de Vries H - Search Results

1

Small molecule absorption by PDMS in the context of drug response bioassays.

van Meer BJ, de Vries H, Firth KSA, van Weerd J, Tertoolen LGJ, Karperien HBJ, Jonkheijm P, Denning C, IJzerman AP, Mummery CL. van Meer BJ, et al. Among authors: de vries h. Biochem Biophys Res Commun. 2017 Jan 8;482(2):323-328. doi: 10.1016/j.bbrc.2016.11.062. Epub 2016 Nov 14. Biochem Biophys Res Commun. 2017. PMID: 27856254 Free PMC article.

2

Scintillation proximity assay (SPA) as a new approach to determine a ligand's kinetic profile. A case in point for the adenosine A1 receptor.

Xia L, de Vries H, IJzerman AP, Heitman LH. Xia L, et al. Among authors: de vries h. Purinergic Signal. 2016 Mar;12(1):115-26. doi: 10.1007/s11302-015-9485-0. Epub 2015 Dec 9. Purinergic Signal. 2016. PMID: 26647040 Free PMC article.

3

Synthesis and biological evaluation of a new series of 2,3,5-substituted [1,2,4]-thiadiazoles as modulators of adenosine A1 receptors and their molecular mechanism of action.

Göblyös A, de Vries H, Brussee J, Ijzerman AP. Göblyös A, et al. Among authors: de vries h. J Med Chem. 2005 Feb 24;48(4):1145-51. doi: 10.1021/jm049337s. J Med Chem. 2005. PMID: 15715480

4

Kinetics of human cannabinoid 1 (CB1) receptor antagonists: Structure-kinetics relationships (SKR) and implications for insurmountable antagonism.

Xia L, de Vries H, Yang X, Lenselink EB, Kyrizaki A, Barth F, Louvel J, Dreyer MK, van der Es D, IJzerman AP, Heitman LH. Xia L, et al. Among authors: de vries h. Biochem Pharmacol. 2018 May;151:166-179. doi: 10.1016/j.bcp.2017.10.014. Epub 2017 Nov 2. Biochem Pharmacol. 2018. PMID: 29102677 Free article.

5

Synthesis and evaluation of N-substituted 2-amino-4,5-diarylpyrimidines as selective adenosine A₁ receptor antagonists.

Alachouzos G, Lenselink EB, Mulder-Krieger T, de Vries H, IJzerman AP, Louvel J. Alachouzos G, et al. Among authors: de vries h. Eur J Med Chem. 2017 Jan 5;125:586-602. doi: 10.1016/j.ejmech.2016.09.081. Epub 2016 Sep 26. Eur J Med Chem. 2017. PMID: 27718474

6

Kinetic profiling and functional characterization of 8-phenylxanthine derivatives as A_2B adenosine receptor antagonists.

Vlachodimou A, de Vries H, Pasoli M, Goudswaard M, Kim SA, Kim YC, Scortichini M, Marshall M, Linden J, Heitman LH, Jacobson KA, IJzerman AP. Vlachodimou A, et al. Among authors: de vries h. Biochem Pharmacol. 2022 Jun;200:115027. doi: 10.1016/j.bcp.2022.115027. Epub 2022 Apr 6. Biochem Pharmacol. 2022. PMID: 35395239 Free PMC article.

7

Identifying novel adenosine receptor ligands by simultaneous proteochemometric modeling of rat and human bioactivity data.

van Westen GJ, van den Hoven OO, van der Pijl R, Mulder-Krieger T, de Vries H, Wegner JK, Ijzerman AP, van Vlijmen HW, Bender A. van Westen GJ, et al. Among authors: de vries h. J Med Chem. 2012 Aug 23;55(16):7010-20. doi: 10.1021/jm3003069. Epub 2012 Aug 3. J Med Chem. 2012. PMID: 22827545

8

Putative role of the adenosine A(3) receptor in the antiproliferative action of N (6)-(2-isopentenyl)adenosine.

Blad CC, von Frijtag Drabbe Künzel JK, de Vries H, Mulder-Krieger T, Bar-Yehuda S, Fishman P, Ijzerman AP. Blad CC, et al. Among authors: de vries h. Purinergic Signal. 2011 Dec;7(4):453-62. doi: 10.1007/s11302-011-9244-9. Epub 2011 Jul 1. Purinergic Signal. 2011. PMID: 21720785 Free PMC article.

9

Effects of pyrazole partial agonists on HCA(2) -mediated flushing and VLDL-triglyceride levels in mice.

Li Z, Blad CC, van der Sluis RJ, de Vries H, Van Berkel TJ, Ijzerman AP, Hoekstra M. Li Z, et al. Among authors: de vries h. Br J Pharmacol. 2012 Oct;167(4):818-25. doi: 10.1111/j.1476-5381.2012.02039.x. Br J Pharmacol. 2012. PMID: 22616721 Free PMC article.

10

Substituted terphenyl compounds as the first class of low molecular weight allosteric inhibitors of the luteinizing hormone receptor.

Heitman LH, Narlawar R, de Vries H, Willemsen MN, Wolfram D, Brussee J, Ijzerman AP. Heitman LH, et al. Among authors: de vries h. J Med Chem. 2009 Apr 9;52(7):2036-42. doi: 10.1021/jm801561h. J Med Chem. 2009. PMID: 19296599

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