Davis MI - Search Results

1

Assessing inhibitors of mutant isocitrate dehydrogenase using a suite of pre-clinical discovery assays.

Urban DJ, Martinez NJ, Davis MI, Brimacombe KR, Cheff DM, Lee TD, Henderson MJ, Titus SA, Pragani R, Rohde JM, Liu L, Fang Y, Karavadhi S, Shah P, Lee OW, Wang A, McIver A, Zheng H, Wang X, Xu X, Jadhav A, Simeonov A, Shen M, Boxer MB, Hall MD. Urban DJ, et al. Among authors: davis mi. Sci Rep. 2017 Oct 6;7(1):12758. doi: 10.1038/s41598-017-12630-x. Sci Rep. 2017. PMID: 28986582 Free PMC article.

2

Literature search and review.

Auld D, Lea W, Davis MI, Simeonov A. Auld D, et al. Among authors: davis mi. Assay Drug Dev Technol. 2011 Jun;9(3):198-212. doi: 10.1089/adt.2011.0903.lr. Assay Drug Dev Technol. 2011. PMID: 21612549 Review. No abstract available.

3

A homogeneous, high-throughput assay for phosphatidylinositol 5-phosphate 4-kinase with a novel, rapid substrate preparation.

Davis MI, Sasaki AT, Shen M, Emerling BM, Thorne N, Michael S, Pragani R, Boxer M, Sumita K, Takeuchi K, Auld DS, Li Z, Cantley LC, Simeonov A. Davis MI, et al. PLoS One. 2013;8(1):e54127. doi: 10.1371/journal.pone.0054127. Epub 2013 Jan 10. PLoS One. 2013. PMID: 23326584 Free PMC article.

4

none.

Auld D, Lea W, Davis MI, Simeonov A. Auld D, et al. Among authors: davis mi. Assay Drug Dev Technol. 2013 Apr;11(3):139-51. doi: 10.1089/adt.2013.1103.lr. Assay Drug Dev Technol. 2013. PMID: 23560851 No abstract available.

5

Identification of potent Yes1 kinase inhibitors using a library screening approach.

Patel PR, Sun H, Li SQ, Shen M, Khan J, Thomas CJ, Davis MI. Patel PR, et al. Among authors: davis mi. Bioorg Med Chem Lett. 2013 Aug 1;23(15):4398-403. doi: 10.1016/j.bmcl.2013.05.072. Epub 2013 May 29. Bioorg Med Chem Lett. 2013. PMID: 23787099 Free PMC article.

6

A panel of diverse assays to interrogate the interaction between glucokinase and glucokinase regulatory protein, two vital proteins in human disease.

Rees MG, Davis MI, Shen M, Titus S, Raimondo A, Barrett A, Gloyn AL, Collins FS, Simeonov A. Rees MG, et al. Among authors: davis mi. PLoS One. 2014 Feb 19;9(2):e89335. doi: 10.1371/journal.pone.0089335. eCollection 2014. PLoS One. 2014. PMID: 24586696 Free PMC article.

7

Biochemical, cellular, and biophysical characterization of a potent inhibitor of mutant isocitrate dehydrogenase IDH1.

Davis MI, Gross S, Shen M, Straley KS, Pragani R, Lea WA, Popovici-Muller J, DeLaBarre B, Artin E, Thorne N, Auld DS, Li Z, Dang L, Boxer MB, Simeonov A. Davis MI, et al. J Biol Chem. 2014 May 16;289(20):13717-25. doi: 10.1074/jbc.M113.511030. Epub 2014 Mar 25. J Biol Chem. 2014. PMID: 24668804 Free PMC article.

8

Method for Assaying the Lipid Kinase Phosphatidylinositol-5-phosphate 4-kinase α in Quantitative High-Throughput Screening (qHTS) Bioluminescent Format.

Davis MI, Sasaki AT, Simeonov A. Davis MI, et al. Methods Mol Biol. 2016;1376:1-9. doi: 10.1007/978-1-4939-3170-5_1. Methods Mol Biol. 2016. PMID: 26552670 Free PMC article.

9

Ubiquitin-Specific Proteases as Druggable Targets.

Davis MI, Simeonov A. Davis MI, et al. Drug Target Rev. 2015 Fall;2(3):60-64. Drug Target Rev. 2015. PMID: 26835158 Free PMC article. No abstract available.

10

Avoiding Fluorescence Assay Interference-The Case for Diaphorase.

Hall MD, Simeonov A, Davis MI. Hall MD, et al. Among authors: davis mi. Assay Drug Dev Technol. 2016 Apr;14(3):175-9. doi: 10.1089/adt.2016.707. Assay Drug Dev Technol. 2016. PMID: 27078679 Free PMC article. Review.

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