Déprez B - Search Results

1

Discovery of novel N-phenylphenoxyacetamide derivatives as EthR inhibitors and ethionamide boosters by combining high-throughput screening and synthesis.

Flipo M, Willand N, Lecat-Guillet N, Hounsou C, Desroses M, Leroux F, Lens Z, Villeret V, Wohlkönig A, Wintjens R, Christophe T, Kyoung Jeon H, Locht C, Brodin P, Baulard AR, Déprez B. Flipo M, et al. Among authors: deprez b. J Med Chem. 2012 Jul 26;55(14):6391-402. doi: 10.1021/jm300377g. Epub 2012 Jul 17. J Med Chem. 2012. PMID: 22738293

2

Automated parallel synthesis of a tetrahydroisoquinolin-based library: potential prolyl endopeptidase inhibitors.

Vendeville S, Bourel L, Davioud-Charvet E, Grellier P, Deprez B, Sergheraert C. Vendeville S, et al. Among authors: deprez b. Bioorg Med Chem Lett. 1999 Feb 8;9(3):437-42. doi: 10.1016/s0960-894x(99)00003-7. Bioorg Med Chem Lett. 1999. PMID: 10091698

3

Parallel synthesis of a library of 1,4-naphthoquinones and automated screening of potential inhibitors of trypanothione reductase from Trypanosoma cruzi.

Salmon-Chemin L, Lemaire A, De Freitas S, Deprez B, Sergheraert C, Davioud-Charvet E. Salmon-Chemin L, et al. Among authors: deprez b. Bioorg Med Chem Lett. 2000 Apr 3;10(7):631-5. doi: 10.1016/s0960-894x(00)00056-1. Bioorg Med Chem Lett. 2000. PMID: 10762041

4

From hit to lead. Combining two complementary methods for focused library design. Application to mu opiate ligands.

Poulain R, Horvath D, Bonnet B, Eckhoff C, Chapelain B, Bodinier MC, Déprez B. Poulain R, et al. Among authors: deprez b. J Med Chem. 2001 Oct 11;44(21):3378-90. doi: 10.1021/jm010877o. J Med Chem. 2001. PMID: 11585443

5

From hit to lead. Analyzing structure-profile relationships.

Poulain R, Horvath D, Bonnet B, Eckhoff C, Chapelain B, Bodinier MC, Déprez B. Poulain R, et al. Among authors: deprez b. J Med Chem. 2001 Oct 11;44(21):3391-401. doi: 10.1021/jm010878g. J Med Chem. 2001. PMID: 11585444

6

Control of protein-protein interactions: structure-based discovery of low molecular weight inhibitors of the interactions between Pin1 WW domain and phosphopeptides.

Smet C, Duckert JF, Wieruszeski JM, Landrieu I, Buée L, Lippens G, Déprez B. Smet C, et al. Among authors: deprez b. J Med Chem. 2005 Jul 28;48(15):4815-23. doi: 10.1021/jm0500119. J Med Chem. 2005. PMID: 16033261

7

A library of novel hydroxamic acids targeting the metallo-protease family: design, parallel synthesis and screening.

Flipo M, Beghyn T, Charton J, Leroux VA, Deprez BP, Deprez-Poulain RF. Flipo M, et al. Bioorg Med Chem. 2007 Jan 1;15(1):63-76. doi: 10.1016/j.bmc.2006.10.010. Epub 2006 Oct 12. Bioorg Med Chem. 2007. PMID: 17070058

8

PDE5 inhibitors: An original access to novel potent arylated analogues of tadalafil.

Beghyn T, Hounsou C, Deprez BP. Beghyn T, et al. Bioorg Med Chem Lett. 2007 Feb 1;17(3):789-92. doi: 10.1016/j.bmcl.2006.10.069. Epub 2006 Oct 27. Bioorg Med Chem Lett. 2007. PMID: 17107795

9

Novel selective inhibitors of the zinc plasmodial aminopeptidase PfA-M1 as potential antimalarial agents.

Flipo M, Beghyn T, Leroux V, Florent I, Deprez BP, Deprez-Poulain RF. Flipo M, et al. J Med Chem. 2007 Mar 22;50(6):1322-34. doi: 10.1021/jm061169b. Epub 2007 Feb 28. J Med Chem. 2007. PMID: 17326615

10

Natural compounds: leads or ideas? Bioinspired molecules for drug discovery.

Beghyn T, Deprez-Poulain R, Willand N, Folleas B, Deprez B. Beghyn T, et al. Among authors: deprez poulain r, deprez b. Chem Biol Drug Des. 2008 Jul;72(1):3-15. doi: 10.1111/j.1747-0285.2008.00673.x. Epub 2008 Jun 11. Chem Biol Drug Des. 2008. PMID: 18554253

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