Newman SP - Search Results

1

Synthesis, antitubulin, and antiproliferative SAR of C3/C1-substituted tetrahydroisoquinolines.

Dohle W, Leese MP, Jourdan FL, Major MR, Bai R, Hamel E, Ferrandis E, Kasprzyk PG, Fiore A, Newman SP, Purohit A, Potter BV. Dohle W, et al. Among authors: newman sp. ChemMedChem. 2014 Feb;9(2):350-70. doi: 10.1002/cmdc.201300412. Epub 2014 Jan 16. ChemMedChem. 2014. PMID: 24436228

2

Anti-cancer activities of novel D-ring modified 2-substituted estrogen-3-O-sulfamates.

Leese MP, Leblond B, Newman SP, Purohit A, Reed MJ, Potter BV. Leese MP, et al. Among authors: newman sp. J Steroid Biochem Mol Biol. 2005 Feb;94(1-3):239-51. doi: 10.1016/j.jsbmb.2005.01.005. Epub 2005 Feb 24. J Steroid Biochem Mol Biol. 2005. PMID: 15862971

3

2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity.

Leese MP, Leblond B, Smith A, Newman SP, Di Fiore A, De Simone G, Supuran CT, Purohit A, Reed MJ, Potter BV. Leese MP, et al. Among authors: newman sp. J Med Chem. 2006 Dec 28;49(26):7683-96. doi: 10.1021/jm060705x. J Med Chem. 2006. PMID: 17181151

4

3,17-disubstituted 2-alkylestra-1,3,5(10)-trien-3-ol derivatives: synthesis, in vitro and in vivo anticancer activity.

Bubert C, Leese MP, Mahon MF, Ferrandis E, Regis-Lydi S, Kasprzyk PG, Newman SP, Ho YT, Purohit A, Reed MJ, Potter BV. Bubert C, et al. Among authors: newman sp. J Med Chem. 2007 Sep 6;50(18):4431-43. doi: 10.1021/jm070405v. Epub 2007 Aug 15. J Med Chem. 2007. PMID: 17696419

5

Structure-activity relationships of C-17 cyano-substituted estratrienes as anticancer agents.

Leese MP, Jourdan FL, Gaukroger K, Mahon MF, Newman SP, Foster PA, Stengel C, Regis-Lydi S, Ferrandis E, Di Fiore A, De Simone G, Supuran CT, Purohit A, Reed MJ, Potter BV. Leese MP, et al. Among authors: newman sp. J Med Chem. 2008 Mar 13;51(5):1295-308. doi: 10.1021/jm701319c. Epub 2008 Feb 9. J Med Chem. 2008. PMID: 18260615

6

Effects of C-17 heterocyclic substituents on the anticancer activity of 2-ethylestra-1,3,5(10)-triene-3-O-sulfamates: synthesis, in vitro evaluation and computational modelling.

Jourdan F, Bubert C, Leese MP, Smith A, Ferrandis E, Regis-Lydi S, Newman SP, Purohit A, Reed MJ, Potter BV. Jourdan F, et al. Among authors: newman sp. Org Biomol Chem. 2008 Nov 21;6(22):4108-19. doi: 10.1039/b810300c. Epub 2008 Sep 22. Org Biomol Chem. 2008. PMID: 18972041

7

Synthesis, antitubulin, and antiproliferative SAR of analogues of 2-methoxyestradiol-3,17-O,O-bis-sulfamate.

Jourdan F, Leese MP, Dohle W, Hamel E, Ferrandis E, Newman SP, Purohit A, Reed MJ, Potter BV. Jourdan F, et al. Among authors: newman sp. J Med Chem. 2010 Apr 8;53(7):2942-51. doi: 10.1021/jm9018806. J Med Chem. 2010. PMID: 20225862

8

Structure-activity relationships of C-17-substituted estratriene-3-O-sulfamates as anticancer agents.

Jourdan F, Leese MP, Dohle W, Ferrandis E, Newman SP, Chander S, Purohit A, Potter BV. Jourdan F, et al. Among authors: newman sp. J Med Chem. 2011 Jul 14;54(13):4863-79. doi: 10.1021/jm200483x. Epub 2011 Jun 9. J Med Chem. 2011. PMID: 21604672

9

Synthesis, anti-tubulin and antiproliferative SAR of steroidomimetic dihydroisoquinolinones.

Leese MP, Jourdan FL, Major MR, Dohle W, Thomas MP, Hamel E, Ferrandis E, Mahon MF, Newman SP, Purohit A, Potter BV. Leese MP, et al. Among authors: newman sp. ChemMedChem. 2014 Apr;9(4):798-812. doi: 10.1002/cmdc.201400017. Epub 2014 Mar 5. ChemMedChem. 2014. PMID: 24596315 Free PMC article.

10

A-ring-substituted estrogen-3-O-sulfamates: potent multitargeted anticancer agents.

Leese MP, Hejaz HA, Mahon MF, Newman SP, Purohit A, Reed MJ, Potter BV. Leese MP, et al. Among authors: newman sp. J Med Chem. 2005 Aug 11;48(16):5243-56. doi: 10.1021/jm050066a. J Med Chem. 2005. PMID: 16078843

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