Jacobson KA - Search Results

1

Demystifying P2Y₁ Receptor Ligand Recognition through Docking and Molecular Dynamics Analyses.

Ciancetta A, O'Connor RD, Paoletta S, Jacobson KA. Ciancetta A, et al. Among authors: jacobson ka. J Chem Inf Model. 2017 Dec 26;57(12):3104-3123. doi: 10.1021/acs.jcim.7b00528. Epub 2017 Nov 28. J Chem Inf Model. 2017. PMID: 29182323 Free PMC article.

2

Site-directed mutagenesis identifies residues involved in ligand recognition in the human A2a adenosine receptor.

Kim J, Wess J, van Rhee AM, Schöneberg T, Jacobson KA. Kim J, et al. Among authors: jacobson ka. J Biol Chem. 1995 Jun 9;270(23):13987-97. doi: 10.1074/jbc.270.23.13987. J Biol Chem. 1995. PMID: 7775460 Free PMC article.

3

Comparative molecular field analysis of selective A3 adenosine receptor agonists.

Siddiqi SM, Pearlstein RA, Sanders LH, Jacobson KA. Siddiqi SM, et al. Among authors: jacobson ka. Bioorg Med Chem. 1995 Oct;3(10):1331-43. doi: 10.1016/0968-0896(95)00116-x. Bioorg Med Chem. 1995. PMID: 8564399 Free PMC article.

4

Glutamate residues in the second extracellular loop of the human A2a adenosine receptor are required for ligand recognition.

Kim J, Jiang Q, Glashofer M, Yehle S, Wess J, Jacobson KA. Kim J, et al. Among authors: jacobson ka. Mol Pharmacol. 1996 Apr;49(4):683-91. Mol Pharmacol. 1996. PMID: 8609897 Free PMC article.

5

Hydrophilic side chains in the third and seventh transmembrane helical domains of human A2A adenosine receptors are required for ligand recognition.

Jiang Q, Van Rhee AM, Kim J, Yehle S, Wess J, Jacobson KA. Jiang Q, et al. Among authors: jacobson ka. Mol Pharmacol. 1996 Sep;50(3):512-21. Mol Pharmacol. 1996. PMID: 8794889 Free PMC article.

6

A mutational analysis of residues essential for ligand recognition at the human P2Y1 receptor.

Jiang Q, Guo D, Lee BX, Van Rhee AM, Kim YC, Nicholas RA, Schachter JB, Harden TK, Jacobson KA. Jiang Q, et al. Among authors: jacobson ka. Mol Pharmacol. 1997 Sep;52(3):499-507. doi: 10.1124/mol.52.3.499. Mol Pharmacol. 1997. PMID: 9281613 Free PMC article.

7

Deoxyadenosine bisphosphate derivatives as potent antagonists at P2Y1 receptors.

Camaioni E, Boyer JL, Mohanram A, Harden TK, Jacobson KA. Camaioni E, et al. Among authors: jacobson ka. J Med Chem. 1998 Jan 15;41(2):183-90. doi: 10.1021/jm970433l. J Med Chem. 1998. PMID: 9457242 Free PMC article.

8

Human P2Y1 receptor: molecular modeling and site-directed mutagenesis as tools to identify agonist and antagonist recognition sites.

Moro S, Guo D, Camaioni E, Boyer JL, Harden TK, Jacobson KA. Moro S, et al. Among authors: jacobson ka. J Med Chem. 1998 Apr 23;41(9):1456-66. doi: 10.1021/jm970684u. J Med Chem. 1998. PMID: 9554879 Free PMC article.

9

Molecular modeling studies of human A3 adenosine antagonists: structural homology and receptor docking.

Moro S, Li AH, Jacobson KA. Moro S, et al. Among authors: jacobson ka. J Chem Inf Comput Sci. 1998 Nov-Dec;38(6):1239-48. doi: 10.1021/ci980080e. J Chem Inf Comput Sci. 1998. PMID: 9845970 Free PMC article.

10

Synthesis, CoMFA analysis, and receptor docking of 3,5-diacyl-2, 4-dialkylpyridine derivatives as selective A3 adenosine receptor antagonists.

Li AH, Moro S, Forsyth N, Melman N, Ji XD, Jacobson KA. Li AH, et al. Among authors: jacobson ka. J Med Chem. 1999 Feb 25;42(4):706-21. doi: 10.1021/jm980550w. J Med Chem. 1999. PMID: 10052977 Free PMC article.

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