Gaspar A - Search Results

1

Discovery of New Chemical Entities for Old Targets: Insights on the Lead Optimization of Chromone-Based Monoamine Oxidase B (MAO-B) Inhibitors.

Reis J, Cagide F, Chavarria D, Silva T, Fernandes C, Gaspar A, Uriarte E, Remião F, Alcaro S, Ortuso F, Borges F. Reis J, et al. Among authors: gaspar a. J Med Chem. 2016 Jun 23;59(12):5879-93. doi: 10.1021/acs.jmedchem.6b00527. Epub 2016 Jun 10. J Med Chem. 2016. PMID: 27244485

2

Antioxidant versus cytotoxic properties of hydroxycinnamic acid derivatives - a new paradigm in phenolic research.

Esteves M, Siquet C, Gaspar A, Rio V, Sousa JB, Reis S, Marques MP, Borges F. Esteves M, et al. Among authors: gaspar a. Arch Pharm (Weinheim). 2008 Mar;341(3):164-73. doi: 10.1002/ardp.200700168. Arch Pharm (Weinheim). 2008. PMID: 18275037

3

New insights into the antioxidant activity of hydroxycinnamic acids: Synthesis and physicochemical characterization of novel halogenated derivatives.

Gaspar A, Garrido EM, Esteves M, Quezada E, Milhazes N, Garrido J, Borges F. Gaspar A, et al. Eur J Med Chem. 2009 May;44(5):2092-9. doi: 10.1016/j.ejmech.2008.10.027. Epub 2008 Nov 5. Eur J Med Chem. 2009. PMID: 19058883

4

Chromone-2- and -3-carboxylic acids inhibit differently monoamine oxidases A and B.

Alcaro S, Gaspar A, Ortuso F, Milhazes N, Orallo F, Uriarte E, Yáñez M, Borges F. Alcaro S, et al. Among authors: gaspar a. Bioorg Med Chem Lett. 2010 May 1;20(9):2709-12. doi: 10.1016/j.bmcl.2010.03.081. Epub 2010 Mar 27. Bioorg Med Chem Lett. 2010. PMID: 20382016

5

Dietary phenolic acids and derivatives. Evaluation of the antioxidant activity of sinapic acid and its alkyl esters.

Gaspar A, Martins M, Silva P, Garrido EM, Garrido J, Firuzi O, Miri R, Saso L, Borges F. Gaspar A, et al. J Agric Food Chem. 2010 Nov 10;58(21):11273-80. doi: 10.1021/jf103075r. Epub 2010 Oct 15. J Agric Food Chem. 2010. PMID: 20949946

6

Chromone 3-phenylcarboxamides as potent and selective MAO-B inhibitors.

Gaspar A, Reis J, Fonseca A, Milhazes N, Viña D, Uriarte E, Borges F. Gaspar A, et al. Bioorg Med Chem Lett. 2011 Jan 15;21(2):707-9. doi: 10.1016/j.bmcl.2010.11.128. Epub 2010 Dec 5. Bioorg Med Chem Lett. 2011. PMID: 21194943

7

Synthesis and antioxidant activity of long chain alkyl hydroxycinnamates.

Menezes JC, Kamat SP, Cavaleiro JA, Gaspar A, Garrido J, Borges F. Menezes JC, et al. Among authors: gaspar a. Eur J Med Chem. 2011 Feb;46(2):773-7. doi: 10.1016/j.ejmech.2010.12.016. Epub 2010 Dec 21. Eur J Med Chem. 2011. PMID: 21216503

8

Towards the discovery of a novel class of monoamine oxidase inhibitors: structure-property-activity and docking studies on chromone amides.

Gaspar A, Teixeira F, Uriarte E, Milhazes N, Melo A, Cordeiro MN, Ortuso F, Alcaro S, Borges F. Gaspar A, et al. ChemMedChem. 2011 Apr 4;6(4):628-32. doi: 10.1002/cmdc.201000452. Epub 2011 Jan 25. ChemMedChem. 2011. PMID: 21442758 No abstract available.

9

Chromone, a privileged scaffold for the development of monoamine oxidase inhibitors.

Gaspar A, Silva T, Yáñez M, Vina D, Orallo F, Ortuso F, Uriarte E, Alcaro S, Borges F. Gaspar A, et al. J Med Chem. 2011 Jul 28;54(14):5165-73. doi: 10.1021/jm2004267. Epub 2011 Jul 1. J Med Chem. 2011. PMID: 21696156

10

Alkyl esters of hydroxycinnamic acids with improved antioxidant activity and lipophilicity protect PC12 cells against oxidative stress.

Garrido J, Gaspar A, Garrido EM, Miri R, Tavakkoli M, Pourali S, Saso L, Borges F, Firuzi O. Garrido J, et al. Among authors: gaspar a. Biochimie. 2012 Apr;94(4):961-7. doi: 10.1016/j.biochi.2011.12.015. Epub 2011 Dec 23. Biochimie. 2012. PMID: 22210493

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