Case BL - Search Results

1

Discovery of an Oral Potent Selective Inhibitor of Hematopoietic Prostaglandin D Synthase (HPGDS).

Carron CP, Trujillo JI, Olson KL, Huang W, Hamper BC, Dice T, Neal BE, Pelc MJ, Day JE, Rohrer DC, Kiefer JR, Moon JB, Schweitzer BA, Blake TD, Turner SR, Woerndle R, Case BL, Bono CP, Dilworth VM, Funckes-Shippy CL, Hood BL, Jerome GM, Kornmeier CM, Radabaugh MR, Williams ML, Davies MS, Wegner CD, Welsch DJ, Abraham WM, Warren CJ, Dowty ME, Hua F, Zutshi A, Yang JZ, Thorarensen A. Carron CP, et al. Among authors: case bl. ACS Med Chem Lett. 2010 Feb 2;1(2):59-63. doi: 10.1021/ml900025z. eCollection 2010 May 13. ACS Med Chem Lett. 2010. PMID: 24900177 Free PMC article.

2

Discovery of novel cyanodihydropyridines as potent mineralocorticoid receptor antagonists.

Arhancet GB, Woodard SS, Iyanar K, Case BL, Woerndle R, Dietz JD, Garland DJ, Collins JT, Payne MA, Blinn JR, Pomposiello SI, Hu X, Heron MI, Huang HC, Lee LF. Arhancet GB, et al. Among authors: case bl. J Med Chem. 2010 Aug 26;53(16):5970-8. doi: 10.1021/jm100506y. J Med Chem. 2010. PMID: 20672820

3

Piperazinyl-glutamate-pyrimidines as potent P2Y12 antagonists for inhibition of platelet aggregation.

Parlow JJ, Burney MW, Case BL, Girard TJ, Hall KA, Hiebsch RR, Huff RM, Lachance RM, Mischke DA, Rapp SR, Woerndle RS, Ennis MD. Parlow JJ, et al. Among authors: case bl. Bioorg Med Chem Lett. 2009 Nov 1;19(21):6148-56. doi: 10.1016/j.bmcl.2009.09.017. Epub 2009 Sep 10. Bioorg Med Chem Lett. 2009. PMID: 19796941

4

Piperazinyl glutamate pyridines as potent orally bioavailable P2Y12 antagonists for inhibition of platelet aggregation.

Parlow JJ, Burney MW, Case BL, Girard TJ, Hall KA, Harris PK, Hiebsch RR, Huff RM, Lachance RM, Mischke DA, Rapp SR, Woerndle RS, Ennis MD. Parlow JJ, et al. Among authors: case bl. J Med Chem. 2010 Mar 11;53(5):2010-37. doi: 10.1021/jm901518t. J Med Chem. 2010. PMID: 20141147

5

Biochemical, cellular, and anti-inflammatory properties of a potent, selective, orally bioavailable benzamide inhibitor of Rho kinase activity.

Rajagopalan LE, Davies MS, Kahn LE, Kornmeier CM, Shimada H, Steiner TA, Zweifel BS, Wendling JM, Payne MA, Loeffler RF, Case BL, Norton MB, Parikh MD, Nemirovskiy OV, Mourey RJ, Masferrer JL, Misko TP, Kolodziej SA. Rajagopalan LE, et al. Among authors: case bl. J Pharmacol Exp Ther. 2010 Jun;333(3):707-16. doi: 10.1124/jpet.110.166033. Epub 2010 Mar 12. J Pharmacol Exp Ther. 2010. PMID: 20228155

6

Piperazinyl-glutamate-pyridines as potent orally bioavailable P2Y12 antagonists for inhibition of platelet aggregation.

Parlow JJ, Burney MW, Case BL, Girard TJ, Hall KA, Hiebsch RR, Huff RM, Lachance RM, Mischke DA, Rapp SR, Woerndle RS, Ennis MD. Parlow JJ, et al. Among authors: case bl. Bioorg Med Chem Lett. 2009 Aug 15;19(16):4657-63. doi: 10.1016/j.bmcl.2009.06.075. Epub 2009 Jun 25. Bioorg Med Chem Lett. 2009. PMID: 19604694

7

Part II: piperazinyl-glutamate-pyridines as potent orally bioavailable P2Y12 antagonists for inhibition of platelet aggregation.

Parlow JJ, Burney MW, Case BL, Girard TJ, Hall KA, Harris PK, Hiebsch RR, Huff RM, Lachance RM, Mischke DA, Rapp SR, Woerndle RS, Ennis MD. Parlow JJ, et al. Among authors: case bl. Bioorg Med Chem Lett. 2010 Feb 15;20(4):1388-94. doi: 10.1016/j.bmcl.2009.12.110. Epub 2010 Jan 4. Bioorg Med Chem Lett. 2010. PMID: 20097563

8

A method for determining whether hypotension caused by novel compounds in preclinical development results from histamine release.

Blom JD, Yang PC, Nicholson NS, Case BL, Parlow JJ, South MS, Wegner CD. Blom JD, et al. Among authors: case bl. J Pharmacol Toxicol Methods. 2004 Jan-Feb;49(1):31-7. doi: 10.1016/j.vascn.2003.08.002. J Pharmacol Toxicol Methods. 2004. PMID: 14670692

9

Design, parallel synthesis, and crystal structures of pyrazinone antithrombotics as selective inhibitors of the tissue factor VIIa complex.

Parlow JJ, Case BL, Dice TA, Fenton RL, Hayes MJ, Jones DE, Neumann WL, Wood RS, Lachance RM, Girard TJ, Nicholson NS, Clare M, Stegeman RA, Stevens AM, Stallings WC, Kurumbail RG, South MS. Parlow JJ, et al. Among authors: case bl. J Med Chem. 2003 Sep 11;46(19):4050-62. doi: 10.1021/jm030131l. J Med Chem. 2003. PMID: 12954058

10

Multi-step polymer-assisted solution-phase (PASP) library synthesis of functionalized diaminobenzamides.

South MS, Case BL, Dice TA, Franklin GW, Hayes MJ, Jones DE, Lindmark RJ, Zeng Q, Parlow JJ. South MS, et al. Among authors: case bl. Comb Chem High Throughput Screen. 2000 Apr;3(2):139-51. doi: 10.2174/1386207003331724. Comb Chem High Throughput Screen. 2000. PMID: 10788585

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