Gunther JR - Search Results

1

Estrogen receptor alpha/co-activator interaction assay: TR-FRET.

Moore TW, Gunther JR, Katzenellenbogen JA. Moore TW, et al. Among authors: gunther jr. Methods Mol Biol. 2015;1278:545-53. doi: 10.1007/978-1-4939-2425-7_36. Methods Mol Biol. 2015. PMID: 25859975 Free PMC article.

2

Bicyclo[2.2.2]octanes: close structural mimics of the nuclear receptor-binding motif of steroid receptor coactivators.

Zhou HB, Collins ML, Gunther JR, Comninos JS, Katzenellenbogen JA. Zhou HB, et al. Among authors: gunther jr. Bioorg Med Chem Lett. 2007 Aug 1;17(15):4118-22. doi: 10.1016/j.bmcl.2007.05.058. Epub 2007 May 23. Bioorg Med Chem Lett. 2007. PMID: 17560105 Free PMC article.

3

Blocking estrogen signaling after the hormone: pyrimidine-core inhibitors of estrogen receptor-coactivator binding.

Parent AA, Gunther JR, Katzenellenbogen JA. Parent AA, et al. Among authors: gunther jr. J Med Chem. 2008 Oct 23;51(20):6512-30. doi: 10.1021/jm800698b. Epub 2008 Sep 12. J Med Chem. 2008. PMID: 18785725 Free PMC article.

4

Nonclassical SNAPFL analogue as a Cy5 resonance energy transfer partner.

Kim SH, Gunther JR, Katzenellenbogen JA. Kim SH, et al. Among authors: gunther jr. Org Lett. 2008 Nov 6;10(21):4931-4. doi: 10.1021/ol801907b. Epub 2008 Oct 9. Org Lett. 2008. PMID: 18841988 Free PMC article.

5

Synthesis and biological evaluation of guanylhydrazone coactivator binding inhibitors for the estrogen receptor.

LaFrate AL, Gunther JR, Carlson KE, Katzenellenbogen JA. LaFrate AL, et al. Among authors: gunther jr. Bioorg Med Chem. 2008 Dec 1;16(23):10075-84. doi: 10.1016/j.bmc.2008.10.007. Epub 2008 Oct 7. Bioorg Med Chem. 2008. PMID: 18976929 Free PMC article.

6

A set of time-resolved fluorescence resonance energy transfer assays for the discovery of inhibitors of estrogen receptor-coactivator binding.

Gunther JR, Du Y, Rhoden E, Lewis I, Revennaugh B, Moore TW, Kim SH, Dingledine R, Fu H, Katzenellenbogen JA. Gunther JR, et al. J Biomol Screen. 2009 Feb;14(2):181-93. doi: 10.1177/1087057108329349. Epub 2009 Feb 4. J Biomol Screen. 2009. PMID: 19196699 Free PMC article.

7

Monitoring a coordinated exchange process in a four-component biological interaction system: development of a time-resolved terbium-based one-donor/three-acceptor multicolor FRET system.

Kim SH, Gunther JR, Katzenellenbogen JA. Kim SH, et al. Among authors: gunther jr. J Am Chem Soc. 2010 Apr 7;132(13):4685-92. doi: 10.1021/ja100248q. J Am Chem Soc. 2010. PMID: 20230029 Free PMC article.

8

Probing the topological tolerance of multimeric protein interactions: evaluation of an estrogen/synthetic ligand for FK506 binding protein conjugate.

Moore TW, Gunther JR, Katzenellenbogen JA. Moore TW, et al. Among authors: gunther jr. Bioconjug Chem. 2010 Oct 20;21(10):1880-9. doi: 10.1021/bc100266v. Bioconjug Chem. 2010. PMID: 20919698 Free PMC article.

9

Exploration of dimensions of estrogen potency: parsing ligand binding and coactivator binding affinities.

Jeyakumar M, Carlson KE, Gunther JR, Katzenellenbogen JA. Jeyakumar M, et al. Among authors: gunther jr. J Biol Chem. 2011 Apr 15;286(15):12971-82. doi: 10.1074/jbc.M110.205112. Epub 2011 Feb 14. J Biol Chem. 2011. PMID: 21321128 Free PMC article.

10

Amphipathic benzenes are designed inhibitors of the estrogen receptor alpha/steroid receptor coactivator interaction.

Gunther JR, Moore TW, Collins ML, Katzenellenbogen JA. Gunther JR, et al. ACS Chem Biol. 2008 May 16;3(5):282-6. doi: 10.1021/cb800056r. ACS Chem Biol. 2008. PMID: 18484708 Free PMC article.

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