Augustyns K - Search Results

1

Tozasertib Analogues as Inhibitors of Necroptotic Cell Death.

Hofmans S, Devisscher L, Martens S, Van Rompaey D, Goossens K, Divert T, Nerinckx W, Takahashi N, De Winter H, Van Der Veken P, Goossens V, Vandenabeele P, Augustyns K. Hofmans S, et al. Among authors: augustyns k. J Med Chem. 2018 Mar 8;61(5):1895-1920. doi: 10.1021/acs.jmedchem.7b01449. Epub 2018 Feb 20. J Med Chem. 2018. PMID: 29437386

2

Structure-activity relationship of diaryl phosphonate esters as potent irreversible dipeptidyl peptidase IV inhibitors.

Belyaev A, Zhang X, Augustyns K, Lambeir AM, De Meester I, Vedernikova I, Scharpé S, Haemers A. Belyaev A, et al. Among authors: augustyns k. J Med Chem. 1999 Mar 25;42(6):1041-52. doi: 10.1021/jm981033g. J Med Chem. 1999. PMID: 10090787

3

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 2: substitution of the glycine part.

Amssoms K, Oza SL, Augustyns K, Yamani A, Lambeir AM, Bal G, Van der Veken P, Fairlamb AH, Haemers A. Amssoms K, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2002 Oct 7;12(19):2703-5. doi: 10.1016/s0960-894x(02)00538-3. Bioorg Med Chem Lett. 2002. PMID: 12217358

4

Development of potent and selective dipeptidyl peptidase II inhibitors.

Senten K, Van der Veken P, Bal G, De Meester I, Lambeir AM, Scharpé S, Bauvois B, Haemers A, Augustyns K. Senten K, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2002 Oct 21;12(20):2825-8. doi: 10.1016/s0960-894x(02)00603-0. Bioorg Med Chem Lett. 2002. PMID: 12270155

5

Rapid parallel synthesis of dipeptide diphenyl phosphonate esters as inhibitors of dipeptidyl peptidases.

Senten K, Daniëls L, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: augustyns k. J Comb Chem. 2003 May-Jun;5(3):336-44. doi: 10.1021/cc020096o. J Comb Chem. 2003. PMID: 12739951

6

Design, synthesis, and SAR of potent and selective dipeptide-derived inhibitors for dipeptidyl peptidases.

Senten K, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: augustyns k. J Med Chem. 2003 Nov 6;46(23):5005-14. doi: 10.1021/jm0308803. J Med Chem. 2003. PMID: 14584950

7

Prolylisoxazoles: potent inhibitors of prolyloligopeptidase with antitrypanosomal activity.

Bal G, Van der Veken P, Antonov D, Lambeir AM, Grellier P, Croft SL, Augustyns K, Haemers A. Bal G, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2003 Sep 1;13(17):2875-8. doi: 10.1016/s0960-894x(03)00579-1. Bioorg Med Chem Lett. 2003. PMID: 14611847

8

Development of irreversible diphenyl phosphonate inhibitors for urokinase plasminogen activator.

Joossens J, Van der Veken P, Lambeir AM, Augustyns K, Haemers A. Joossens J, et al. Among authors: augustyns k. J Med Chem. 2004 May 6;47(10):2411-3. doi: 10.1021/jm0499209. J Med Chem. 2004. PMID: 15115382

9

Synthesis and electrophysiological characterization of cyclic morphiceptin analogues.

Pil J, Van der Veken P, Bal G, Augustyns K, Haemers A, Tytgat J. Pil J, et al. Among authors: augustyns k. Biochem Pharmacol. 2004 May 15;67(10):1887-95. doi: 10.1016/j.bcp.2004.02.011. Biochem Pharmacol. 2004. PMID: 15130765

10

Gamma-amino-substituted analogues of 1-[(S)-2,4-diaminobutanoyl]piperidine as highly potent and selective dipeptidyl peptidase II inhibitors.

Senten K, Van Der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: augustyns k. J Med Chem. 2004 May 20;47(11):2906-16. doi: 10.1021/jm031122f. J Med Chem. 2004. PMID: 15139769

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