Geitmann M - Search Results

1

Development of 5-hydroxypyrazole derivatives as reversible inhibitors of lysine specific demethylase 1.

Mould DP, Bremberg U, Jordan AM, Geitmann M, Maiques-Diaz A, McGonagle AE, Small HF, Somervaille TCP, Ogilvie D. Mould DP, et al. Among authors: geitmann m. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195. doi: 10.1016/j.bmcl.2017.05.018. Epub 2017 May 8. Bioorg Med Chem Lett. 2017. PMID: 28545974

2

Development of (4-Cyanophenyl)glycine Derivatives as Reversible Inhibitors of Lysine Specific Demethylase 1.

Mould DP, Alli C, Bremberg U, Cartic S, Jordan AM, Geitmann M, Maiques-Diaz A, McGonagle AE, Somervaille TCP, Spencer GJ, Turlais F, Ogilvie D. Mould DP, et al. Among authors: geitmann m. J Med Chem. 2017 Oct 12;60(19):7984-7999. doi: 10.1021/acs.jmedchem.7b00462. Epub 2017 Sep 21. J Med Chem. 2017. PMID: 28892629

3

Development and evaluation of 4-(pyrrolidin-3-yl)benzonitrile derivatives as inhibitors of lysine specific demethylase 1.

Mould DP, Bremberg U, Jordan AM, Geitmann M, McGonagle AE, Somervaille TCP, Spencer GJ, Ogilvie DJ. Mould DP, et al. Among authors: geitmann m. Bioorg Med Chem Lett. 2017 Oct 15;27(20):4755-4759. doi: 10.1016/j.bmcl.2017.08.052. Epub 2017 Aug 24. Bioorg Med Chem Lett. 2017. PMID: 28927796

4

Deconstruction of non-nucleoside reverse transcriptase inhibitors of human immunodeficiency virus type 1 for exploration of the optimization landscape of fragments.

Brandt P, Geitmann M, Danielson UH. Brandt P, et al. Among authors: geitmann m. J Med Chem. 2011 Feb 10;54(3):709-18. doi: 10.1021/jm101052g. Epub 2011 Jan 5. J Med Chem. 2011. PMID: 21207958

5

Identification of a novel scaffold for allosteric inhibition of wild type and drug resistant HIV-1 reverse transcriptase by fragment library screening.

Geitmann M, Elinder M, Seeger C, Brandt P, de Esch IJ, Danielson UH. Geitmann M, et al. J Med Chem. 2011 Feb 10;54(3):699-708. doi: 10.1021/jm1010513. Epub 2011 Jan 5. J Med Chem. 2011. PMID: 21207961

6

Biosensor-based kinetic characterization of the interaction between HIV-1 reverse transcriptase and non-nucleoside inhibitors.

Geitmann M, Unge T, Danielson UH. Geitmann M, et al. J Med Chem. 2006 Apr 20;49(8):2367-74. doi: 10.1021/jm0504048. J Med Chem. 2006. PMID: 16610780

7

Interaction kinetic characterization of HIV-1 reverse transcriptase non-nucleoside inhibitor resistance.

Geitmann M, Unge T, Danielson UH. Geitmann M, et al. J Med Chem. 2006 Apr 20;49(8):2375-87. doi: 10.1021/jm0504050. J Med Chem. 2006. PMID: 16610781

8

Identification and Characterization of an Irreversible Inhibitor of CDK2.

Anscombe E, Meschini E, Mora-Vidal R, Martin MP, Staunton D, Geitmann M, Danielson UH, Stanley WA, Wang LZ, Reuillon T, Golding BT, Cano C, Newell DR, Noble ME, Wedge SR, Endicott JA, Griffin RJ. Anscombe E, et al. Among authors: geitmann m. Chem Biol. 2015 Sep 17;22(9):1159-64. doi: 10.1016/j.chembiol.2015.07.018. Epub 2015 Aug 27. Chem Biol. 2015. PMID: 26320860 Free PMC article.

9

Additional level of information about complex interaction between non-nucleoside inhibitor and HIV-1 reverse transcriptase using biosensor-based thermodynamic analysis.

Geitmann M, Danielson UH. Geitmann M, et al. Bioorg Med Chem. 2007 Dec 1;15(23):7344-54. doi: 10.1016/j.bmc.2007.08.018. Epub 2007 Aug 22. Bioorg Med Chem. 2007. PMID: 17870544

10

Surface plasmon resonance biosensor based fragment screening using acetylcholine binding protein identifies ligand efficiency hot spots (LE hot spots) by deconstruction of nicotinic acetylcholine receptor α7 ligands.

de Kloe GE, Retra K, Geitmann M, Källblad P, Nahar T, van Elk R, Smit AB, van Muijlwijk-Koezen JE, Leurs R, Irth H, Danielson UH, de Esch IJ. de Kloe GE, et al. Among authors: geitmann m. J Med Chem. 2010 Oct 14;53(19):7192-201. doi: 10.1021/jm100834y. J Med Chem. 2010. PMID: 20828128

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