Keov P - Search Results

1

Reverse engineering of the selective agonist TBPB unveils both orthosteric and allosteric modes of action at the M₁ muscarinic acetylcholine receptor.

Keov P, Valant C, Devine SM, Lane JR, Scammells PJ, Sexton PM, Christopoulos A. Keov P, et al. Mol Pharmacol. 2013 Sep;84(3):425-37. doi: 10.1124/mol.113.087320. Epub 2013 Jun 24. Mol Pharmacol. 2013. PMID: 23798605

2

Allosteric modulation of G protein-coupled receptors: a pharmacological perspective.

Keov P, Sexton PM, Christopoulos A. Keov P, et al. Neuropharmacology. 2011 Jan;60(1):24-35. doi: 10.1016/j.neuropharm.2010.07.010. Epub 2010 Jul 15. Neuropharmacology. 2011. PMID: 20637785 Review.

3

Molecular determinants of allosteric modulation at the M1 muscarinic acetylcholine receptor.

Abdul-Ridha A, López L, Keov P, Thal DM, Mistry SN, Sexton PM, Lane JR, Canals M, Christopoulos A. Abdul-Ridha A, et al. Among authors: keov p. J Biol Chem. 2014 Feb 28;289(9):6067-79. doi: 10.1074/jbc.M113.539080. Epub 2014 Jan 17. J Biol Chem. 2014. PMID: 24443568 Free PMC article.

4

Molecular mechanisms of bitopic ligand engagement with the M1 muscarinic acetylcholine receptor.

Keov P, López L, Devine SM, Valant C, Lane JR, Scammells PJ, Sexton PM, Christopoulos A. Keov P, et al. J Biol Chem. 2014 Aug 22;289(34):23817-37. doi: 10.1074/jbc.M114.582874. Epub 2014 Jul 8. J Biol Chem. 2014. PMID: 25006252 Free PMC article.

5

AM833 Is a Novel Agonist of Calcitonin Family G Protein-Coupled Receptors: Pharmacological Comparison with Six Selective and Nonselective Agonists.

Fletcher MM, Keov P, Truong TT, Mennen G, Hick CA, Zhao P, Furness SGB, Kruse T, Clausen TR, Wootten D, Sexton PM. Fletcher MM, et al. Among authors: keov p. J Pharmacol Exp Ther. 2021 Jun;377(3):417-440. doi: 10.1124/jpet.121.000567. Epub 2021 Mar 16. J Pharmacol Exp Ther. 2021. PMID: 33727283

6

Development of a human vasopressin V_1a-receptor antagonist from an evolutionary-related insect neuropeptide.

Di Giglio MG, Muttenthaler M, Harpsøe K, Liutkeviciute Z, Keov P, Eder T, Rattei T, Arrowsmith S, Wray S, Marek A, Elbert T, Alewood PF, Gloriam DE, Gruber CW. Di Giglio MG, et al. Among authors: keov p. Sci Rep. 2017 Feb 1;7:41002. doi: 10.1038/srep41002. Sci Rep. 2017. PMID: 28145450 Free PMC article.

7

I8-arachnotocin-an arthropod-derived G protein-biased ligand of the human vasopressin V₂ receptor.

Duerrauer L, Muratspahić E, Gattringer J, Keov P, Mendel HC, Pfleger KDG, Muttenthaler M, Gruber CW. Duerrauer L, et al. Among authors: keov p. Sci Rep. 2019 Dec 17;9(1):19295. doi: 10.1038/s41598-019-55675-w. Sci Rep. 2019. PMID: 31848378 Free PMC article.

8

The TRPV4 Agonist GSK1016790A Regulates the Membrane Expression of TRPV4 Channels.

Baratchi S, Keov P, Darby WG, Lai A, Khoshmanesh K, Thurgood P, Vahidi P, Ejendal K, McIntyre P. Baratchi S, et al. Among authors: keov p. Front Pharmacol. 2019 Jan 23;10:6. doi: 10.3389/fphar.2019.00006. eCollection 2019. Front Pharmacol. 2019. PMID: 30728775 Free PMC article.

9

Cyclotides Isolated from an Ipecac Root Extract Antagonize the Corticotropin Releasing Factor Type 1 Receptor.

Fahradpour M, Keov P, Tognola C, Perez-Santamarina E, McCormick PJ, Ghassempour A, Gruber CW. Fahradpour M, et al. Among authors: keov p. Front Pharmacol. 2017 Sep 25;8:616. doi: 10.3389/fphar.2017.00616. eCollection 2017. Front Pharmacol. 2017. PMID: 29033832 Free PMC article.

10

Discovery of peptide probes to modulate oxytocin-type receptors of insects.

Keov P, Liutkevičiūtė Z, Hellinger R, Clark RJ, Gruber CW. Keov P, et al. Sci Rep. 2018 Jul 3;8(1):10020. doi: 10.1038/s41598-018-28380-3. Sci Rep. 2018. PMID: 29968789 Free PMC article.

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