Asami T - Search Results

1

Design, synthesis, and biological evaluation of novel investigational nonapeptide KISS1R agonists with testosterone-suppressive activity.

Asami T, Nishizawa N, Matsui H, Nishibori K, Ishibashi Y, Horikoshi Y, Nakayama M, Matsumoto S, Tarui N, Yamaguchi M, Matsumoto H, Ohtaki T, Kitada C. Asami T, et al. J Med Chem. 2013 Nov 14;56(21):8298-307. doi: 10.1021/jm401056w. Epub 2013 Oct 17. J Med Chem. 2013. PMID: 24047141

2

Design and synthesis of ETA receptor antagonists and study of ETA receptor distribution.

Kitada C, Ohtaki T, Masuda Y, Masuo Y, Nomura H, Asami T, Matsumoto Y, Satou M, Fujino M. Kitada C, et al. Among authors: asami t. J Cardiovasc Pharmacol. 1993;22 Suppl 8:S128-31. doi: 10.1097/00005344-199322008-00035. J Cardiovasc Pharmacol. 1993. PMID: 7509923

3

Cyclic hexapeptide endothelin receptor antagonists highly potent for both receptor subtypes ETA and ETB.

Kikuchi T, Ohtaki T, Kawata A, Imada T, Asami T, Masuda Y, Sugo T, Kusumoto K, Kubo K, Watanabe T, et al. Kikuchi T, et al. Among authors: asami t. Biochem Biophys Res Commun. 1994 May 16;200(3):1708-12. doi: 10.1006/bbrc.1994.1649. Biochem Biophys Res Commun. 1994. PMID: 8185629

4

Endothelin-1 analogues substituted at both position 18 and 19: highly potent endothelin antagonists with no selectivity for either receptor subtype ETA or ETB.

Kikuchi T, Kubo K, Ohtaki T, Suzuki N, Asami T, Shimamoto N, Wakimasu M, Fujino M. Kikuchi T, et al. Among authors: asami t. J Med Chem. 1993 Dec 10;36(25):4087-93. doi: 10.1021/jm00077a013. J Med Chem. 1993. PMID: 8258832

5

Identification of a neuropeptide modified with bromine as an endogenous ligand for GPR7.

Fujii R, Yoshida H, Fukusumi S, Habata Y, Hosoya M, Kawamata Y, Yano T, Hinuma S, Kitada C, Asami T, Mori M, Fujisawa Y, Fujino M. Fujii R, et al. Among authors: asami t. J Biol Chem. 2002 Sep 13;277(37):34010-6. doi: 10.1074/jbc.M205883200. Epub 2002 Jul 12. J Biol Chem. 2002. PMID: 12118011 Free article.

6

Identification of neuropeptide W as the endogenous ligand for orphan G-protein-coupled receptors GPR7 and GPR8.

Shimomura Y, Harada M, Goto M, Sugo T, Matsumoto Y, Abe M, Watanabe T, Asami T, Kitada C, Mori M, Onda H, Fujino M. Shimomura Y, et al. Among authors: asami t. J Biol Chem. 2002 Sep 27;277(39):35826-32. doi: 10.1074/jbc.M205337200. Epub 2002 Jul 18. J Biol Chem. 2002. PMID: 12130646 Free article.

7

Development and validation of sensitive sandwich ELISAs for two investigational nonapeptide metastin receptor agonists, TAK-448 and TAK-683.

Yoshida N, Nishizawa N, Matsui H, Moriya Y, Kitada C, Asami T, Matsumoto H. Yoshida N, et al. Among authors: asami t. J Pharm Biomed Anal. 2012 Nov;70:369-77. doi: 10.1016/j.jpba.2012.05.033. Epub 2012 Jun 1. J Pharm Biomed Anal. 2012. PMID: 22748666

8

Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides.

Asami T, Nishizawa N, Ishibashi Y, Nishibori K, Nakayama M, Horikoshi Y, Matsumoto S, Yamaguchi M, Matsumoto H, Tarui N, Ohtaki T, Kitada C. Asami T, et al. Bioorg Med Chem Lett. 2012 Oct 15;22(20):6391-6. doi: 10.1016/j.bmcl.2012.08.069. Epub 2012 Aug 23. Bioorg Med Chem Lett. 2012. PMID: 22975302

9

Trypsin resistance of a decapeptide KISS1R agonist containing an Nω-methylarginine substitution.

Asami T, Nishizawa N, Ishibashi Y, Nishibori K, Horikoshi Y, Matsumoto H, Ohtaki T, Kitada C. Asami T, et al. Bioorg Med Chem Lett. 2012 Oct 15;22(20):6328-32. doi: 10.1016/j.bmcl.2012.08.087. Epub 2012 Aug 30. Bioorg Med Chem Lett. 2012. PMID: 22995619

10

Chronic administration of the metastin/kisspeptin analog KISS1-305 or the investigational agent TAK-448 suppresses hypothalamic pituitary gonadal function and depletes plasma testosterone in adult male rats.

Matsui H, Tanaka A, Yokoyama K, Takatsu Y, Ishikawa K, Asami T, Nishizawa N, Suzuki A, Kumano S, Terada M, Kusaka M, Kitada C, Ohtaki T. Matsui H, et al. Among authors: asami t. Endocrinology. 2012 Nov;153(11):5297-308. doi: 10.1210/en.2012-1388. Epub 2012 Oct 1. Endocrinology. 2012. PMID: 23027808

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