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Targeting the DNA-binding activity of the human ERG transcription factor using new heterocyclic dithiophene diamidines.
Nhili R, Peixoto P, Depauw S, Flajollet S, Dezitter X, Munde MM, Ismail MA, Kumar A, Farahat AA, Stephens CE, Duterque-Coquillaud M, David Wilson W, Boykin DW, David-Cordonnier MH. Nhili R, et al. Among authors: peixoto p. Nucleic Acids Res. 2013 Jan 7;41(1):125-38. doi: 10.1093/nar/gks971. Epub 2012 Oct 23. Nucleic Acids Res. 2013. PMID: 23093599 Free PMC article.
Heterocyclic Diamidine DNA Ligands as HOXA9 Transcription Factor Inhibitors: Design, Molecular Evaluation, and Cellular Consequences in a HOXA9-Dependant Leukemia Cell Model.
Depauw S, Lambert M, Jambon S, Paul A, Peixoto P, Nhili R, Marongiu L, Figeac M, Dassi C, Paul-Constant C, Billoré B, Kumar A, Farahat AA, Ismail MA, Mineva E, Sweat DP, Stephens CE, Boykin DW, Wilson WD, David-Cordonnier MH. Depauw S, et al. Among authors: peixoto p. J Med Chem. 2019 Feb 14;62(3):1306-1329. doi: 10.1021/acs.jmedchem.8b01448. Epub 2019 Feb 1. J Med Chem. 2019. PMID: 30645099 Free PMC article.
The unusual monomer recognition of guanine-containing mixed sequence DNA by a dithiophene heterocyclic diamidine.
Munde M, Kumar A, Peixoto P, Depauw S, Ismail MA, Farahat AA, Paul A, Say MV, David-Cordonnier MH, Boykin DW, Wilson WD. Munde M, et al. Among authors: peixoto p. Biochemistry. 2014 Feb 25;53(7):1218-27. doi: 10.1021/bi401582t. Epub 2014 Feb 13. Biochemistry. 2014. PMID: 24495039 Free PMC article.
DB1255 is a symmetrical diamidinophenyl-dithiophene that exhibits cellular activity by binding to DNA and inhibiting binding of ERG, an ETS family transcription factor that is commonly overexpressed or translocated in leukemia and prostate cancer [Nhili, R., Peixoto, P …
DB1255 is a symmetrical diamidinophenyl-dithiophene that exhibits cellular activity by binding to DNA and inhibiting binding of ERG, an ETS …
Novel diamidino-substituted derivatives of phenyl benzothiazolyl and dibenzothiazolyl furans and thiophenes: synthesis, antiproliferative and DNA binding properties.
Racané L, Tralić-Kulenović V, Kraljević Pavelić S, Ratkaj I, Peixoto P, Nhili R, Depauw S, Hildebrand MP, David-Cordonnier MH, Pavelić K, Karminski-Zamola G. Racané L, et al. Among authors: peixoto p. J Med Chem. 2010 Mar 25;53(6):2418-32. doi: 10.1021/jm901441b. J Med Chem. 2010. PMID: 20170096
Unusual cellular uptake of cytotoxic 4-hydroxymethyl-3-aminoacridine.
Peixoto P, Zeghida W, Carrez D, Wu TD, Wattez N, Croisy A, Demeunynck M, Guerquin-Kern JL, Lansiaux A. Peixoto P, et al. Eur J Med Chem. 2009 Nov;44(11):4758-63. doi: 10.1016/j.ejmech.2009.06.034. Epub 2009 Jul 4. Eur J Med Chem. 2009. PMID: 19640614
239 results