Frédérick R - Search Results

1

New selective carbonic anhydrase IX inhibitors: synthesis and pharmacological evaluation of diarylpyrazole-benzenesulfonamides.

Rogez-Florent T, Meignan S, Foulon C, Six P, Gros A, Bal-Mahieu C, Supuran CT, Scozzafava A, Frédérick R, Masereel B, Depreux P, Lansiaux A, Goossens JF, Gluszok S, Goossens L. Rogez-Florent T, et al. Among authors: frederick r. Bioorg Med Chem. 2013 Mar 15;21(6):1451-64. doi: 10.1016/j.bmc.2012.10.029. Epub 2012 Oct 29. Bioorg Med Chem. 2013. PMID: 23168081

2

Coumarin and isocoumarin as serine protease inhibitors.

Pochet L, Frédérick R, Masereel B. Pochet L, et al. Among authors: frederick r. Curr Pharm Des. 2004;10(30):3781-96. doi: 10.2174/1381612043382684. Curr Pharm Des. 2004. PMID: 15579071 Review.

3

Modulators of the coagulation cascade: focus and recent advances in inhibitors of tissue factor, factor VIIa and their complex.

Frédérick R, Pochet L, Charlier C, Masereel B. Frédérick R, et al. Curr Med Chem. 2005;12(4):397-417. doi: 10.2174/0929867053363108. Curr Med Chem. 2005. PMID: 15720249 Review.

4

3,6-disubstituted coumarins as mechanism-based inhibitors of thrombin and factor Xa.

Frédérick R, Robert S, Charlier C, de Ruyck J, Wouters J, Pirotte B, Masereel B, Pochet L. Frédérick R, et al. J Med Chem. 2005 Dec 1;48(24):7592-603. doi: 10.1021/jm050448g. J Med Chem. 2005. PMID: 16302799

5

Investigation of mechanism-based thrombin inhibitors: Implications of a highly conserved water molecule for the binding of coumarins within the S pocket.

Frédérick R, Charlier C, Robert S, Wouters J, Masereel B, Pochet L. Frédérick R, et al. Bioorg Med Chem Lett. 2006 Apr 1;16(7):2017-21. doi: 10.1016/j.bmcl.2005.12.070. Epub 2006 Jan 18. Bioorg Med Chem Lett. 2006. PMID: 16413781

6

Mechanism-based thrombin inhibitors: design, synthesis, and molecular docking of a new selective 2-oxo-2H-1-benzopyran derivative.

Frédérick R, Robert S, Charlier C, Wouters J, Masereel B, Pochet L. Frédérick R, et al. J Med Chem. 2007 Jul 26;50(15):3645-50. doi: 10.1021/jm061368v. Epub 2007 Jun 20. J Med Chem. 2007. PMID: 17580844

7

Synthesis, biological evaluation and molecular modelling of sulfonohydrazides as selective PI3K p110alpha inhibitors.

Kendall JD, Rewcastle GW, Frederick R, Mawson C, Denny WA, Marshall ES, Baguley BC, Chaussade C, Jackson SP, Shepherd PR. Kendall JD, et al. Among authors: frederick r. Bioorg Med Chem. 2007 Dec 15;15(24):7677-87. doi: 10.1016/j.bmc.2007.08.062. Epub 2007 Sep 4. Bioorg Med Chem. 2007. PMID: 17869522

8

Ligand-based and structure-based virtual screening to identify carbonic anhydrase IX inhibitors.

Thiry A, Ledecq M, Cecchi A, Frederick R, Dogné JM, Supuran CT, Wouters J, Masereel B. Thiry A, et al. Among authors: frederick r. Bioorg Med Chem. 2009 Jan 15;17(2):553-7. doi: 10.1016/j.bmc.2008.11.071. Epub 2008 Dec 6. Bioorg Med Chem. 2009. PMID: 19097911

9

Pyrazolo[4,3-c]isoquinolines as potential inhibitors of NF-kappaB activation.

Mortier J, Frederick R, Ganeff C, Remouchamps C, Talaga P, Pochet L, Wouters J, Piette J, Dejardin E, Masereel B. Mortier J, et al. Among authors: frederick r. Biochem Pharmacol. 2010 May 15;79(10):1462-72. doi: 10.1016/j.bcp.2010.01.007. Epub 2010 Jan 21. Biochem Pharmacol. 2010. PMID: 20096267

10

NF-kappaB inducing kinase (NIK) inhibitors: identification of new scaffolds using virtual screening.

Mortier J, Masereel B, Remouchamps C, Ganeff C, Piette J, Frederick R. Mortier J, et al. Among authors: frederick r. Bioorg Med Chem Lett. 2010 Aug 1;20(15):4515-20. doi: 10.1016/j.bmcl.2010.06.027. Epub 2010 Jun 8. Bioorg Med Chem Lett. 2010. PMID: 20580552

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