Moitessier N - Search Results

1

Integrated Synthetic, Biophysical, and Computational Investigations of Covalent Inhibitors of Prolyl Oligopeptidase and Fibroblast Activation Protein α.

Plescia J, De Cesco S, Patrascu MB, Kurian J, Di Trani J, Dufresne C, Wahba AS, Janmamode N, Mittermaier AK, Moitessier N. Plescia J, et al. Among authors: moitessier n. J Med Chem. 2019 Sep 12;62(17):7874-7884. doi: 10.1021/acs.jmedchem.9b00642. Epub 2019 Aug 22. J Med Chem. 2019. PMID: 31393718

2

Structure-based design, synthesis, and memapsin 2 (BACE) inhibitory activity of carbocyclic and heterocyclic peptidomimetics.

Hanessian S, Yun H, Hou Y, Yang G, Bayrakdarian M, Therrien E, Moitessier N, Roggo S, Veenstra S, Tintelnot-Blomley M, Rondeau JM, Ostermeier C, Strauss A, Ramage P, Paganetti P, Neumann U, Betschart C. Hanessian S, et al. Among authors: moitessier n. J Med Chem. 2005 Aug 11;48(16):5175-90. doi: 10.1021/jm050142+. J Med Chem. 2005. PMID: 16078837

3

A method for induced-fit docking, scoring, and ranking of flexible ligands. Application to peptidic and pseudopeptidic beta-secretase (BACE 1) inhibitors.

Moitessier N, Therrien E, Hanessian S. Moitessier N, et al. J Med Chem. 2006 Oct 5;49(20):5885-94. doi: 10.1021/jm050138y. J Med Chem. 2006. PMID: 17004704

4

Constrained peptidomimetics reveal detailed geometric requirements of covalent prolyl oligopeptidase inhibitors.

Lawandi J, Toumieux S, Seyer V, Campbell P, Thielges S, Juillerat-Jeanneret L, Moitessier N. Lawandi J, et al. Among authors: moitessier n. J Med Chem. 2009 Nov 12;52(21):6672-84. doi: 10.1021/jm901013a. J Med Chem. 2009. PMID: 19888757

5

Inhibitors of prolyl oligopeptidases for the therapy of human diseases: defining diseases and inhibitors.

Lawandi J, Gerber-Lemaire S, Juillerat-Jeanneret L, Moitessier N. Lawandi J, et al. Among authors: moitessier n. J Med Chem. 2010 May 13;53(9):3423-38. doi: 10.1021/jm901104g. J Med Chem. 2010. PMID: 20058865 Review. No abstract available.

6

An o-aminoanilide analogue of 1α,25-dihydroxyvitamin D(3) functions as a strong vitamin D receptor antagonist.

Lamblin M, Spingarn R, Wang TT, Burger MC, Dabbas B, Moitessier N, White JH, Gleason JL. Lamblin M, et al. Among authors: moitessier n. J Med Chem. 2010 Oct 28;53(20):7461-5. doi: 10.1021/jm1007159. J Med Chem. 2010. PMID: 20883026

7

Platinum(II) phenanthroimidazoles for targeting telomeric G-quadruplexes.

Castor KJ, Mancini J, Fakhoury J, Weill N, Kieltyka R, Englebienne P, Avakyan N, Mittermaier A, Autexier C, Moitessier N, Sleiman HF. Castor KJ, et al. Among authors: moitessier n. ChemMedChem. 2012 Jan 2;7(1):85-94. doi: 10.1002/cmdc.201100453. Epub 2011 Nov 3. ChemMedChem. 2012. PMID: 22052801

8

Virtual screening and computational optimization for the discovery of covalent prolyl oligopeptidase inhibitors with activity in human cells.

De Cesco S, Deslandes S, Therrien E, Levan D, Cueto M, Schmidt R, Cantin LD, Mittermaier A, Juillerat-Jeanneret L, Moitessier N. De Cesco S, et al. Among authors: moitessier n. J Med Chem. 2012 Jul 26;55(14):6306-15. doi: 10.1021/jm3002839. Epub 2012 Jul 17. J Med Chem. 2012. PMID: 22765237

9

A platinum(II) phenylphenanthroimidazole with an extended side-chain exhibits slow dissociation from a c-Kit G-quadruplex motif.

Castor KJ, Liu Z, Fakhoury J, Hancock MA, Mittermaier A, Moitessier N, Sleiman HF. Castor KJ, et al. Among authors: moitessier n. Chemistry. 2013 Dec 23;19(52):17836-45. doi: 10.1002/chem.201301590. Epub 2013 Nov 18. Chemistry. 2013. PMID: 24249701

10

Discovery of novel small-molecule antagonists for GluK2.

Schiavini P, Dawe GB, Bowie D, Moitessier N. Schiavini P, et al. Among authors: moitessier n. Bioorg Med Chem Lett. 2015 Jun 1;25(11):2416-20. doi: 10.1016/j.bmcl.2015.04.008. Epub 2015 Apr 10. Bioorg Med Chem Lett. 2015. PMID: 25913117

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