Patel BA - Search Results

1

Design and synthesis of L- and D-phenylalanine derived rhodanines with novel C5-arylidenes as inhibitors of HCV NS5B polymerase.

Patel BA, Krishnan R, Khadtare N, Gurukumar KR, Basu A, Arora P, Bhatt A, Patel MR, Dana D, Kumar S, Kaushik-Basu N, Talele TT. Patel BA, et al. Among authors: patel mr. Bioorg Med Chem. 2013 Jun 1;21(11):3262-71. doi: 10.1016/j.bmc.2013.03.041. Epub 2013 Mar 31. Bioorg Med Chem. 2013. PMID: 23598249 Free PMC article.

2

The synthesis and SAR study of phenylalanine-derived (Z)-5-arylmethylidene rhodanines as anti-methicillin-resistant Staphylococcus aureus (MRSA) compounds.

Patel BA, Ashby CR Jr, Hardej D, Talele TT. Patel BA, et al. Bioorg Med Chem Lett. 2013 Oct 15;23(20):5523-7. doi: 10.1016/j.bmcl.2013.08.059. Epub 2013 Aug 20. Bioorg Med Chem Lett. 2013. PMID: 24012180

3

Design and synthesis of human ABCB1 (P-glycoprotein) inhibitors by peptide coupling of diverse chemical scaffolds on carboxyl and amino termini of (S)-valine-derived thiazole amino acid.

Singh S, Prasad NR, Chufan EE, Patel BA, Wang YJ, Chen ZS, Ambudkar SV, Talele TT. Singh S, et al. Among authors: patel ba. J Med Chem. 2014 May 22;57(10):4058-72. doi: 10.1021/jm401966m. Epub 2014 May 7. J Med Chem. 2014. PMID: 24773054 Free PMC article.

4

Novel 4-thiazolidinones as non-nucleoside inhibitors of hepatitis C virus NS5B RNA-dependent RNA polymerase.

Çakir G, Küçükgüzel İ, Guhamazumder R, Tatar E, Manvar D, Basu A, Patel BA, Zia J, Talele TT, Kaushik-Basu N. Çakir G, et al. Among authors: patel ba. Arch Pharm (Weinheim). 2015 Jan;348(1):10-22. doi: 10.1002/ardp.201400247. Epub 2014 Dec 2. Arch Pharm (Weinheim). 2015. PMID: 25449674

5

Dual inhibition of Staphylococcus aureus DNA gyrase and topoisomerase IV activity by phenylalanine-derived (Z)-5-arylmethylidene rhodanines.

Werner MM, Patel BA, Talele TT, Ashby CR, Li Z, Zauhar RJ. Werner MM, et al. Among authors: patel ba. Bioorg Med Chem. 2015 Sep 15;23(18):6125-37. doi: 10.1016/j.bmc.2015.08.004. Epub 2015 Aug 14. Bioorg Med Chem. 2015. PMID: 26320664

6

Comprehensive Synthesis of Amino Acid-Derived Thiazole Peptidomimetic Analogues to Understand the Enigmatic Drug/Substrate-Binding Site of P-Glycoprotein.

Patel BA, Abel B, Barbuti AM, Velagapudi UK, Chen ZS, Ambudkar SV, Talele TT. Patel BA, et al. J Med Chem. 2018 Feb 8;61(3):834-864. doi: 10.1021/acs.jmedchem.7b01340. Epub 2018 Jan 23. J Med Chem. 2018. PMID: 29251928 Free PMC article.

7

Design and Synthesis of Poly(ADP-ribose) Polymerase Inhibitors: Impact of Adenosine Pocket-Binding Motif Appendage to the 3-Oxo-2,3-dihydrobenzofuran-7-carboxamide on Potency and Selectivity.

Velagapudi UK, Langelier MF, Delgado-Martin C, Diolaiti ME, Bakker S, Ashworth A, Patel BA, Shao X, Pascal JM, Talele TT. Velagapudi UK, et al. Among authors: patel ba. J Med Chem. 2019 Jun 13;62(11):5330-5357. doi: 10.1021/acs.jmedchem.8b01709. Epub 2019 May 24. J Med Chem. 2019. PMID: 31042381 Free PMC article.

8

Design, synthesis, and biological evaluation of (S)-valine thiazole-derived cyclic and noncyclic peptidomimetic oligomers as modulators of human P-glycoprotein (ABCB1).

Singh S, Prasad NR, Kapoor K, Chufan EE, Patel BA, Ambudkar SV, Talele TT. Singh S, et al. Among authors: patel ba. Chembiochem. 2014 Jan 3;15(1):157-69. doi: 10.1002/cbic.201300565. Epub 2013 Nov 29. Chembiochem. 2014. PMID: 24288265 Free PMC article.

9

Recent development in the discovery of PARP inhibitors as anticancer agents: a patent update (2016-2020).

Velagapudi UK, Patel BA, Shao X, Pathak SK, Ferraris DV, Talele TT. Velagapudi UK, et al. Among authors: patel ba. Expert Opin Ther Pat. 2021 Jul;31(7):609-623. doi: 10.1080/13543776.2021.1886275. Epub 2021 Mar 12. Expert Opin Ther Pat. 2021. PMID: 33554679 Review.

10

Bafetinib (INNO-406) reverses multidrug resistance by inhibiting the efflux function of ABCB1 and ABCG2 transporters.

Zhang YK, Zhang GN, Wang YJ, Patel BA, Talele TT, Yang DH, Chen ZS. Zhang YK, et al. Among authors: patel ba. Sci Rep. 2016 May 9;6:25694. doi: 10.1038/srep25694. Sci Rep. 2016. PMID: 27157787 Free PMC article.

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