Gutiérrez-de-Terán H - Search Results

1

Enantiospecific Recognition at the A_2B Adenosine Receptor by Alkyl 2-Cyanoimino-4-substituted-6-methyl-1,2,3,4-tetrahydropyrimidine-5-carboxylates.

Carbajales C, Azuaje J, Oliveira A, Loza MI, Brea J, Cadavid MI, Masaguer CF, García-Mera X, Gutiérrez-de-Terán H, Sotelo E. Carbajales C, et al. J Med Chem. 2017 Apr 27;60(8):3372-3382. doi: 10.1021/acs.jmedchem.7b00138. Epub 2017 Apr 11. J Med Chem. 2017. PMID: 28368607

2

Synthesis, adenosine receptor binding and 3D-QSAR of 4-substituted 2-(2'-furyl)-1,2,4-triazolo[1,5-a]quinoxalines.

Martínez A, Gutiérrez-de-Terán H, Brea J, Raviña E, Loza MI, Cadavid MI, Sanz F, Vidal B, Segarra V, Sotelo E. Martínez A, et al. Bioorg Med Chem. 2008 Feb 15;16(4):2103-13. doi: 10.1016/j.bmc.2007.10.103. Epub 2008 Jan 24. Bioorg Med Chem. 2008. PMID: 18249548

3

In silico directed chemical probing of the adenosine receptor family.

Areias FM, Brea J, Gregori-Puigjané E, Zaki ME, Carvalho MA, Domínguez E, Gutiérrez-de-Terán H, Proença MF, Loza MI, Mestres J. Areias FM, et al. Bioorg Med Chem. 2010 May 1;18(9):3043-52. doi: 10.1016/j.bmc.2010.03.048. Epub 2010 Mar 27. Bioorg Med Chem. 2010. PMID: 20382540

4

Pyrimidine derivatives as potent and selective A3 adenosine receptor antagonists.

Yaziji V, Rodríguez D, Gutiérrez-de-Terán H, Coelho A, Caamaño O, García-Mera X, Brea J, Loza MI, Cadavid MI, Sotelo E. Yaziji V, et al. J Med Chem. 2011 Jan 27;54(2):457-71. doi: 10.1021/jm100843z. Epub 2010 Dec 27. J Med Chem. 2011. PMID: 21186795

5

Selective and potent adenosine A3 receptor antagonists by methoxyaryl substitution on the N-(2,6-diarylpyrimidin-4-yl)acetamide scaffold.

Yaziji V, Rodríguez D, Coelho A, García-Mera X, El Maatougui A, Brea J, Loza MI, Cadavid MI, Gutiérrez-de-Terán H, Sotelo E. Yaziji V, et al. Eur J Med Chem. 2013 Jan;59:235-42. doi: 10.1016/j.ejmech.2012.11.010. Epub 2012 Nov 24. Eur J Med Chem. 2013. PMID: 23231967

6

Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists.

Crespo A, El Maatougui A, Biagini P, Azuaje J, Coelho A, Brea J, Loza MI, Cadavid MI, García-Mera X, Gutiérrez-de-Terán H, Sotelo E. Crespo A, et al. ACS Med Chem Lett. 2013 Oct 3;4(11):1031-6. doi: 10.1021/ml400185v. eCollection 2013 Nov 14. ACS Med Chem Lett. 2013. PMID: 24900602 Free PMC article.

7

Structure-based design of new KSP-Eg5 inhibitors assisted by a targeted multicomponent reaction.

Carbajales C, Prado MÁ, Gutiérrez-de-Terán H, Cores A, Azuaje J, Novio S, Nuñez MJ, Fernández-García B, Sotelo E, García-Mera X, Sánchez-Lazo P, Freire-Garabal M, Coelho A. Carbajales C, et al. Chembiochem. 2014 Jul 7;15(10):1471-80. doi: 10.1002/cbic.201402089. Epub 2014 Jun 18. Chembiochem. 2014. PMID: 24943831

8

Computer-aided design of GPCR ligands.

Gutiérrez-de-Terán H, Keränen H, Azuaje J, Rodríguez D, Åqvist J, Sotelo E. Gutiérrez-de-Terán H, et al. Methods Mol Biol. 2015;1272:271-91. doi: 10.1007/978-1-4939-2336-6_19. Methods Mol Biol. 2015. PMID: 25563191

9

Pyrazin-2(1H)-ones as a novel class of selective A3 adenosine receptor antagonists.

Azuaje J, Carbajales C, González-Gómez M, Coelho A, Caamaño O, Gutiérrez-de-Terán H, Sotelo E. Azuaje J, et al. Future Med Chem. 2015;7(11):1373-80. doi: 10.4155/fmc.15.69. Future Med Chem. 2015. PMID: 26230877

10

Discovery of Potent and Highly Selective A2B Adenosine Receptor Antagonist Chemotypes.

El Maatougui A, Azuaje J, González-Gómez M, Miguez G, Crespo A, Carbajales C, Escalante L, García-Mera X, Gutiérrez-de-Terán H, Sotelo E. El Maatougui A, et al. J Med Chem. 2016 Mar 10;59(5):1967-83. doi: 10.1021/acs.jmedchem.5b01586. Epub 2016 Feb 9. J Med Chem. 2016. PMID: 26824742

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

102 results

Search Page

Filters