El Kazzouli S - Search Results

1

N-methyl-substituted fluorescent DAG-indololactone isomers exhibit dramatic differences in membrane interactions and biological activity.

Gal N, Kolusheva S, Kedei N, Telek A, Naeem TA, Lewin NE, Lim L, Mannan P, Garfield SH, El Kazzouli S, Sigano DM, Marquez VE, Blumberg PM, Jelinek R. Gal N, et al. Among authors: el kazzouli s. Chembiochem. 2011 Oct 17;12(15):2331-40. doi: 10.1002/cbic.201100246. Chembiochem. 2011. PMID: 23106081 Free PMC article.

2

Membrane-surface anchoring of charged diacylglycerol-lactones correlates with biological activities.

Raifman O, Kolusheva S, El Kazzouli S, Sigano DM, Kedei N, Lewin NE, Lopez-Nicolas R, Ortiz-Espin A, Gomez-Fernandez JC, Blumberg PM, Marquez VE, Corbalan-Garcia S, Jelinek R. Raifman O, et al. Among authors: el kazzouli s. Chembiochem. 2010 Sep 24;11(14):2003-9. doi: 10.1002/cbic.201000343. Chembiochem. 2010. PMID: 20715268 Free PMC article.

3

Conformationally constrained analogues of diacylglycerol. 30. An investigation of diacylglycerol-lactones containing heteroaryl groups reveals compounds with high selectivity for Ras guanyl nucleotide-releasing proteins.

El Kazzouli S, Lewin NE, Blumberg PM, Marquez VE. El Kazzouli S, et al. J Med Chem. 2008 Sep 11;51(17):5371-86. doi: 10.1021/jm800380b. Epub 2008 Aug 16. J Med Chem. 2008. PMID: 18707088 Free PMC article.

4

Conformationally constrained analogues of diacylglycerol. 29. Cells sort diacylglycerol-lactone chemical zip codes to produce diverse and selective biological activities.

Duan D, Sigano DM, Kelley JA, Lai CC, Lewin NE, Kedei N, Peach ML, Lee J, Abeyweera TP, Rotenberg SA, Kim H, Kim YH, El Kazzouli S, Chung JU, Young HA, Young MR, Baker A, Colburn NH, Haimovitz-Friedman A, Truman JP, Parrish DA, Deschamps JR, Perry NA, Surawski RJ, Blumberg PM, Marquez VE. Duan D, et al. Among authors: el kazzouli s. J Med Chem. 2008 Sep 11;51(17):5198-220. doi: 10.1021/jm8001907. Epub 2008 Aug 13. J Med Chem. 2008. PMID: 18698758 Free PMC article.

5

Molecular basis for failure of "atypical" C1 domain of Vav1 to bind diacylglycerol/phorbol ester.

Geczy T, Peach ML, El Kazzouli S, Sigano DM, Kang JH, Valle CJ, Selezneva J, Woo W, Kedei N, Lewin NE, Garfield SH, Lim L, Mannan P, Marquez VE, Blumberg PM. Geczy T, et al. Among authors: el kazzouli s. J Biol Chem. 2012 Apr 13;287(16):13137-58. doi: 10.1074/jbc.M111.320010. Epub 2012 Feb 18. J Biol Chem. 2012. PMID: 22351766 Free PMC article.

6

Synthesis and biological evaluation of N-(7-indazolyl)benzenesulfonamide derivatives as potent cell cycle inhibitors.

Bouissane L, El Kazzouli S, Léonce S, Pfeiffer B, Rakib EM, Khouili M, Guillaumet G. Bouissane L, et al. Among authors: el kazzouli s. Bioorg Med Chem. 2006 Feb 15;14(4):1078-88. doi: 10.1016/j.bmc.2005.09.037. Epub 2005 Nov 7. Bioorg Med Chem. 2006. PMID: 16274996

7

Design and synthesis of 2-phenylimidazo[1,2-a]pyridines as a novel class of melatonin receptor ligands.

El Kazzouli S, Griffon du Bellay A, Berteina-Raboin S, Delagrange P, Caignard DH, Guillaumet G. El Kazzouli S, et al. Eur J Med Chem. 2011 Sep;46(9):4252-7. doi: 10.1016/j.ejmech.2011.06.030. Epub 2011 Jul 1. Eur J Med Chem. 2011. PMID: 21764185

8

Synthesis and biological evaluation of ethacrynic acid derivatives bearing sulfonamides as potent anti-cancer agents.

El Abbouchi A, El Brahmi N, Hiebel MA, Bignon J, Guillaumet G, Suzenet F, El Kazzouli S. El Abbouchi A, et al. Among authors: el brahmi n, el kazzouli s. Bioorg Med Chem Lett. 2020 Oct 1;30(19):127426. doi: 10.1016/j.bmcl.2020.127426. Epub 2020 Aug 2. Bioorg Med Chem Lett. 2020. PMID: 32755677

9

Synthesis of polysubstituted imidazo[1,2-a]pyridines via microwave-assisted one-pot cyclization/Suzuki coupling/palladium-catalyzed heteroarylation.

Koubachi J, El Kazzouli S, Berteina-Raboin S, Mouaddib A, Guillaumet G. Koubachi J, et al. Among authors: el kazzouli s. J Org Chem. 2007 Sep 28;72(20):7650-5. doi: 10.1021/jo0712603. Epub 2007 Sep 5. J Org Chem. 2007. PMID: 17784775

10

Palladium-Catalyzed C3-Arylations of 1 H- and 2 H-Pyrazolo[4,3- b]pyridines on Water.

Faarasse S, El Kazzouli S, Suzenet F, Guillaumet G. Faarasse S, et al. Among authors: el kazzouli s. J Org Chem. 2018 Oct 19;83(20):12847-12854. doi: 10.1021/acs.joc.8b01728. Epub 2018 Oct 4. J Org Chem. 2018. PMID: 30240222

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

40 results

Search Page

Filters