Schostarez HJ - Search Results

1

Structure-Activity Relationship of Flavin Analogues That Target the Flavin Mononucleotide Riboswitch.

Vicens Q, Mondragón E, Reyes FE, Coish P, Aristoff P, Berman J, Kaur H, Kells KW, Wickens P, Wilson J, Gadwood RC, Schostarez HJ, Suto RK, Blount KF, Batey RT. Vicens Q, et al. Among authors: schostarez hj. ACS Chem Biol. 2018 Oct 19;13(10):2908-2919. doi: 10.1021/acschembio.8b00533. Epub 2018 Sep 20. ACS Chem Biol. 2018. PMID: 30107111 Free PMC article.

2

Novel riboswitch-binding flavin analog that protects mice against Clostridium difficile infection without inhibiting cecal flora.

Blount KF, Megyola C, Plummer M, Osterman D, O'Connell T, Aristoff P, Quinn C, Chrusciel RA, Poel TJ, Schostarez HJ, Stewart CA, Walker DP, Wuts PG, Breaker RR. Blount KF, et al. Among authors: schostarez hj. Antimicrob Agents Chemother. 2015 Sep;59(9):5736-46. doi: 10.1128/AAC.01282-15. Epub 2015 Jul 13. Antimicrob Agents Chemother. 2015. PMID: 26169403 Free PMC article.

3

Exploiting the molecular template of angiotensinogen in the discovery and design of peptidyl, pseudopeptidyl and peptidimimetic inhibitors of human renin: a structure-activity perspective.

Sawyer TK, Hester JB, Schostarez HJ, Thaisrivongs S, Bundy GL, Liu L, Bradford VS, De Vaux AE, Staples DJ, Maggiora LL, et al. Sawyer TK, et al. Among authors: schostarez hj. Adv Exp Med Biol. 1991;306:307-23. doi: 10.1007/978-1-4684-6012-4_37. Adv Exp Med Biol. 1991. PMID: 1812721 Review. No abstract available.

4

Determination of dissociation constants of high affinity (pM) human renin inhibitors: application to analogues of ditekiren (U-71,038).

Epps DE, Poorman RA, Mandel F, Schostarez HJ. Epps DE, et al. Among authors: schostarez hj. J Med Chem. 1991 Jul;34(7):2107-12. doi: 10.1021/jm00111a028. J Med Chem. 1991. PMID: 2066983

5

Synthesis and biological activity of a novel class of small molecular weight peptidomimetic competitive inhibitors of protein tyrosine phosphatase 1B.

Larsen SD, Barf T, Liljebris C, May PD, Ogg D, O'Sullivan TJ, Palazuk BJ, Schostarez HJ, Stevens FC, Bleasdale JE. Larsen SD, et al. Among authors: schostarez hj. J Med Chem. 2002 Jan 31;45(3):598-622. doi: 10.1021/jm010393s. J Med Chem. 2002. PMID: 11806712

6

alpha,alpha-Difluoro-beta-aminodeoxystatine-containing renin inhibitory peptides.

Thaisrivongs S, Schostarez HJ, Pals DT, Turner SR. Thaisrivongs S, et al. Among authors: schostarez hj. J Med Chem. 1987 Oct;30(10):1837-42. doi: 10.1021/jm00393a026. J Med Chem. 1987. PMID: 3309315

7

HIV protease (HIV PR) inhibitor structure-activity-selectivity, and active site molecular modeling of high affinity Leu [CH(OH)CH2]Val modified viral and nonviral substrate analogs.

Sawyer TK, Staples DJ, Liu L, Tomasselli AG, Hui JO, O'Connell K, Schostarez H, Hester JB, Moon J, Howe WJ, et al. Sawyer TK, et al. Int J Pept Protein Res. 1992 Sep-Oct;40(3-4):274-81. doi: 10.1111/j.1399-3011.1992.tb00302.x. Int J Pept Protein Res. 1992. PMID: 1478785

8

Thermodynamics of the interaction of inhibitors with the binding site of recombinant human renin.

Epps DE, Cheney J, Schostarez H, Sawyer TK, Prairie M, Krueger WC, Mandel F. Epps DE, et al. J Med Chem. 1990 Aug;33(8):2080-6. doi: 10.1021/jm00170a006. J Med Chem. 1990. PMID: 2197411

9

An experimental method for the determination of enzyme-competitive inhibitor dissociation constants from displacement curves: application to human renin using fluorescence energy transfer to a synthetic dansylated inhibitor peptide.

Epps DE, Schostarez H, Argoudelis CV, Poorman R, Hinzmann J, Sawyer TK, Mandel F. Epps DE, et al. Anal Biochem. 1989 Aug 15;181(1):172-81. doi: 10.1016/0003-2697(89)90413-2. Anal Biochem. 1989. PMID: 2683862

10

Synthesis of a series of stromelysin-selective thiadiazole urea matrix metalloproteinase inhibitors.

Jacobsen EJ, Mitchell MA, Hendges SK, Belonga KL, Skaletzky LL, Stelzer LS, Lindberg TJ, Fritzen EL, Schostarez HJ, O'Sullivan TJ, Maggiora LL, Stuchly CW, Laborde AL, Kubicek MF, Poorman RA, Beck JM, Miller HR, Petzold GL, Scott PS, Truesdell SE, Wallace TL, Wilks JW, Fisher C, Goodman LV, Kaytes PS, et al. Jacobsen EJ, et al. Among authors: schostarez hj. J Med Chem. 1999 May 6;42(9):1525-36. doi: 10.1021/jm9803222. J Med Chem. 1999. PMID: 10229623

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

15 results

Search Page

Filters