Ernst M - Search Results

1

Structural Studies of GABAA Receptor Binding Sites: Which Experimental Structure Tells us What?

Puthenkalam R, Hieckel M, Simeone X, Suwattanasophon C, Feldbauer RV, Ecker GF, Ernst M. Puthenkalam R, et al. Among authors: ernst m. Front Mol Neurosci. 2016 Jun 16;9:44. doi: 10.3389/fnmol.2016.00044. eCollection 2016. Front Mol Neurosci. 2016. PMID: 27378845 Free PMC article.

2

Comparative models of GABAA receptor extracellular and transmembrane domains: important insights in pharmacology and function.

Ernst M, Bruckner S, Boresch S, Sieghart W. Ernst M, et al. Mol Pharmacol. 2005 Nov;68(5):1291-300. doi: 10.1124/mol.105.015982. Epub 2005 Aug 15. Mol Pharmacol. 2005. PMID: 16103045

3

An updated unified pharmacophore model of the benzodiazepine binding site on gamma-aminobutyric acid(a) receptors: correlation with comparative models.

Clayton T, Chen JL, Ernst M, Richter L, Cromer BA, Morton CJ, Ng H, Kaczorowski CC, Helmstetter FJ, Furtmüller R, Ecker G, Parker MW, Sieghart W, Cook JM. Clayton T, et al. Among authors: ernst m. Curr Med Chem. 2007;14(26):2755-75. doi: 10.2174/092986707782360097. Curr Med Chem. 2007. PMID: 18045122 Review.

4

The GABAA receptor alpha+beta- interface: a novel target for subtype selective drugs.

Ramerstorfer J, Furtmüller R, Sarto-Jackson I, Varagic Z, Sieghart W, Ernst M. Ramerstorfer J, et al. Among authors: ernst m. J Neurosci. 2011 Jan 19;31(3):870-7. doi: 10.1523/JNEUROSCI.5012-10.2011. J Neurosci. 2011. PMID: 21248110 Free PMC article.

5

Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligands.

Richter L, de Graaf C, Sieghart W, Varagic Z, Mörzinger M, de Esch IJ, Ecker GF, Ernst M. Richter L, et al. Among authors: ernst m. Nat Chem Biol. 2012 Mar 25;8(5):455-64. doi: 10.1038/nchembio.917. Nat Chem Biol. 2012. PMID: 22446838 Free PMC article.

6

Identification of novel positive allosteric modulators and null modulators at the GABAA receptor α+β- interface.

Varagic Z, Wimmer L, Schnürch M, Mihovilovic MD, Huang S, Rallapalli S, Cook JM, Mirheydari P, Ecker GF, Sieghart W, Ernst M. Varagic Z, et al. Among authors: ernst m. Br J Pharmacol. 2013 May;169(2):371-83. doi: 10.1111/bph.12151. Br J Pharmacol. 2013. PMID: 23472852 Free PMC article.

7

Molecular analysis of the site for 2-arachidonylglycerol (2-AG) on the β₂ subunit of GABA(A) receptors.

Baur R, Kielar M, Richter L, Ernst M, Ecker GF, Sigel E. Baur R, et al. Among authors: ernst m. J Neurochem. 2013 Jul;126(1):29-36. doi: 10.1111/jnc.12270. Epub 2013 May 3. J Neurochem. 2013. PMID: 23600744 Free article.

8

Accelerated discovery of novel benzodiazepine ligands by experiment-guided virtual screening.

Middendorp SJ, Puthenkalam R, Baur R, Ernst M, Sigel E. Middendorp SJ, et al. Among authors: ernst m. ACS Chem Biol. 2014 Aug 15;9(8):1854-9. doi: 10.1021/cb5001873. Epub 2014 Jun 27. ACS Chem Biol. 2014. PMID: 24960548

9

A pentasymmetric open channel blocker for Cys-loop receptor channels.

Carta V, Pangerl M, Baur R, Puthenkalam R, Ernst M, Trauner D, Sigel E. Carta V, et al. Among authors: ernst m. PLoS One. 2014 Sep 3;9(9):e106688. doi: 10.1371/journal.pone.0106688. eCollection 2014. PLoS One. 2014. PMID: 25184303 Free PMC article.

10

Metal-assisted synthesis of unsymmetrical magnolol and honokiol analogs and their biological assessment as GABAA receptor ligands.

Rycek L, Puthenkalam R, Schnürch M, Ernst M, Mihovilovic MD. Rycek L, et al. Among authors: ernst m. Bioorg Med Chem Lett. 2015 Jan 15;25(2):400-3. doi: 10.1016/j.bmcl.2014.10.091. Epub 2014 Nov 4. Bioorg Med Chem Lett. 2015. PMID: 25510374 Free PMC article.

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