Burnett DA - Search Results

1

Discovery of Novel Tricyclic Heterocycles as Potent and Selective DPP-4 Inhibitors for the Treatment of Type 2 Diabetes.

Wu WL, Hao J, Domalski M, Burnett DA, Pissarnitski D, Zhao Z, Stamford A, Scapin G, Gao YD, Soriano A, Kelly TM, Yao Z, Powles MA, Chen S, Mei H, Hwa J. Wu WL, et al. Among authors: burnett da. ACS Med Chem Lett. 2016 Mar 12;7(5):498-501. doi: 10.1021/acsmedchemlett.6b00027. eCollection 2016 May 12. ACS Med Chem Lett. 2016. PMID: 27190600 Free PMC article.

2

2-Azetidinone cholesterol absorption inhibitors: structure-activity relationships on the heterocyclic nucleus.

Clader JW, Burnett DA, Caplen MA, Domalski MS, Dugar S, Vaccaro W, Sher R, Browne ME, Zhao H, Burrier RE, Salisbury B, Davis HR Jr. Clader JW, et al. Among authors: burnett da. J Med Chem. 1996 Sep 13;39(19):3684-93. doi: 10.1021/jm960405n. J Med Chem. 1996. PMID: 8809157

3

Structure-activity relationships of pyrroloquinazolines as thrombin receptor antagonists.

Ahn HS, Arik L, Boykow G, Burnett DA, Caplen MA, Czarniecki M, Domalski MS, Foster C, Manna M, Stamford AW, Wu Y. Ahn HS, et al. Among authors: burnett da. Bioorg Med Chem Lett. 1999 Jul 19;9(14):2073-8. doi: 10.1016/s0960-894x(99)00339-x. Bioorg Med Chem Lett. 1999. PMID: 10450984

4

Synthesis of iodinated biochemical tools related to the 2-azetidinone class of cholesterol absorption inhibitors.

Burnett DA, Caplen MA, Domalski MS, Browne ME, Davis HR Jr, Clader JW. Burnett DA, et al. Bioorg Med Chem Lett. 2002 Feb 11;12(3):311-4. doi: 10.1016/s0960-894x(01)00750-8. Bioorg Med Chem Lett. 2002. PMID: 11814785

5

Synthesis and structure-activity relationships of aminoalkylazetidines as ORL1 receptor ligands.

Wu WL, Caplen MA, Domalski MS, Zhang H, Fawzi A, Burnett DA. Wu WL, et al. Among authors: burnett da. Bioorg Med Chem Lett. 2002 Nov 4;12(21):3157-60. doi: 10.1016/s0960-894x(02)00652-2. Bioorg Med Chem Lett. 2002. PMID: 12372523

6

Dopamine D1/D5 receptor antagonists with improved pharmacokinetics: design, synthesis, and biological evaluation of phenol bioisosteric analogues of benzazepine D1/D5 antagonists.

Wu WL, Burnett DA, Spring R, Greenlee WJ, Smith M, Favreau L, Fawzi A, Zhang H, Lachowicz JE. Wu WL, et al. Among authors: burnett da. J Med Chem. 2005 Feb 10;48(3):680-93. doi: 10.1021/jm030614p. J Med Chem. 2005. PMID: 15689153

7

Synthesis and structure-activity relationships of piperidine-based melanin-concentrating hormone receptor 1 antagonists.

Wu WL, Burnett DA, Spring R, Qiang L, Sasikumar TK, Domalski MS, Greenlee WJ, O'Neill K, Hawes BE. Wu WL, et al. Among authors: burnett da. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3668-73. doi: 10.1016/j.bmcl.2006.04.061. Epub 2006 May 11. Bioorg Med Chem Lett. 2006. PMID: 16690312

8

Design and synthesis of orally efficacious benzimidazoles as melanin-concentrating hormone receptor 1 antagonists.

Wu WL, Burnett DA, Caplen MA, Domalski MS, Bennett C, Greenlee WJ, Hawes BE, O'Neill K, Weig B, Weston D, Spar B, Kowalski T. Wu WL, et al. Among authors: burnett da. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3674-8. doi: 10.1016/j.bmcl.2006.04.062. Epub 2006 May 11. Bioorg Med Chem Lett. 2006. PMID: 16690315

9

Discovery of orally efficacious tetracyclic metabotropic glutamate receptor 1 (mGluR1) antagonists for the treatment of chronic pain.

Wu WL, Burnett DA, Domalski M, Greenlee WJ, Li C, Bertorelli R, Fredduzzi S, Lozza G, Veltri A, Reggiani A. Wu WL, et al. Among authors: burnett da. J Med Chem. 2007 Nov 15;50(23):5550-3. doi: 10.1021/jm070590c. Epub 2007 Oct 11. J Med Chem. 2007. PMID: 17929793

10

Tricyclic thienopyridine-pyrimidones/thienopyrimidine-pyrimidones as orally efficacious mGluR1 antagonists for neuropathic pain.

Sasikumar TK, Qiang L, Burnett DA, Greenlee WJ, Li C, Heimark L, Pramanik B, Grilli M, Bertorelli R, Lozza G, Reggiani A. Sasikumar TK, et al. Among authors: burnett da. Bioorg Med Chem Lett. 2009 Jun 15;19(12):3199-203. doi: 10.1016/j.bmcl.2009.04.104. Epub 2009 May 3. Bioorg Med Chem Lett. 2009. PMID: 19433355

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