Nefzi A - Search Results

1

Striking reduction of amyloid plaque burden in an Alzheimer's mouse model after chronic administration of carmustine.

Hayes CD, Dey D, Palavicini JP, Wang H, Patkar KA, Minond D, Nefzi A, Lakshmana MK. Hayes CD, et al. Among authors: nefzi a. BMC Med. 2013 Mar 26;11:81. doi: 10.1186/1741-7015-11-81. BMC Med. 2013. PMID: 23531149 Free PMC article.

2

AlphaLISA-based high-throughput screening assay to measure levels of soluble amyloid precursor protein α.

Wang H, Nefzi A, Fields GB, Lakshmana MK, Minond D. Wang H, et al. Among authors: nefzi a. Anal Biochem. 2014 Aug 15;459:24-30. doi: 10.1016/j.ab.2014.05.007. Epub 2014 May 20. Anal Biochem. 2014. PMID: 24857774

3

Substituted dithiazole piperazine benzamides as novel amyloid beta peptide reducing agents.

Wang H, Wang R, Lakshmana MK, Nefzi A. Wang H, et al. Among authors: nefzi a. Bioorg Med Chem Lett. 2014 Sep 15;24(18):4384-4388. doi: 10.1016/j.bmcl.2014.08.022. Epub 2014 Aug 13. Bioorg Med Chem Lett. 2014. PMID: 25155386 Free PMC article.

4

Synthesis of dihydroimidazole tethered imidazolinethiones and their activity as novel antagonists of the nuclear retinoic acid receptor-related orphan receptors (RORs).

Nefzi A, Marconi GD, Ortiz MA, Davis JC, Piedrafita FJ. Nefzi A, et al. Bioorg Med Chem Lett. 2017 Apr 1;27(7):1608-1610. doi: 10.1016/j.bmcl.2017.02.014. Epub 2017 Feb 10. Bioorg Med Chem Lett. 2017. PMID: 28242276 Free PMC article.

5

Integrating virtual screening and combinatorial chemistry for accelerated drug discovery.

López-Vallejo F, Caulfield T, Martínez-Mayorga K, Giulianotti MA, Nefzi A, Houghten RA, Medina-Franco JL. López-Vallejo F, et al. Among authors: nefzi a. Comb Chem High Throughput Screen. 2011 Jul;14(6):475-87. doi: 10.2174/138620711795767866. Comb Chem High Throughput Screen. 2011. PMID: 21521151 Review.

6

Combinatorial Libraries As a Tool for the Discovery of Novel, Broad-Spectrum Antibacterial Agents Targeting the ESKAPE Pathogens.

Fleeman R, LaVoi TM, Santos RG, Morales A, Nefzi A, Welmaker GS, Medina-Franco JL, Giulianotti MA, Houghten RA, Shaw LN. Fleeman R, et al. Among authors: nefzi a. J Med Chem. 2015 Apr 23;58(8):3340-55. doi: 10.1021/jm501628s. Epub 2015 Apr 1. J Med Chem. 2015. PMID: 25780985 Free PMC article.

7

Increased diversity of libraries from libraries: chemoinformatic analysis of bis-diazacyclic libraries.

López-Vallejo F, Nefzi A, Bender A, Owen JR, Nabney IT, Houghten RA, Medina-Franco JL. López-Vallejo F, et al. Among authors: nefzi a. Chem Biol Drug Des. 2011 May;77(5):328-42. doi: 10.1111/j.1747-0285.2011.01100.x. Epub 2011 Mar 1. Chem Biol Drug Des. 2011. PMID: 21294850 Free PMC article.

8

Scaffold ranking and positional scanning utilized in the discovery of nAChR-selective compounds suitable for optimization studies.

Wu J, Zhang Y, Maida LE, Santos RG, Welmaker GS, LaVoi TM, Nefzi A, Yu Y, Houghten RA, Toll L, Giulianotti MA. Wu J, et al. Among authors: nefzi a. J Med Chem. 2013 Dec 27;56(24):10103-17. doi: 10.1021/jm401543h. Epub 2013 Dec 12. J Med Chem. 2013. PMID: 24274400 Free PMC article.

9

Direct Phenotypic Screening in Mice: Identification of Individual, Novel Antinociceptive Compounds from a Library of 734,821 Pyrrolidine Bis-piperazines.

Houghten RA, Ganno ML, McLaughlin JP, Dooley CT, Eans SO, Santos RG, LaVoi T, Nefzi A, Welmaker G, Giulianotti MA, Toll L. Houghten RA, et al. Among authors: nefzi a. ACS Comb Sci. 2016 Jan 11;18(1):51-64. doi: 10.1021/acscombsci.5b00126. Epub 2016 Jan 5. ACS Comb Sci. 2016. PMID: 26651386 Free PMC article.

10

Hantzsch based macrocyclization approach for the synthesis of thiazole containing cyclopeptides.

Nefzi A. Nefzi A. Methods Mol Biol. 2013;1081:1-11. doi: 10.1007/978-1-62703-652-8_1. Methods Mol Biol. 2013. PMID: 24014430

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

92 results

Search Page

Filters