Akram M - Search Results

1

Pharmacophore Models and Pharmacophore-Based Virtual Screening: Concepts and Applications Exemplified on Hydroxysteroid Dehydrogenases.

Kaserer T, Beck KR, Akram M, Odermatt A, Schuster D. Kaserer T, et al. Among authors: akram m. Molecules. 2015 Dec 19;20(12):22799-832. doi: 10.3390/molecules201219880. Molecules. 2015. PMID: 26703541 Free PMC article. Review.

2

Inhibition of 11β-hydroxysteroid dehydrogenase 2 by the fungicides itraconazole and posaconazole.

Beck KR, Bächler M, Vuorinen A, Wagner S, Akram M, Griesser U, Temml V, Klusonova P, Yamaguchi H, Schuster D, Odermatt A. Beck KR, et al. Among authors: akram m. Biochem Pharmacol. 2017 Apr 15;130:93-103. doi: 10.1016/j.bcp.2017.01.010. Epub 2017 Jan 25. Biochem Pharmacol. 2017. PMID: 28131847 Free PMC article.

3

Potential Antiosteoporotic Natural Product Lead Compounds That Inhibit 17β-Hydroxysteroid Dehydrogenase Type 2.

Vuorinen A, Engeli RT, Leugger S, Bachmann F, Akram M, Atanasov AG, Waltenberger B, Temml V, Stuppner H, Krenn L, Ateba SB, Njamen D, Davis RA, Odermatt A, Schuster D. Vuorinen A, et al. Among authors: akram m. J Nat Prod. 2017 Apr 28;80(4):965-974. doi: 10.1021/acs.jnatprod.6b00950. Epub 2017 Mar 20. J Nat Prod. 2017. PMID: 28319389 Free PMC article.

4

A combinatorial approach for the discovery of cytochrome P450 2D6 inhibitors from nature.

Hochleitner J, Akram M, Ueberall M, Davis RA, Waltenberger B, Stuppner H, Sturm S, Ueberall F, Gostner JM, Schuster D. Hochleitner J, et al. Among authors: akram m. Sci Rep. 2017 Aug 14;7(1):8071. doi: 10.1038/s41598-017-08404-0. Sci Rep. 2017. PMID: 28808272 Free PMC article.

5

Pharmacophore Modeling and in Silico/in Vitro Screening for Human Cytochrome P450 11B1 and Cytochrome P450 11B2 Inhibitors.

Akram M, Waratchareeyakul W, Haupenthal J, Hartmann RW, Schuster D. Akram M, et al. Front Chem. 2017 Dec 19;5:104. doi: 10.3389/fchem.2017.00104. eCollection 2017. Front Chem. 2017. PMID: 29312923 Free PMC article.

6

Identification of the fungicide epoxiconazole by virtual screening and biological assessment as inhibitor of human 11β-hydroxylase and aldosterone synthase.

Akram M, Patt M, Kaserer T, Temml V, Waratchareeyakul W, Kratschmar DV, Haupenthal J, Hartmann RW, Odermatt A, Schuster D. Akram M, et al. J Steroid Biochem Mol Biol. 2019 Sep;192:105358. doi: 10.1016/j.jsbmb.2019.04.007. Epub 2019 Apr 6. J Steroid Biochem Mol Biol. 2019. PMID: 30965118

7

Honokiol and Magnolol: Insights into Their Antidermatophytic Effects.

Trifan A, Bostănaru AC, Luca SV, Temml V, Akram M, Herdlinger S, Kulinowski Ł, Skalicka-Woźniak K, Granica S, Czerwińska ME, Kruk A, Greige-Gerges H, Mareș M, Schuster D. Trifan A, et al. Among authors: akram m. Plants (Basel). 2021 Nov 19;10(11):2522. doi: 10.3390/plants10112522. Plants (Basel). 2021. PMID: 34834886 Free PMC article.

8

Synthesis, Crystal Structure, DFT Calculations, Hirshfeld Surface Analysis and In Silico Drug-Target Profiling of (R)-2-(2-(1,3-Dioxoisoindolin-2-yl)propanamido)benzoic Acid Methyl Ester.

Rubab SL, Raza AR, Nisar B, Ashfaq M, Altaf Y, Hussain R, Sajjad N, Akram MS, Tahir MN, Shaheen MA, Rehman MFU, Ali HM. Rubab SL, et al. Among authors: akram ms. Molecules. 2023 May 26;28(11):4375. doi: 10.3390/molecules28114375. Molecules. 2023. PMID: 37298851 Free PMC article.

9

Synthesis, crystal structure determination, biological screening and docking studies of N¹-substituted derivatives of 2,3-dihydroquinazolin-4(1H)-one as inhibitors of cholinesterases.

Sultana N, Sarfraz M, Tanoli ST, Akram MS, Sadiq A, Rashid U, Tariq MI. Sultana N, et al. Among authors: akram ms. Bioorg Chem. 2017 Jun;72:256-267. doi: 10.1016/j.bioorg.2017.04.009. Epub 2017 Apr 17. Bioorg Chem. 2017. PMID: 28495556

10

Synthesis, biological evaluation and docking studies of 2,3-dihydroquinazolin-4(1H)-one derivatives as inhibitors of cholinesterases.

Sarfraz M, Sultana N, Rashid U, Akram MS, Sadiq A, Tariq MI. Sarfraz M, et al. Among authors: akram ms. Bioorg Chem. 2017 Feb;70:237-244. doi: 10.1016/j.bioorg.2017.01.004. Epub 2017 Jan 17. Bioorg Chem. 2017. PMID: 28126287 Free article.

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