. doi: 10.1016/j.bmcl.2013.08.059. Epub 2013 Aug 20. Bioorg Med Chem Lett. 2013. PMID: 24012180

10

Identification of novel PARP-1 inhibitors by structure-based virtual screening.

Hannigan K, Kulkarni SS, Bdzhola VG, Golub AG, Yarmoluk SM, Talele TT. Hannigan K, et al. Among authors: talele tt. Bioorg Med Chem Lett. 2013 Nov 1;23(21):5790-4. doi: 10.1016/j.bmcl.2013.09.007. Epub 2013 Sep 10. Bioorg Med Chem Lett. 2013. PMID: 24074844

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