Pieroni M - Search Results

1

Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A.

Pieroni M, Annunziato G, Azzali E, Dessanti P, Mercurio C, Meroni G, Trifiró P, Vianello P, Villa M, Beato C, Varasi M, Costantino G. Pieroni M, et al. Eur J Med Chem. 2015 Mar 6;92:377-86. doi: 10.1016/j.ejmech.2014.12.032. Epub 2015 Jan 7. Eur J Med Chem. 2015. PMID: 25585008

2

Synthesis, biological evaluation, and structure-activity relationships for 5-[(E)-2-arylethenyl]-3-isoxazolecarboxylic acid alkyl ester derivatives as valuable antitubercular chemotypes.

Pieroni M, Lilienkampf A, Wan B, Wang Y, Franzblau SG, Kozikowski AP. Pieroni M, et al. J Med Chem. 2009 Oct 22;52(20):6287-96. doi: 10.1021/jm900513a. J Med Chem. 2009. PMID: 19757815

3

Rational design of 5-phenyl-3-isoxazolecarboxylic acid ethyl esters as growth inhibitors of Mycobacterium tuberculosis. a potent and selective series for further drug development.

Lilienkampf A, Pieroni M, Wan B, Wang Y, Franzblau SG, Kozikowski AP. Lilienkampf A, et al. Among authors: pieroni m. J Med Chem. 2010 Jan 28;53(2):678-88. doi: 10.1021/jm901273n. J Med Chem. 2010. PMID: 20000577

4

From 6-aminoquinolone antibacterials to 6-amino-7-thiopyranopyridinylquinolone ethyl esters as inhibitors of Staphylococcus aureus multidrug efflux pumps.

Pieroni M, Dimovska M, Brincat JP, Sabatini S, Carosati E, Massari S, Kaatz GW, Fravolini A. Pieroni M, et al. J Med Chem. 2010 Jun 10;53(11):4466-80. doi: 10.1021/jm1003304. J Med Chem. 2010. PMID: 20446747

5

Synthesis, biological evaluation, and structure-activity relationships of N-benzoyl-2-hydroxybenzamides as agents active against P. falciparum (K1 strain), Trypanosomes, and Leishmania.

Stec J, Huang Q, Pieroni M, Kaiser M, Fomovska A, Mui E, Witola WH, Bettis S, McLeod R, Brun R, Kozikowski AP. Stec J, et al. Among authors: pieroni m. J Med Chem. 2012 Apr 12;55(7):3088-100. doi: 10.1021/jm2015183. Epub 2012 Mar 20. J Med Chem. 2012. PMID: 22352841 Free PMC article.

6

Design, synthesis and investigation on the structure-activity relationships of N-substituted 2-aminothiazole derivatives as antitubercular agents.

Pieroni M, Wan B, Cho S, Franzblau SG, Costantino G. Pieroni M, et al. Eur J Med Chem. 2014 Jan 24;72:26-34. doi: 10.1016/j.ejmech.2013.11.007. Epub 2013 Nov 13. Eur J Med Chem. 2014. PMID: 24333612

7

Inhibitors of the sulfur assimilation pathway in bacterial pathogens as enhancers of antibiotic therapy.

Campanini B, Pieroni M, Raboni S, Bettati S, Benoni R, Pecchini C, Costantino G, Mozzarelli A. Campanini B, et al. Among authors: pieroni m. Curr Med Chem. 2015;22(2):187-213. doi: 10.2174/0929867321666141112122553. Curr Med Chem. 2015. PMID: 25388010 Review.

8

Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design.

Pieroni M, Wan B, Zuliani V, Franzblau SG, Costantino G, Rivara M. Pieroni M, et al. Eur J Med Chem. 2015 Jul 15;100:44-9. doi: 10.1016/j.ejmech.2015.05.048. Epub 2015 Jun 5. Eur J Med Chem. 2015. PMID: 26071857

9

Cyclopropane derivatives as potential human serine racemase inhibitors: unveiling novel insights into a difficult target.

Beato C, Pecchini C, Cocconcelli C, Campanini B, Marchetti M, Pieroni M, Mozzarelli A, Costantino G. Beato C, et al. Among authors: pieroni m. J Enzyme Inhib Med Chem. 2016 Aug;31(4):645-52. doi: 10.3109/14756366.2015.1057720. Epub 2015 Jul 2. J Enzyme Inhib Med Chem. 2016. PMID: 26133542 Free article.

10

Rational Design and Synthesis of Thioridazine Analogues as Enhancers of the Antituberculosis Therapy.

Pieroni M, Machado D, Azzali E, Santos Costa S, Couto I, Costantino G, Viveiros M. Pieroni M, et al. J Med Chem. 2015 Aug 13;58(15):5842-53. doi: 10.1021/acs.jmedchem.5b00428. Epub 2015 Aug 3. J Med Chem. 2015. PMID: 26197353

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